Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0187 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0134 | 0.3392 | 0.3392 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | epsilon tubulin | 0.0134 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | hypothetical protein | 0.0187 | 0.6486 | 0.5571 |
Brugia malayi | tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | tubulin gamma chain | 0.0134 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0129 | 0.3094 | 0.1296 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0129 | 0.3094 | 0.1296 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0134 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0134 | 0.3392 | 0.3392 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0134 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.5571 |
Trypanosoma brucei | epsilon tubulin | 0.0134 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0134 | 0.3392 | 0.1672 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6486 | 0.5571 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0134 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0134 | 0.3392 | 0.3392 |
Brugia malayi | Tubulin alpha chain | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0129 | 0.3094 | 0.1296 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0187 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6486 | 0.5571 |
Plasmodium falciparum | alpha tubulin 1 | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0129 | 0.3094 | 0.3094 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6486 | 0.5571 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0111 | 0.2066 | 0.2066 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0129 | 0.3094 | 0.1296 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 6 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.