Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | tubulin subunit alpha | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0383 | 0.4774 | 0.4774 |
Schistosoma mansoni | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0383 | 0.4774 | 0.4774 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0383 | 0.4774 | 0.4774 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | Tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.3517 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | tubulin alpha chain - mouse | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | alpha-tubulin | 0.0383 | 0.4774 | 0.4774 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0383 | 0.4774 | 0.3517 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0259 | 0.111 | 0.111 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0259 | 0.111 | 0.111 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin subunit TubB | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Loa Loa (eye worm) | hypothetical protein | 0.0259 | 0.111 | 0.111 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0287 | 0.1939 | 0.1939 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Giardia lamblia | Alpha-tubulin | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0383 | 0.4774 | 0.3517 |
Plasmodium falciparum | alpha tubulin 1 | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | hypothetical protein | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0287 | 0.1939 | 0.1939 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0287 | 0.1939 | 0.1939 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | hypothetical protein | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | alpha-tubulin | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0259 | 0.111 | 0.111 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0383 | 0.4774 | 0.4774 |
Loa Loa (eye worm) | alpha-tubulin | 0.0383 | 0.4774 | 0.4774 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0259 | 0.111 | 0.111 |
Giardia lamblia | Alpha-tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0383 | 0.4774 | 0.4774 |
Plasmodium falciparum | alpha tubulin 2 | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | Tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | tubulin subunit alpha | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | tubulin subunit alpha | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0287 | 0.1939 | 0.1939 |
Brugia malayi | Tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 5 uM | Cytotoxicity against mouse J774 cells assessed as cell viability after 72 hrs by Alamar blue assay | ChEMBL. | 23265887 |
Species name | Source | Reference | Is orphan |
---|---|---|---|
Mus musculus | ChEMBL23 | 23265887 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.