Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | tar DNA-binding protein | 0.0062 | 0.3288 | 0.299 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | CMGC family protein kinase | 0.005 | 0.2504 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0062 | 0.3288 | 0.299 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0018 | 0.0427 | 0.0011 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Schistosoma mansoni | tar DNA-binding protein | 0.0062 | 0.3288 | 0.299 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trypanosoma cruzi | mitogen activated protein kinase 4, putative | 0.005 | 0.2504 | 1 |
Echinococcus granulosus | serine protein kinase ATM | 0.0024 | 0.0852 | 0.0446 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Echinococcus multilocularis | mitogen activated protein kinase | 0.005 | 0.2504 | 0.2172 |
Echinococcus granulosus | tar DNA binding protein | 0.0062 | 0.3288 | 0.299 |
Trichomonas vaginalis | CMGC family protein kinase | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Echinococcus multilocularis | geminin | 0.0167 | 1 | 1 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0024 | 0.0852 | 0.0515 |
Toxoplasma gondii | CMGC kinase, MAPK family (ERK) MAPK-1 | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Echinococcus granulosus | muscleblind protein | 0.0147 | 0.873 | 0.8674 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0018 | 0.0425 | 0.0487 |
Schistosoma mansoni | hypothetical protein | 0.0167 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0632 | 0.0724 |
Echinococcus multilocularis | serine protein kinase ATM | 0.0024 | 0.0852 | 0.0446 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trypanosoma cruzi | mitogen-activated protein kinase 11, putative | 0.005 | 0.2504 | 1 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0018 | 0.0425 | 0.0487 |
Echinococcus multilocularis | mitogen activated protein kinase 3 | 0.005 | 0.2504 | 0.2172 |
Brugia malayi | RNA binding protein | 0.0062 | 0.3288 | 0.3447 |
Leishmania major | mitogen activated protein kinase 4, putative;with=GeneDB:LmxM19.1440 | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0024 | 0.0852 | 0.2055 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Brugia malayi | MAP kinase sur-1 | 0.005 | 0.2504 | 0.2504 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0024 | 0.0852 | 0.3404 |
Echinococcus granulosus | mitogen activated protein kinase | 0.005 | 0.2504 | 0.2172 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm) | 0.0024 | 0.0852 | 0.0446 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Giardia lamblia | Kinase, CMGC MAPK | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | CMGC family protein kinase | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Leishmania major | mitogen activated protein kinase, putative,map kinase, putative | 0.005 | 0.2504 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0062 | 0.3288 | 0.299 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.0018 | 0.0425 | 0.1697 |
Entamoeba histolytica | hypothetical protein | 0.0024 | 0.0852 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trypanosoma brucei | mitogen activated protein kinase 4, putative | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.005 | 0.2504 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0062 | 0.3288 | 0.299 |
Leishmania major | phosphatidylinositol kinase related protein, putative | 0.0018 | 0.0427 | 0.0011 |
Trypanosoma brucei | phosphatidylinositol 3-related kinase, putative | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Schistosoma mansoni | serine/threonine protein kinase | 0.005 | 0.2504 | 0.2172 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Brugia malayi | TAR-binding protein | 0.0062 | 0.3288 | 0.3447 |
Trypanosoma brucei | phosphatidylinositol kinase related protein, putative | 0.0024 | 0.0852 | 0.3404 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0021 | 0.0632 | 0.0997 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Loa Loa (eye worm) | RNA binding protein | 0.0062 | 0.3288 | 0.3766 |
Trypanosoma cruzi | mitogen activated protein kinase 2, putative | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Loa Loa (eye worm) | hypothetical protein | 0.0147 | 0.873 | 1 |
Brugia malayi | Muscleblind-like protein | 0.0147 | 0.873 | 1 |
Echinococcus multilocularis | muscleblind protein | 0.0147 | 0.873 | 0.8674 |
Loa Loa (eye worm) | hypothetical protein | 0.0147 | 0.873 | 1 |
Echinococcus multilocularis | muscleblind protein 1 | 0.0147 | 0.873 | 0.8674 |
Loa Loa (eye worm) | CMGC/MAPK/ERK1 protein kinase | 0.005 | 0.2504 | 0.2869 |
Echinococcus granulosus | mitogen activated protein kinase 3 | 0.005 | 0.2504 | 0.2172 |
Trypanosoma brucei | phosphatidylinositol 3-kinase, putative | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Toxoplasma gondii | target of rapamycin (TOR), putative | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.0018 | 0.0425 | 0.1697 |
Loa Loa (eye worm) | RNA recognition domain-containing protein domain-containing protein | 0.0062 | 0.3288 | 0.3766 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.0018 | 0.0425 | 0.1697 |
Loa Loa (eye worm) | TAR-binding protein | 0.0062 | 0.3288 | 0.3766 |
Brugia malayi | RNA recognition motif domain containing protein | 0.0062 | 0.3288 | 0.3447 |
Toxoplasma gondii | FATC domain-containing protein | 0.0024 | 0.0852 | 0.3404 |
Trypanosoma cruzi | mitogen-activated protein kinase 11, putative | 0.005 | 0.2504 | 1 |
Echinococcus multilocularis | tar DNA binding protein | 0.0062 | 0.3288 | 0.299 |
Trypanosoma brucei | protein kinase, putative | 0.005 | 0.2504 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0018 | 0.0425 | 0.1697 |
Schistosoma mansoni | hypothetical protein | 0.0167 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | 23.0999 uM | PUBCHEM_BIOASSAY: qHTS screen for small molecules that inhibit ELG1-dependent DNA repair in human embryonic kidney (HEK293T) cells expressing luciferase-tagged ELG1. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493107, AID493125] | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.