Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | hypothetical protein | 0.0381 | 0.0848 | 0.0848 |
Echinococcus multilocularis | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0381 | 0.0848 | 0.0848 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0595 | 0.3645 | 0.173 |
Schistosoma mansoni | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0493 | 0.2315 | 0.2315 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Giardia lamblia | Alpha-tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin subunit TubB | 0.0595 | 0.3645 | 0.173 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | hypothetical protein | 0.0595 | 0.3645 | 0.3645 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0595 | 0.3645 | 0.3645 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0595 | 0.3645 | 0.3645 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0595 | 0.3645 | 0.3645 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0595 | 0.3645 | 0.3645 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0595 | 0.3645 | 0.3645 |
Trypanosoma brucei | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Schistosoma mansoni | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Brugia malayi | Tubulin alpha-2 chain | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0381 | 0.0848 | 0.0848 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0493 | 0.2315 | 0.2315 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0595 | 0.3645 | 0.3645 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0595 | 0.3645 | 0.173 |
Brugia malayi | Tubulin alpha-2 chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Schistosoma mansoni | tubulin subunit alpha | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | alpha-tubulin | 0.0595 | 0.3645 | 0.3645 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0595 | 0.3645 | 0.3645 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0595 | 0.3645 | 0.173 |
Schistosoma mansoni | tubulin subunit alpha | 0.0595 | 0.3645 | 0.173 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0493 | 0.2315 | 0.2315 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0595 | 0.3645 | 0.3645 |
Giardia lamblia | Alpha-tubulin | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0493 | 0.2315 | 0.2315 |
Plasmodium falciparum | alpha tubulin 2 | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0595 | 0.3645 | 0.3645 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0595 | 0.3645 | 0.173 |
Brugia malayi | tubulin alpha chain - mouse | 0.0595 | 0.3645 | 0.173 |
Plasmodium falciparum | alpha tubulin 1 | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0595 | 0.3645 | 0.3645 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0595 | 0.3645 | 0.3645 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0381 | 0.0848 | 0.0848 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | alpha-tubulin | 0.0595 | 0.3645 | 0.3645 |
Echinococcus multilocularis | hypothetical protein | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0595 | 0.3645 | 0.173 |
Brugia malayi | tubulin alpha-2 chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0595 | 0.3645 | 0.3645 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0595 | 0.3645 | 0.173 |
Trypanosoma brucei | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Trypanosoma brucei | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0595 | 0.3645 | 0.173 |
Schistosoma mansoni | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Brugia malayi | Tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Leishmania major | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Schistosoma mansoni | tubulin subunit alpha | 0.0595 | 0.3645 | 0.173 |
Echinococcus granulosus | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Brugia malayi | alpha-tubulin | 0.0595 | 0.3645 | 0.173 |
Trypanosoma brucei | alpha tubulin | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | tubulin alpha chain | 0.0595 | 0.3645 | 0.173 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0595 | 0.3645 | 0.173 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0381 | 0.0848 | 0.0848 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | = 45.6 uM | Cytotoxicity against human PC3 cells after 48 hrs by MTT assay | ChEMBL. | 23021967 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.