TDR Targets

Basic information

Technical information

TDR Targets ID: 1407505
Name: N-(4,5-dihydro-1,3-thiazol-2-yl)-7-methyl-[1, 2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
MW: 262.291 | Formula: C10H10N6OS
H donors: 1 H acceptors: 4 LogP: 0.52 Rotable bonds: 3
Rule of 5 violations (Lipinski): 1
SMILES: O=C(c1nn2c(n1)nccc2C)NC1=NCCS1
InChi: 1S/C10H10N6OS/c1-6-2-3-11-9-13-7(15-16(6)9)8(17)14-10-12-4-5-18-10/h2-3H,4-5H2,1H3,(H,12,14,17)
InChiKey: ORNPFKPINMNCGQ-UHFFFAOYSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

N-(4,5-dihydrothiazol-2-yl)-7-methyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
MLS000054852
SMR000066789
ZINC02648582

Targets

Known targets for this compound

No curated genes were found associated with this compound

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

No druggable targets predicted by sequence similarity

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0092	0.1136	0.0606
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Schistosoma mansoni	cathepsin F (C01 family)	0.012	0.2085	0.2088
Entamoeba histolytica	cysteine proteinase, putative	0.0179	0.4119	1
Schistosoma mansoni	calpain (C02 family)	0.0124	0.2223	0.2226
Plasmodium falciparum	cysteine proteinase falcipain 2a	0.0179	0.4119	1
Trypanosoma cruzi	cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.5396
Trypanosoma cruzi	kinesin, putative	0.0087	0.0943	0.2289
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Trypanosoma cruzi	cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.5396
Schistosoma mansoni	calpain-7 (C02 family)	0.0124	0.2223	0.2226
Plasmodium vivax	vivapain-1	0.0092	0.1136	0.2757
Onchocerca volvulus		0.0179	0.4119	0.6993
Toxoplasma gondii	cathepsin CPL	0.0179	0.4119	0.5
Trypanosoma brucei	antigen, putative	0.0124	0.2223	0.4029
Echinococcus multilocularis	hypothetical protein	0.0124	0.2223	0.1227
Brugia malayi	calpain 7	0.0124	0.2223	0.2403
Trypanosoma cruzi	calpain-like cysteine peptidase, putative	0.0124	0.2223	0.5396
Echinococcus granulosus	family C2 unassigned peptidase C02 family	0.035	0.9984	0.9982
Schistosoma mansoni	cathepsin F (C01 family)	0.0179	0.4119	0.4126
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Brugia malayi	Cathepsin L-like precursor	0.0179	0.4119	0.4453
Loa Loa (eye worm)	hypothetical protein	0.0179	0.4119	0.4453
Echinococcus granulosus	cathepsin l cysteine peptidase	0.0179	0.4119	0.3366
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0092	0.1136	0.0606
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Trypanosoma cruzi	calpain-like cysteine peptidase, putative	0.0124	0.2223	0.5396
Entamoeba histolytica	cysteine proteinase, putative	0.0092	0.1136	0.0606
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Trypanosoma brucei	calpain-like protein, putative	0.0124	0.2223	0.4029
Loa Loa (eye worm)	hypothetical protein	0.012	0.2085	0.2254
Schistosoma mansoni	SmCL2-like peptidase (C01 family)	0.0092	0.1136	0.1137
Trypanosoma cruzi	cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.5396
Trypanosoma cruzi	kinesin, putative	0.0087	0.0943	0.2289
Echinococcus granulosus	calpain 5	0.0124	0.2223	0.1227
Echinococcus granulosus	calpain 7 C02 family	0.0124	0.2223	0.1227
Leishmania major	calpain-like cysteine peptidase, putative,cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.4029
Onchocerca volvulus	Cathepsin F homolog	0.0179	0.4119	0.6993
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Trypanosoma cruzi	calpain-like cysteine peptidase, putative	0.0124	0.2223	0.5396
Entamoeba histolytica	cysteine proteinase, putative	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Echinococcus multilocularis	calpain family protein 1, d	0.0242	0.6274	0.5797
Plasmodium vivax	vivapain-3	0.0092	0.1136	0.2757
Echinococcus granulosus	calpain A	0.0124	0.2223	0.1227
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Loa Loa (eye worm)	hypothetical protein	0.0329	0.9252	1
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Brugia malayi	Cathepsin L-like precursor	0.0179	0.4119	0.4453
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Echinococcus multilocularis	calpain	0.0124	0.2223	0.1227
Trypanosoma cruzi	calpain-like cysteine peptidase, putative	0.0124	0.2223	0.5396
Loa Loa (eye worm)	hypothetical protein	0.012	0.2085	0.2254
Trypanosoma brucei	calpain-like protein, putative	0.0124	0.2223	0.4029
Schistosoma mansoni	calpain C (C02 family)	0.0124	0.2223	0.2226
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Trypanosoma cruzi	cysteine protease, putative	0.0092	0.1136	0.2757
Schistosoma mansoni	SmCL2-like peptidase (C01 family)	0.0092	0.1136	0.1137
Echinococcus granulosus	cathepsin L cysteine proteinase	0.0179	0.4119	0.3366
Trypanosoma cruzi	cysteine peptidase, putative	0.0092	0.1136	0.2757
Entamoeba histolytica	cysteine proteinase 2	0.0092	0.1136	0.0606
Echinococcus multilocularis	cathepsin L cysteine protease	0.0179	0.4119	0.3366
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Schistosoma mansoni	family C2 unassigned peptidase (C02 family)	0.035	0.9984	1
Schistosoma mansoni	calpain-7 (C02 family)	0.0124	0.2223	0.2226
Loa Loa (eye worm)	cysteine protease	0.0179	0.4119	0.4453
Plasmodium vivax	unspecified product	0.0092	0.1136	0.2757
Brugia malayi	Cathepsin L-like precursor	0.012	0.2085	0.2254
Trypanosoma cruzi	cysteine proteinase, putative	0.0092	0.1136	0.2757
Loa Loa (eye worm)	papain family cysteine protease containing protein	0.0179	0.4119	0.4453
Trichomonas vaginalis	Clan CA, family C1, cathepsin L or K-like cysteine peptidase	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Loa Loa (eye worm)	hypothetical protein	0.0242	0.6274	0.6782
Plasmodium vivax	vivapain-2	0.0179	0.4119	1
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Brugia malayi	calpain 5	0.0087	0.0943	0.1019
Entamoeba histolytica	cysteine proteinase, putative	0.0092	0.1136	0.0606
Trypanosoma cruzi	cysteine peptidase, putative	0.0179	0.4119	1
Entamoeba histolytica	cysteine proteinase, putative	0.0092	0.1136	0.0606
Onchocerca volvulus		0.0205	0.4994	1
Brugia malayi	Cathepsin L-like precursor	0.012	0.2085	0.2254
Onchocerca volvulus	Cathepsin L homolog	0.0179	0.4119	0.6993
Onchocerca volvulus		0.0179	0.4119	0.6993
Trypanosoma brucei	cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.4029
Loa Loa (eye worm)	calpain 5	0.0087	0.0943	0.1019
Schistosoma mansoni	family C2 unassigned peptidase (C02 family)	0.0329	0.9252	0.9266
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Trypanosoma cruzi	calpain cysteine peptidase, putative	0.0124	0.2223	0.5396
Trypanosoma cruzi	cysteine peptidase, putative	0.0179	0.4119	1
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Schistosoma mansoni	SmCL2-like peptidase (C01 family)	0.0092	0.1136	0.1137
Entamoeba histolytica	cysteine proteinase, putative	0.0092	0.1136	0.0606
Trypanosoma cruzi	cysteine proteinase, putative	0.0092	0.1136	0.2757
Entamoeba histolytica	cysteine proteinase, putative	0.012	0.2085	0.3595
Entamoeba histolytica	cysteine proteinase 1, putative	0.0092	0.1136	0.0606
Entamoeba histolytica	cysteine protease, putative	0.0179	0.4119	1
Brugia malayi	Cathepsin L-like precursor	0.0179	0.4119	0.4453
Brugia malayi	Papain family cysteine protease containing protein	0.0092	0.1136	0.1227
Trypanosoma cruzi	cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.5396
Plasmodium falciparum	cysteine proteinase falcipain 3	0.0179	0.4119	1
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Schistosoma mansoni	Mername-AA248 (C02 family)	0.0124	0.2223	0.2226
Echinococcus multilocularis	calpain 5	0.0124	0.2223	0.1227
Loa Loa (eye worm)	calpain	0.0124	0.2223	0.2403
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Brugia malayi	Papain family cysteine protease containing protein	0.0092	0.1136	0.1227
Brugia malayi	Cathepsin L-like precursor	0.0179	0.4119	0.4453
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Brugia malayi	Cathepsin L-like precursor	0.0179	0.4119	0.4453
Trypanosoma brucei	calpain-like protein, putative	0.0124	0.2223	0.4029
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Plasmodium vivax	calpain, putative	0.0124	0.2223	0.5396
Echinococcus granulosus	cathepsin l1	0.0179	0.4119	0.3366
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Plasmodium falciparum	cysteine proteinase falcipain 2b	0.0179	0.4119	1
Leishmania major	cysteine peptidase A (CPA)	0.0179	0.4119	1
Brugia malayi	cathepsin L-like precursor	0.012	0.2085	0.2254
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Loa Loa (eye worm)	ctsf protein	0.0179	0.4119	0.4453
Onchocerca volvulus		0.0179	0.4119	0.6993
Echinococcus multilocularis	cysteine protease	0.0179	0.4119	0.3366
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Brugia malayi	Cathepsin L-like precursor	0.0179	0.4119	0.4453
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Echinococcus multilocularis	cathepsin l cysteine peptidase	0.0179	0.4119	0.3366
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Schistosoma mansoni	family C2 unassigned peptidase (C02 family)	0.035	0.9984	1
Echinococcus multilocularis	cysteine protease	0.0179	0.4119	0.3366
Loa Loa (eye worm)	hypothetical protein	0.0291	0.7972	0.8617
Onchocerca volvulus		0.0179	0.4119	0.6993
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.012	0.2085	0.3182
Echinococcus granulosus	cathepsin l1	0.012	0.2085	0.1071
Echinococcus granulosus	calpain	0.0124	0.2223	0.1227
Loa Loa (eye worm)	calpain family protein 1	0.0329	0.9252	1
Trypanosoma cruzi	cruzipain precursor, putative	0.0179	0.4119	1
Onchocerca volvulus		0.0179	0.4119	0.6993
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Echinococcus multilocularis	calpain 7 (C02 family)	0.0124	0.2223	0.1227
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Trichomonas vaginalis	Clan CA, family C1, papain-like cysteine peptidase	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Onchocerca volvulus	Cathepsin L homolog	0.0179	0.4119	0.6993
Brugia malayi	Cathepsin L-like cysteine proteinase	0.012	0.2085	0.2254
Leishmania major	calpain-like cysteine peptidase, putative,cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.4029
Echinococcus multilocularis	cathepsin l cysteine peptidase	0.0179	0.4119	0.3366
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Trypanosoma cruzi	calpain-like cysteine peptidase, putative	0.0124	0.2223	0.5396
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Trypanosoma cruzi	cysteine peptidase, clan CA, family C1, cathepsin L-like, putative	0.012	0.2085	0.5061
Trypanosoma brucei	calpain-like protein, putative	0.0124	0.2223	0.4029
Loa Loa (eye worm)	calpain family protein 1	0.0242	0.6274	0.6782
Loa Loa (eye worm)	Papain cysteine protease/cathepsin propeptide inhibitor-containing protein	0.0179	0.4119	0.4453
Trichomonas vaginalis	Clan CA, family C1, cathepsin L or K-like cysteine peptidase	0.0179	0.4119	1
Schistosoma mansoni	cathepsin F (C01 family)	0.0179	0.4119	0.4126
Brugia malayi	calpain family protein 1	0.0329	0.9252	1
Trypanosoma brucei	cysteine peptidase, Clan CA, family C1, Cathepsin L-like	0.0179	0.4119	1
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Onchocerca volvulus		0.0179	0.4119	0.6993
Brugia malayi	calpain family protein 1	0.0329	0.9252	1
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Echinococcus multilocularis	family C2 unassigned peptidase (C02 family)	0.035	0.9984	0.9982
Loa Loa (eye worm)	fibroinase	0.0179	0.4119	0.4453
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.012	0.2085	0.3182
Onchocerca volvulus		0.0179	0.4119	0.6993
Leishmania major	cathepsin L-like protease	0.0179	0.4119	1
Trypanosoma brucei	calpain-like cysteine peptidase, putative	0.0124	0.2223	0.4029
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Loa Loa (eye worm)	hypothetical protein	0.012	0.2085	0.2254
Trichomonas vaginalis	Clan CA, family C1, cathepsin L-like cysteine peptidase	0.0179	0.4119	1
Echinococcus multilocularis	cathepsin L cysteine protease	0.0179	0.4119	0.3366
Leishmania major	calpain, putative,cysteine peptidase, Clan CA, family C2, putative	0.0124	0.2223	0.4029
Trypanosoma cruzi	cysteine peptidase (N-terminal), putative	0.0092	0.1136	0.2757
Brugia malayi	Papain family cysteine protease containing protein	0.0179	0.4119	0.4453
Loa Loa (eye worm)	hypothetical protein	0.0205	0.4994	0.5398
Entamoeba histolytica	cysteine protease, putative	0.0092	0.1136	0.0606
Plasmodium vivax	vivapain-2	0.0179	0.4119	1
Trypanosoma cruzi	cysteine peptidase, putative	0.0179	0.4119	1
Trypanosoma cruzi	cysteine peptidase, putative	0.0179	0.4119	1

Activities

Activity type	Activity value	Assay description	Source	Reference
Potency (functional)	6.3096 uM	PUBCHEM_BIOASSAY: qHTS for Inhibitors of TGF-b: Cytotox Counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID588855, AID588860]	ChEMBL.	No reference
Potency (functional)	7.3753 uM	PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488752, AID488774, AID504848, AID504850]	ChEMBL.	No reference
Potency (functional)	14.7157 uM	PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488745, AID488752, AID488774, AID504848, AID504850]	ChEMBL.	No reference
Potency (functional)	= 28.1838 um	PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1). (Class of assay: confirmatory) [Related pubchem assays: 1030 (qHTS Validation Assay for Inhibitors of aldehyde dehydrogenase 1 (ALDH1A1))]	ChEMBL.	No reference
Potency (functional)	= 39.8107 um	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor. (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	= 50.1187 um	PUBCHEM_BIOASSAY: qHTS Inhibitors of AmpC Beta-Lactamase (assay with detergent). (Class of assay: confirmatory) [Related pubchem assays: 1002 (Confirmation Concentration-Response Assay for Inhibitors of AmpC Beta-Lactamase (assay with detergent)), 585 (Promiscuous and Specific Inhibitors of AmpC Beta-Lactamase (assay without detergent) - a screen old NIH MLSMR collection), 584 (Promiscuous and Specific Inhibitors of AmpC Beta-Lactamase (assay with detergent) - a screen of the old NIH MLSMR collection), 1003 (Confirmation Cuvette-Based Assay for Inhibitors of AmpC Beta-Lactamase (assay with detergent))]	ChEMBL.	No reference

Phenotypes

Whole-cell/tissue/organism interactions

Species name	Source	Reference	Is orphan
Plasmodium falciparum	ChEMBL23
Homo sapiens	ChEMBL23

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL1542938

Bibliographic References

No literature references available for this target.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 1407505