Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0177 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0177 | 0.6486 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0177 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0122 | 0.3094 | 0.1296 |
Giardia lamblia | Alpha-tubulin | 0.0177 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0177 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0177 | 0.6486 | 0.5571 |
Brugia malayi | tubulin alpha chain - mouse | 0.0177 | 0.6486 | 0.6486 |
Giardia lamblia | Alpha-tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0177 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0127 | 0.3392 | 0.1672 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0105 | 0.2066 | 0.2066 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0127 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0177 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0177 | 0.6486 | 0.6486 |
Schistosoma mansoni | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0177 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0177 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0177 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0177 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0177 | 0.6486 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0127 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.0177 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0177 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0177 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0177 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0122 | 0.3094 | 0.3094 |
Schistosoma mansoni | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0177 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0177 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0127 | 0.3392 | 0.3392 |
Schistosoma mansoni | tubulin subunit alpha | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0177 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0177 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0177 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0127 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | alpha-tubulin | 0.0177 | 0.6486 | 0.5571 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0177 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0122 | 0.3094 | 0.1296 |
Trypanosoma brucei | epsilon tubulin | 0.0127 | 0.3392 | 0.3392 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0177 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0177 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0177 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0177 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0127 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0127 | 0.3392 | 0.3392 |
Plasmodium falciparum | alpha tubulin 2 | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0177 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0177 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0177 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0177 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0177 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0177 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0177 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0177 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0122 | 0.3094 | 0.1296 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0122 | 0.3094 | 0.1296 |
Trypanosoma brucei | epsilon tubulin | 0.0127 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0127 | 0.3392 | 0.3392 |
Schistosoma mansoni | tubulin subunit alpha | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0177 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 6.0506 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.