Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Vaccinia virus (strain Copenhagen) (VACV) | Uracil-DNA glycosylase | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.019 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin | 0.019 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0136 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0131 | 0.3094 | 0.1296 |
Loa Loa (eye worm) | tubulin alpha chain | 0.019 | 0.6486 | 0.5571 |
Loa Loa (eye worm) | hypothetical protein | 0.019 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0136 | 0.3392 | 0.3392 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.019 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.019 | 0.6486 | 0.5571 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin subunit TubB | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.019 | 0.6486 | 0.6486 |
Trypanosoma brucei | epsilon tubulin | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin subunit TubB | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0131 | 0.3094 | 0.3094 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0113 | 0.2066 | 0.2066 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.019 | 0.6486 | 0.6486 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0131 | 0.3094 | 0.1296 |
Trypanosoma brucei | epsilon tubulin | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.019 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.019 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0136 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha chain | 0.019 | 0.6486 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0131 | 0.3094 | 0.1296 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0136 | 0.3392 | 0.3392 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0131 | 0.3094 | 0.1296 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0136 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0136 | 0.3392 | 0.1672 |
Trypanosoma cruzi | alpha tubulin, putative | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.019 | 0.6486 | 0.6486 |
Giardia lamblia | Alpha-tubulin | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.019 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 10000 nM | Viral Plaque Reduction Assay | BINDINGDB. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.