Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Trypanosoma brucei | phosphoglycerate kinase | Starlite/ChEMBL | No references |
Trypanosoma brucei gambiense | phosphoglycerate kinase, putative | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Toxoplasma gondii | phosphoglycerate kinase PGKI | 0.0206 | 0.5 | 0.5 |
Echinococcus multilocularis | phosphoglycerate kinase 1 | 0.0206 | 0.5 | 0.5 |
Treponema pallidum | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Mycobacterium ulcerans | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Plasmodium vivax | phosphoglycerate kinase, putative | 0.0206 | 0.5 | 0.5 |
Toxoplasma gondii | phosphoglycerate kinase PGKII | 0.0206 | 0.5 | 0.5 |
Schistosoma mansoni | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Schistosoma mansoni | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Trypanosoma brucei | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Echinococcus granulosus | phosphoglycerate kinase 1 | 0.0206 | 0.5 | 0.5 |
Trypanosoma cruzi | phosphoglycerate kinase, putative | 0.0206 | 0.5 | 0.5 |
Plasmodium falciparum | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0206 | 0.5 | 0.5 |
Entamoeba histolytica | phosphoglycerate kinase, putative | 0.0206 | 0.5 | 0.5 |
Trichomonas vaginalis | phosphoglycerate kinase, putative | 0.0206 | 0.5 | 0.5 |
Chlamydia trachomatis | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Trichomonas vaginalis | phosphoglycerate kinase, putative | 0.0206 | 0.5 | 0.5 |
Mycobacterium tuberculosis | Probable phosphoglycerate kinase Pgk | 0.0206 | 0.5 | 0.5 |
Trypanosoma brucei | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Mycobacterium leprae | Probable phosphoglycerate kinase Pgk | 0.0206 | 0.5 | 0.5 |
Trypanosoma cruzi | phosphoglycerate kinase, putative | 0.0206 | 0.5 | 0.5 |
Leishmania major | phosphoglycerate kinase C, glycosomal | 0.0206 | 0.5 | 0.5 |
Leishmania major | phosphoglycerate kinase B, cytosolic | 0.0206 | 0.5 | 0.5 |
Wolbachia endosymbiont of Brugia malayi | phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Giardia lamblia | Phosphoglycerate kinase | 0.0206 | 0.5 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | 10 uM | PUBCHEM_BIOASSAY: qHTS Assay to Find Inhibitors of Phosphoglycerate Kinase. (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | 13.1154 uM | PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488745, AID488752, AID488774, AID504848, AID504850] | ChEMBL. | No reference |
Potency (functional) | = 28.1838 um | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E). (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | 35.4813 uM | PUBCHEM_BIOASSAY: qHTS for Inhibitors of binding or entry into cells for Lassa Virus. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID463114, AID540249] | ChEMBL. | No reference |
Potency (functional) | 89.1251 uM | PUBCHEM_BIOASSAY: qHTS for Inhibitors of Polymerase Iota. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID588623] | ChEMBL. | No reference |
Species name | Source | Reference | Is orphan |
---|---|---|---|
Plasmodium falciparum | ChEMBL23 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.