Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0386 | 0.479 | 0.479 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0386 | 0.479 | 0.479 |
Echinococcus granulosus | tubulin subunit TubB | 0.0386 | 0.479 | 0.3541 |
Plasmodium falciparum | alpha tubulin 2 | 0.0386 | 0.479 | 0.3541 |
Schistosoma mansoni | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0386 | 0.479 | 0.3541 |
Schistosoma mansoni | tubulin subunit beta | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0289 | 0.1933 | 0.1933 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0386 | 0.479 | 0.3541 |
Entamoeba histolytica | tubulin family protein | 0.0564 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0564 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0564 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0289 | 0.1933 | 0.1933 |
Brugia malayi | Tubulin alpha-2 chain | 0.0386 | 0.479 | 0.3541 |
Loa Loa (eye worm) | BEN-1 protein | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0386 | 0.479 | 0.3541 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Loa Loa (eye worm) | tubulin beta chain | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0564 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | hypothetical protein | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0386 | 0.479 | 0.3541 |
Schistosoma mansoni | tubulin subunit alpha | 0.0386 | 0.479 | 0.3541 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0386 | 0.479 | 0.3541 |
Trypanosoma brucei | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0386 | 0.479 | 0.3541 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0564 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0386 | 0.479 | 0.3541 |
Giardia lamblia | Alpha-tubulin | 0.0386 | 0.479 | 0.3541 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0386 | 0.479 | 0.479 |
Schistosoma mansoni | tubulin subunit beta | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0386 | 0.479 | 0.479 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0564 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0564 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0564 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0386 | 0.479 | 0.3541 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0289 | 0.1933 | 0.1933 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | tubulin subunit beta | 0.0564 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0564 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0564 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Trypanosoma brucei | beta tubulin | 0.0564 | 1 | 1 |
Brugia malayi | tubulin alpha-2 chain | 0.0386 | 0.479 | 0.3541 |
Schistosoma mansoni | tubulin subunit beta | 0.0564 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Loa Loa (eye worm) | hypothetical protein | 0.0261 | 0.1114 | 0.1114 |
Loa Loa (eye worm) | alpha-tubulin | 0.0386 | 0.479 | 0.479 |
Trypanosoma brucei | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Schistosoma mansoni | tubulin subunit beta | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0564 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0289 | 0.1933 | 0.1933 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0386 | 0.479 | 0.479 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0386 | 0.479 | 0.479 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0261 | 0.1114 | 0.1114 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0386 | 0.479 | 0.3541 |
Giardia lamblia | Beta tubulin | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0261 | 0.1114 | 0.1114 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0386 | 0.479 | 0.3541 |
Trypanosoma brucei | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0386 | 0.479 | 0.479 |
Giardia lamblia | Beta tubulin | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0386 | 0.479 | 0.479 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0386 | 0.479 | 0.3541 |
Trypanosoma brucei | beta tubulin | 0.0564 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0564 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Plasmodium falciparum | alpha tubulin 1 | 0.0386 | 0.479 | 0.3541 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0386 | 0.479 | 0.479 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin subunit beta | 0.0564 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Toxoplasma gondii | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0386 | 0.479 | 0.479 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0386 | 0.479 | 0.3541 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0386 | 0.479 | 0.3541 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0386 | 0.479 | 0.479 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | beta tubulin | 0.0564 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0564 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0261 | 0.1114 | 0.1114 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0564 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0386 | 0.479 | 0.3541 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0564 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Trypanosoma brucei | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus granulosus | tubulin alpha chain | 0.0386 | 0.479 | 0.3541 |
Brugia malayi | Tubulin alpha-2 chain | 0.0386 | 0.479 | 0.3541 |
Brugia malayi | tubulin alpha chain - mouse | 0.0386 | 0.479 | 0.3541 |
Giardia lamblia | Alpha-tubulin | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0261 | 0.1114 | 0.1114 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Plasmodium vivax | tubulin beta chain, putative | 0.0564 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0386 | 0.479 | 0.479 |
Leishmania major | alpha tubulin | 0.0386 | 0.479 | 0.3541 |
Trypanosoma brucei | beta tubulin | 0.0564 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0386 | 0.479 | 0.479 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0386 | 0.479 | 0.3541 |
Loa Loa (eye worm) | beta-tubulin | 0.0564 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0386 | 0.479 | 0.3541 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0564 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0564 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0386 | 0.479 | 0.3541 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0386 | 0.479 | 0.479 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0564 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0386 | 0.479 | 0.3541 |
Trichomonas vaginalis | tubulin, putative | 0.0564 | 1 | 1 |
Leishmania major | beta tubulin | 0.0564 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (functional) | = 16 % | Antiinflammatory activity in human whole blood assessed as inhibition of LPS-induced TNFalpha production at 10 uM treated for 30 mins followed by 5 hrs LPS challenge by ELISA-based WBCCS assay | ChEMBL. | 21600765 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.