Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Plasmodium falciparum | conserved protein, unknown function | 0.0125 | 0.0945 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | haspin protein kinase | 0.0586 | 0.9999 | 1 |
Trichomonas vaginalis | serine/threonine kinase, putative | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | protein kinase atmrk1, putative | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus granulosus | dual specificity | 0.0189 | 0.2206 | 0.1991 |
Echinococcus multilocularis | dual specificity | 0.0454 | 0.7398 | 0.7394 |
Loa Loa (eye worm) | carboxylesterase | 0.0091 | 0.0292 | 0.0292 |
Brugia malayi | Endochitinase | 0.0088 | 0.0227 | 0.0188 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus granulosus | acetylcholinesterase | 0.0541 | 0.9098 | 0.9163 |
Onchocerca volvulus | Putative endochitinase | 0.0088 | 0.0227 | 0.2052 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Toxoplasma gondii | cell-cycle-associated protein kinase DYRK2, putative | 0.0454 | 0.7398 | 1 |
Trypanosoma cruzi | dual specificity tyrosine-phosphorylation-regulated kinase 2, putative | 0.0454 | 0.7398 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus multilocularis | serine:threonine protein kinase NLK | 0.0105 | 0.0568 | 0.0287 |
Echinococcus granulosus | serine:threonine protein kinase NLK | 0.0105 | 0.0568 | 0.0287 |
Brugia malayi | Carboxylesterase family protein | 0.0541 | 0.9098 | 0.9184 |
Trypanosoma cruzi | CMGC/DYRK protein kinase, putative | 0.0189 | 0.2206 | 0.2399 |
Entamoeba histolytica | protein kinase, putative | 0.0189 | 0.2206 | 0.2943 |
Loa Loa (eye worm) | CMGC/DYRK/DYRK2 protein kinase | 0.0454 | 0.7398 | 0.7399 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus multilocularis | Cell division cycle 2 protein kinase | 0.0105 | 0.0568 | 0.0287 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Onchocerca volvulus | 0.0091 | 0.0292 | 0.2778 | |
Schistosoma mansoni | serine/threonine kinase | 0.0105 | 0.0568 | 0.0287 |
Trypanosoma cruzi | CMGC/DYRK protein kinase, putative | 0.0189 | 0.2206 | 0.2399 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus granulosus | acetylcholinesterase | 0.0541 | 0.9098 | 0.9163 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0454 | 0.7398 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Entamoeba histolytica | protein kinase, putative | 0.0454 | 0.7398 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0189 | 0.2206 | 0.2943 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | hypothetical protein | 0.0541 | 0.9098 | 0.91 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0105 | 0.0568 | 0.0716 |
Brugia malayi | Carboxylesterase family protein | 0.0091 | 0.0292 | 0.0255 |
Echinococcus granulosus | dual specificity | 0.0454 | 0.7398 | 0.7394 |
Schistosoma mansoni | hypothetical protein | 0.01 | 0.0472 | 0.0187 |
Loa Loa (eye worm) | carboxylesterase | 0.0091 | 0.0292 | 0.0292 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0189 | 0.2206 | 0.1991 |
Brugia malayi | cyclin-dependent kinase 7 homolog | 0.0105 | 0.0568 | 0.0534 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Echinococcus granulosus | serine:threonine protein kinase haspin | 0.0582 | 0.9903 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | CMGC/CDK/CRK7 protein kinase | 0.0105 | 0.0568 | 0.0568 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus multilocularis | dual specificity | 0.0454 | 0.7398 | 0.7394 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0454 | 0.7398 | 1 |
Trichomonas vaginalis | G protein-coupled receptor kinase, putative | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | CMGC/DYRK/DYRK1 protein kinase | 0.0189 | 0.2206 | 0.2206 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Brugia malayi | hypothetical protein | 0.0091 | 0.0292 | 0.0255 |
Echinococcus granulosus | Hepatocellular carcinoma associated antigen 59 | 0.0125 | 0.0945 | 0.068 |
Loa Loa (eye worm) | hypothetical protein | 0.0541 | 0.9098 | 0.91 |
Brugia malayi | endochitinase | 0.0088 | 0.0227 | 0.0188 |
Loa Loa (eye worm) | hypothetical protein | 0.0125 | 0.0945 | 0.0946 |
Echinococcus granulosus | carboxylesterase 5A | 0.0541 | 0.9098 | 0.9163 |
Leishmania major | protein kinase, putative,dual-specificity protein kinase, putative | 0.0454 | 0.7398 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0454 | 0.7398 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Mycobacterium ulcerans | flavin-containing monoamine oxidase AofH | 0.0587 | 1 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Entamoeba histolytica | hypothetical protein | 0.01 | 0.0472 | 0.0586 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Leishmania major | serine/threonine kinase-like protein, putative | 0.0105 | 0.0568 | 0.0716 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Onchocerca volvulus | Putative endochitinase | 0.0088 | 0.0227 | 0.2052 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Brugia malayi | Protein kinase domain containing protein | 0.0105 | 0.0568 | 0.0534 |
Entamoeba histolytica | hypothetical protein | 0.0189 | 0.2206 | 0.2943 |
Schistosoma mansoni | protein kinase | 0.0105 | 0.0568 | 0.0287 |
Trypanosoma brucei | dual specificity tyrosine-phosphorylation-regulated kinase 2, putative | 0.0454 | 0.7398 | 1 |
Echinococcus multilocularis | serine:threonine protein kinase haspin | 0.0582 | 0.9903 | 1 |
Onchocerca volvulus | 0.0091 | 0.0292 | 0.2778 | |
Brugia malayi | Protein kinase domain containing protein | 0.0189 | 0.2206 | 0.2195 |
Giardia lamblia | Kinase, CMGC DYRK | 0.0454 | 0.7398 | 1 |
Leishmania major | serine/threonine-protein kinase, putative,protein kinase, putative | 0.0189 | 0.2206 | 0.2943 |
Echinococcus granulosus | serine:threonine protein kinase haspin | 0.0582 | 0.9903 | 1 |
Brugia malayi | Cell division protein kinase 2 | 0.0105 | 0.0568 | 0.0534 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0105 | 0.0568 | 0.0287 |
Loa Loa (eye worm) | acetylcholinesterase 1 | 0.0541 | 0.9098 | 0.91 |
Onchocerca volvulus | 0.0125 | 0.0945 | 1 | |
Leishmania major | mitogen-activated protein kinase, putative,map kinase-like protein | 0.0105 | 0.0568 | 0.0716 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus multilocularis | acetylcholinesterase | 0.0541 | 0.9098 | 0.9163 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trypanosoma brucei | CMGC/DYRK protein kinase, putative | 0.0189 | 0.2206 | 0.2399 |
Echinococcus granulosus | dual specificity | 0.0454 | 0.7398 | 0.7394 |
Loa Loa (eye worm) | haspin protein kinase | 0.0582 | 0.9903 | 0.9904 |
Echinococcus multilocularis | cyclin dependent kinase 9 | 0.0105 | 0.0568 | 0.0287 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0454 | 0.7398 | 1 |
Brugia malayi | GSG2 | 0.0582 | 0.9903 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0454 | 0.7398 | 0.7394 |
Echinococcus multilocularis | Hepatocellular carcinoma associated antigen 59 | 0.0125 | 0.0945 | 0.068 |
Loa Loa (eye worm) | hypothetical protein | 0.0125 | 0.0945 | 0.0946 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus granulosus | dual specificity | 0.0454 | 0.7398 | 0.7394 |
Schistosoma mansoni | family S9 non-peptidase homologue (S09 family) | 0.0541 | 0.9098 | 0.9163 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Entamoeba histolytica | cell division protein kinase 2, putative | 0.0105 | 0.0568 | 0.0716 |
Loa Loa (eye worm) | cuticular endochitinase | 0.0079 | 0.0041 | 0.0041 |
Echinococcus multilocularis | dual specificity | 0.0189 | 0.2206 | 0.1991 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0454 | 0.7398 | 1 |
Brugia malayi | Dual-specificity tyrosine-phosphorylation regulated kinase 2 | 0.0454 | 0.7398 | 0.746 |
Brugia malayi | Carboxylesterase family protein | 0.0091 | 0.0292 | 0.0255 |
Schistosoma mansoni | hypothetical protein | 0.0125 | 0.0945 | 0.068 |
Brugia malayi | Carboxylesterase family protein | 0.0091 | 0.0292 | 0.0255 |
Onchocerca volvulus | 0.0091 | 0.0292 | 0.2778 | |
Mycobacterium tuberculosis | Probable flavin-containing monoamine oxidase AofH (amine oxidase) (MAO) | 0.0545 | 0.919 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Onchocerca volvulus | 0.0091 | 0.0292 | 0.2778 | |
Echinococcus multilocularis | dual specificity | 0.0454 | 0.7398 | 0.7394 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Entamoeba histolytica | protein kinase, putative | 0.0189 | 0.2206 | 0.2943 |
Brugia malayi | Carboxylesterase family protein | 0.0541 | 0.9098 | 0.9184 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | chitinase I | 0.0079 | 0.0041 | 0.0041 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Onchocerca volvulus | 0.0125 | 0.0945 | 1 | |
Echinococcus granulosus | mitogen activated protein kinase 15 | 0.0105 | 0.0568 | 0.0287 |
Echinococcus multilocularis | serine:threonine protein kinase haspin | 0.0582 | 0.9903 | 1 |
Loa Loa (eye worm) | haspin protein kinase | 0.0582 | 0.9903 | 0.9904 |
Brugia malayi | hypothetical protein | 0.0582 | 0.9903 | 1 |
Echinococcus granulosus | serine:threonine protein kinase haspin | 0.0582 | 0.9903 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Onchocerca volvulus | Putative endochitinase | 0.0088 | 0.0227 | 0.2052 |
Onchocerca volvulus | 0.0091 | 0.0292 | 0.2778 | |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0105 | 0.0568 | 0.0568 |
Schistosoma mansoni | hypothetical protein | 0.0582 | 0.9903 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | hypothetical protein | 0.0184 | 0.211 | 0.2111 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Brugia malayi | Hepatocellular carcinoma-associated antigen 59 family protein | 0.0125 | 0.0945 | 0.0917 |
Echinococcus granulosus | Pfam-B_8186 domain containing protein | 0.01 | 0.0472 | 0.0187 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Loa Loa (eye worm) | hypothetical protein | 0.0184 | 0.211 | 0.2111 |
Echinococcus multilocularis | carboxylesterase 5A | 0.0541 | 0.9098 | 0.9163 |
Loa Loa (eye worm) | carboxylesterase | 0.0541 | 0.9098 | 0.91 |
Echinococcus granulosus | Cell division cycle 2 protein kinase | 0.0105 | 0.0568 | 0.0287 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0454 | 0.7398 | 1 |
Echinococcus granulosus | cyclin dependent kinase 9 | 0.0105 | 0.0568 | 0.0287 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0454 | 0.7398 | 1 |
Echinococcus multilocularis | acetylcholinesterase | 0.0541 | 0.9098 | 0.9163 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Brugia malayi | Carboxylesterase family protein | 0.0091 | 0.0292 | 0.0255 |
Loa Loa (eye worm) | hypothetical protein | 0.0091 | 0.0292 | 0.0292 |
Plasmodium vivax | hypothetical protein, conserved | 0.0125 | 0.0945 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Echinococcus multilocularis | hypothetical protein | 0.01 | 0.0472 | 0.0187 |
Trichomonas vaginalis | AGC family protein kinase | 0.0105 | 0.0568 | 0.0388 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | = 31.6228 um | PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | 125.8925 uM | PubChem BioAssay. qHTS of PTHR Inhibitors: Primary Screen. (Class of assay: confirmatory) | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.