Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | cannabinoid receptor 1 (brain) | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0083 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0083 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0083 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0083 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0083 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0083 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0083 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0083 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0083 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0083 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0083 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0083 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0083 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0083 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0083 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0083 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0083 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0083 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0083 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0083 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0083 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0083 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0083 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0083 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0083 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0083 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0083 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0083 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0083 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Leishmania major | beta tubulin | 0.0083 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0083 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0083 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0083 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0083 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 5423 nM | Agonist activity at human CB1 receptor expressed in HEK293 EBNA cells by [35S]GTPgamma binding assay | ChEMBL. | 22284817 |
Emax (functional) | = 66 % | Agonist activity at human CB1 receptor expressed in HEK293 EBNA cells by [35S]GTPgamma binding assay relative to Win55,212-2 | ChEMBL. | 22284817 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.