Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0023 | 0.6625 | 0.6625 |
Leishmania major | NADPH-cytochrome p450 reductase-like protein | 0.0029 | 1 | 1 |
Plasmodium vivax | NADPH-cytochrome p450 reductase, putative | 0.0029 | 1 | 1 |
Leishmania major | p450 reductase, putative | 0.0029 | 1 | 1 |
Trypanosoma cruzi | cytochrome P450 reductase, putative | 0.0029 | 1 | 1 |
Trypanosoma cruzi | cytochrome P450 reductase, putative | 0.0029 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0023 | 0.6625 | 0.6625 |
Trypanosoma brucei | NADPH--cytochrome P450 reductase, putative | 0.0029 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0023 | 0.6625 | 1 |
Trypanosoma brucei | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Trypanosoma cruzi | NADPH-dependent FMN/FAD containing oxidoreductase, putative | 0.0029 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Loa Loa (eye worm) | tubulin beta chain | 0.0023 | 0.6625 | 0.6625 |
Chlamydia trachomatis | sulfite reductase | 0.0018 | 0.3805 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0023 | 0.6625 | 0.5864 |
Brugia malayi | beta-tubulin, identical | 0.0023 | 0.6625 | 0.6625 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Trypanosoma brucei | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0023 | 0.6625 | 0.4552 |
Schistosoma mansoni | tubulin subunit beta | 0.0023 | 0.6625 | 0.5864 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0023 | 0.6625 | 0.4552 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Trypanosoma brucei | NADPH-dependent diflavin oxidoreductase 1 | 0.0029 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0023 | 0.6625 | 0.4552 |
Echinococcus granulosus | tubulin subunit beta | 0.0023 | 0.6625 | 0.4552 |
Trypanosoma brucei | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Trypanosoma brucei | NADPH-cytochrome p450 reductase, putative | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus multilocularis | NADPH cytochrome P450 reductase | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus granulosus | NADPH cytochrome P450 reductase | 0.0029 | 1 | 1 |
Plasmodium falciparum | nitric oxide synthase, putative | 0.0029 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0023 | 0.6625 | 0.6625 |
Toxoplasma gondii | beta-tubulin, putative | 0.0023 | 0.6625 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0023 | 0.6625 | 0.5864 |
Schistosoma mansoni | 5-methyl tetrahydrofolate-homocysteine methyltransferase reductase | 0.0018 | 0.3805 | 0.2407 |
Schistosoma mansoni | NADPH flavin oxidoreductase | 0.0015 | 0.1964 | 0.0151 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0023 | 0.6625 | 0.6625 |
Giardia lamblia | Hypothetical protein | 0.0026 | 0.8159 | 1 |
Treponema pallidum | flavodoxin | 0.0011 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0023 | 0.6625 | 1 |
Brugia malayi | FAD binding domain containing protein | 0.0029 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Loa Loa (eye worm) | BEN-1 protein | 0.0023 | 0.6625 | 0.6625 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0023 | 0.6625 | 0.6625 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0023 | 0.6625 | 0.6625 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0023 | 0.6625 | 0.6625 |
Schistosoma mansoni | tubulin subunit beta | 0.0023 | 0.6625 | 0.5864 |
Loa Loa (eye worm) | hypothetical protein | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Schistosoma mansoni | tubulin subunit beta | 0.0023 | 0.6625 | 0.5864 |
Entamoeba histolytica | tubulin family protein | 0.0023 | 0.6625 | 1 |
Loa Loa (eye worm) | FAD binding domain-containing protein | 0.0018 | 0.3805 | 0.3805 |
Echinococcus multilocularis | beta tubulin | 0.0023 | 0.6625 | 0.4552 |
Plasmodium falciparum | tubulin beta chain | 0.0023 | 0.6625 | 0.6625 |
Brugia malayi | FAD binding domain containing protein | 0.0018 | 0.3805 | 0.3805 |
Trichomonas vaginalis | sulfite reductase, putative | 0.0029 | 1 | 1 |
Loa Loa (eye worm) | FAD binding domain-containing protein | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0023 | 0.6625 | 0.6625 |
Trypanosoma cruzi | p450 reductase, putative | 0.0029 | 1 | 1 |
Leishmania major | cytochrome P450 reductase, putative | 0.0026 | 0.8159 | 0.8159 |
Echinococcus granulosus | NADPH dependent diflavin oxidoreductase 1 | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Schistosoma mansoni | cytochrome P450 reductase | 0.0029 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0023 | 0.6625 | 0.4552 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Giardia lamblia | Nitric oxide synthase, inducible | 0.0026 | 0.8159 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus multilocularis | NADPH dependent diflavin oxidoreductase 1 | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus multilocularis | beta tubulin | 0.0023 | 0.6625 | 0.4552 |
Schistosoma mansoni | tubulin subunit beta | 0.0023 | 0.6625 | 0.5864 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Plasmodium vivax | flavodoxin domain containing protein | 0.0026 | 0.8159 | 0.8159 |
Brugia malayi | Tubulin beta-1 chain | 0.0023 | 0.6625 | 0.6625 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0023 | 0.6625 | 0.4552 |
Entamoeba histolytica | tubulin family protein | 0.0023 | 0.6625 | 1 |
Trypanosoma brucei | NADPH--cytochrome P450 reductase, putative | 0.0029 | 1 | 1 |
Leishmania major | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0023 | 0.6625 | 0.6625 |
Loa Loa (eye worm) | beta-tubulin | 0.0023 | 0.6625 | 0.6625 |
Trichomonas vaginalis | NADPH fad oxidoreductase, putative | 0.0026 | 0.8159 | 0.8159 |
Echinococcus multilocularis | tubulin subunit beta | 0.0023 | 0.6625 | 0.4552 |
Trichomonas vaginalis | tubulin, putative | 0.0023 | 0.6625 | 0.6625 |
Echinococcus granulosus | beta tubulin | 0.0023 | 0.6625 | 0.4552 |
Mycobacterium ulcerans | formate dehydrogenase H FdhF | 0.0029 | 1 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0023 | 0.6625 | 0.6625 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0023 | 0.6625 | 0.4552 |
Loa Loa (eye worm) | BEN-1 protein | 0.0023 | 0.6625 | 0.6625 |
Plasmodium vivax | tubulin beta chain, putative | 0.0023 | 0.6625 | 0.6625 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.