Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Rattus norvegicus | Cannabinoid receptor | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Schistosoma mansoni | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Mycobacterium tuberculosis | Probable purine nucleoside phosphorylase DeoD (inosine phosphorylase) (PNP) | 0.1658 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Plasmodium falciparum | purine nucleoside phosphorylase | 0.0343 | 0 | 0.5 |
Schistosoma mansoni | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1315 | 0.7389 | 0.7389 |
Trypanosoma cruzi | methylthioadenosine phosphorylase, putative | 0.0343 | 0 | 0.5 |
Toxoplasma gondii | phosphorylase family protein | 0.0343 | 0 | 0.5 |
Trypanosoma brucei | uridine phosphorylase | 0.0343 | 0 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Entamoeba histolytica | MTA/SAH nucleosidase, putative | 0.0343 | 0 | 0.5 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Leishmania major | nucleoside phosphorylase-like protein | 0.0343 | 0 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Toxoplasma gondii | Purine nucleoside phosphorylase | 0.0343 | 0 | 0.5 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Mycobacterium ulcerans | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Treponema pallidum | uridine phosphorylase (udp) | 0.0343 | 0 | 0.5 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Trypanosoma cruzi | nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Onchocerca volvulus | Purine nucleoside phosphorylase homolog | 0.1658 | 1 | 0.5 |
Treponema pallidum | pfs protein (pfs) | 0.0343 | 0 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.1315 | 0.7389 | 1 |
Trichomonas vaginalis | purine nucleoside phosphorylase I, putative | 0.1658 | 1 | 1 |
Leishmania major | methylthioadenosine phosphorylase, putative | 0.0343 | 0 | 0.5 |
Trypanosoma cruzi | methylthioadenosine phosphorylase, putative | 0.0343 | 0 | 0.5 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1315 | 0.7389 | 0.7389 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0343 | 0 | 0.5 |
Giardia lamblia | Purine nucleoside phosphorylase lateral transfer candidate | 0.1658 | 1 | 1 |
Toxoplasma gondii | phosphorylase family protein | 0.0343 | 0 | 0.5 |
Trypanosoma cruzi | nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Plasmodium vivax | purine nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Trypanosoma brucei | methylthioadenosine phosphorylase, putative | 0.0343 | 0 | 0.5 |
Chlamydia trachomatis | AMP nucleosidase | 0.0343 | 0 | 0.5 |
Treponema pallidum | purine nucleoside phosphorylase (deoD) | 0.0343 | 0 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Mycobacterium leprae | Probable purine nucleoside phosphorylase DeoD (INOSINE PHOSPHORYLASE) (PNP) | 0.1658 | 1 | 1 |
Trypanosoma cruzi | nucleoside phosphorylase, putative | 0.0343 | 0 | 0.5 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1658 | 1 | 1 |
Echinococcus granulosus | inosine guanosine and xanthosine phosphorylase | 0.1315 | 0.7389 | 0.7389 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 48.3 nM | Concentration required to displace 50% of 0.5 nM [3H]-(Aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranes | ChEMBL. | 1732519 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.