Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tubulin alpha 3 chain | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0188 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.013 | 0.3094 | 0.1296 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0188 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0135 | 0.3392 | 0.3392 |
Trypanosoma brucei | beta tubulin | 0.0135 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0135 | 0.3392 | 0.1672 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0188 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0135 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0188 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0135 | 0.3392 | 0.3392 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0188 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0135 | 0.3392 | 0.3392 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0188 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0188 | 0.6486 | 0.6486 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0188 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0188 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0188 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0135 | 0.3392 | 0.3392 |
Trypanosoma brucei | epsilon tubulin | 0.0135 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | hypothetical protein | 0.0188 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0188 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0188 | 0.6486 | 0.6486 |
Brugia malayi | tubulin alpha-2 chain | 0.0188 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0135 | 0.3392 | 0.3392 |
Schistosoma mansoni | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.013 | 0.3094 | 0.1296 |
Trypanosoma brucei | alpha tubulin | 0.0188 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0188 | 0.6486 | 0.6486 |
Schistosoma mansoni | tubulin subunit alpha | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0188 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0188 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0188 | 0.6486 | 0.6486 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0188 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0188 | 0.6486 | 0.5571 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0188 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0188 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0188 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.013 | 0.3094 | 0.1296 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0112 | 0.2066 | 0.2066 |
Echinococcus granulosus | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0188 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0188 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0188 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0188 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0188 | 0.6486 | 0.6486 |
Brugia malayi | Tubulin alpha chain | 0.0188 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0188 | 0.6486 | 0.6486 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0135 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0188 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0188 | 0.6486 | 0.5571 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.013 | 0.3094 | 0.1296 |
Brugia malayi | alpha-tubulin | 0.0188 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0188 | 0.6486 | 0.6486 |
Echinococcus granulosus | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0188 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0188 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.0188 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0188 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0188 | 0.6486 | 0.5571 |
Trypanosoma brucei | alpha tubulin | 0.0188 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0188 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.013 | 0.3094 | 0.3094 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0188 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 5.4202 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.