Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Giardia lamblia | Beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Toxoplasma gondii | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0094 | 0.2612 | 0.2612 |
Trypanosoma brucei | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0094 | 0.2612 | 0.2612 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0094 | 0.2612 | 0.2612 |
Schistosoma mansoni | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Trypanosoma brucei | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Loa Loa (eye worm) | tubulin beta chain | 0.0094 | 0.2612 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Loa Loa (eye worm) | beta-tubulin | 0.0094 | 0.2612 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0094 | 0.2612 | 0.5 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0094 | 0.2612 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0094 | 0.2612 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Entamoeba histolytica | tubulin family protein | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0094 | 0.2612 | 0.2612 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0094 | 0.2612 | 1 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Brugia malayi | Tubulin beta-1 chain | 0.0094 | 0.2612 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0094 | 0.2612 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0094 | 0.2612 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Echinococcus granulosus | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0094 | 0.2612 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0094 | 0.2612 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0094 | 0.2612 | 0.2612 |
Echinococcus multilocularis | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Loa Loa (eye worm) | BEN-1 protein | 0.0094 | 0.2612 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Trichomonas vaginalis | tubulin, putative | 0.0094 | 0.2612 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0094 | 0.2612 | 1 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0094 | 0.2612 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0094 | 0.2612 | 0.2612 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Plasmodium vivax | tubulin beta chain, putative | 0.0094 | 0.2612 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0094 | 0.2612 | 0.2612 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0094 | 0.2612 | 0.2612 |
Entamoeba histolytica | tubulin family protein | 0.0094 | 0.2612 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0094 | 0.2612 | 0.2612 |
Schistosoma mansoni | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Leishmania major | beta tubulin | 0.0094 | 0.2612 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0094 | 0.2612 | 0.2612 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0094 | 0.2612 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 438 uM | Inhibition of HDAC in human HeLa cell extract by fluorescence plate reader assay | ChEMBL. | 16921367 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.