Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0178 | 0.5571 | 0.5571 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0178 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0178 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0178 | 0.5571 | 0.5571 |
Schistosoma mansoni | tubulin subunit alpha | 0.0178 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0122 | 0.1296 | 0.1296 |
Echinococcus multilocularis | hypothetical protein | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0178 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0127 | 0.1672 | 0.1672 |
Plasmodium falciparum | alpha tubulin 1 | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0122 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0127 | 0.1672 | 0.1672 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0178 | 0.5571 | 0.5571 |
Plasmodium falciparum | alpha tubulin 2 | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0122 | 0.1296 | 0.1296 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0127 | 0.1672 | 0.1672 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0178 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0122 | 0.1296 | 0.1296 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0127 | 0.1672 | 0.1672 |
Brugia malayi | tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0122 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
FC (binding) | = 1.06 | Inhibition of recombinant 6-His-tagged SLAM associated protein SH2 domain (unknown origin) expressed in Escherichia coli BL21(DE3) binding to biotinyl-KKSLTIpYAQVQK-NH2 attached to NeutrAvidin-coated plates using p-nitrophenyl phosphate as substrate at 10 uM after 1 hr relative to control | ChEMBL. | 23470190 |
Inhibition (binding) | Inhibition of recombinant 6-His-tagged SLAM associated protein SH2 domain (unknown origin) expressed in Escherichia coli BL21(DE3) binding to biotinyl-KKSLTIpYAQVQK-NH2 attached to NeutrAvidin-coated plates using p-nitrophenyl phosphate as substrate at 100 uM after 1 hr | ChEMBL. | 23470190 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.