Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0129 | 0.3094 | 0.1296 |
Brugia malayi | alpha-tubulin | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0187 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0111 | 0.2066 | 0.2066 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0134 | 0.3392 | 0.1672 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0187 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0134 | 0.3392 | 0.3392 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0187 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | epsilon tubulin | 0.0134 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0187 | 0.6486 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6486 | 0.5571 |
Plasmodium falciparum | alpha tubulin 1 | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0129 | 0.3094 | 0.3094 |
Echinococcus multilocularis | hypothetical protein | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0134 | 0.3392 | 0.3392 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0134 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6486 | 0.5571 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0129 | 0.3094 | 0.1296 |
Trypanosoma brucei | epsilon tubulin | 0.0134 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0187 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0134 | 0.3392 | 0.3392 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0134 | 0.3392 | 0.3392 |
Plasmodium falciparum | alpha tubulin 2 | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6486 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0187 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0129 | 0.3094 | 0.1296 |
Brugia malayi | Tubulin alpha chain | 0.0187 | 0.6486 | 0.6486 |
Trypanosoma brucei | epsilon tubulin | 0.0134 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0134 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0129 | 0.3094 | 0.1296 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 6.6383 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.