Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.013 | 0.1427 | 0.1427 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.013 | 0.1427 | 0.1427 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Brugia malayi | tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | hypothetical protein | 0.013 | 0.1427 | 0.1427 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0131 | 0.1484 | 0.1484 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Echinococcus granulosus | tubulin subunit TubB | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0187 | 0.6136 | 0.5463 |
Plasmodium falciparum | alpha tubulin 1 | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6136 | 0.6136 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0187 | 0.6136 | 0.6136 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6136 | 0.6136 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.5463 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | tubulin alpha chain - mouse | 0.0187 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6136 | 0.6136 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | alpha-tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.013 | 0.1427 | 0.1427 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6136 | 0.6136 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.013 | 0.1427 | 0.1427 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6136 | 0.6136 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0131 | 0.1484 | 0.1484 |
Echinococcus granulosus | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Plasmodium falciparum | alpha tubulin 2 | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0131 | 0.1484 | 0.1484 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | hypothetical protein | 0.0187 | 0.6136 | 0.6136 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0131 | 0.1484 | 0.1484 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | hypothetical protein | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0187 | 0.6136 | 0.5463 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
CC50 (ADMET) | > 100 uM | Cytotoxicity against Homo sapiens (human) MT4 cells containing integrated HTLV-1 genome after 96 hr by MTT assay | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.