Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma brucei | epsilon tubulin | 0.0258 | 0.3496 | 0.2724 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0266 | 0.3635 | 0.3628 |
Brugia malayi | Tubulin beta chain | 0.0112 | 0.1061 | 0.1061 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0146 | 0.1627 | 0.0634 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0266 | 0.3635 | 0.3628 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0266 | 0.3635 | 0.288 |
Leishmania major | epsilon tubulin, putative | 0.0258 | 0.3496 | 0.2724 |
Schistosoma mansoni | tubulin subunit epsilon | 0.0258 | 0.3496 | 0.3195 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0266 | 0.3635 | 0.3635 |
Echinococcus multilocularis | tubulin gamma 1 chain | 0.0258 | 0.3496 | 0.3488 |
Loa Loa (eye worm) | tubulin beta chain | 0.0112 | 0.1061 | 0.1061 |
Schistosoma mansoni | tubulin subunit gamma | 0.0258 | 0.3496 | 0.3195 |
Schistosoma mansoni | tubulin subunit alpha | 0.0112 | 0.1061 | 0.0647 |
Echinococcus multilocularis | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Brugia malayi | Tubulin alpha chain | 0.0112 | 0.1061 | 0.1061 |
Schistosoma mansoni | alpha tubulin | 0.0266 | 0.3635 | 0.3341 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0154 | 0.1767 | 0.1767 |
Brugia malayi | Tubulin gamma chain | 0.0258 | 0.3496 | 0.3496 |
Schistosoma mansoni | tubulin subunit alpha | 0.0266 | 0.3635 | 0.3341 |
Loa Loa (eye worm) | hypothetical protein | 0.0266 | 0.3635 | 0.3635 |
Plasmodium falciparum | alpha tubulin 1 | 0.0266 | 0.3635 | 0.3341 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0266 | 0.3635 | 0.3341 |
Plasmodium falciparum | tubulin delta chain, putative | 0.0112 | 0.1061 | 0.0647 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0266 | 0.3635 | 0.3628 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Toxoplasma gondii | tubulin/FtsZ family, GTPase domain-containing protein | 0.0258 | 0.3496 | 0.3195 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0146 | 0.1627 | 0.0634 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0266 | 0.3635 | 0.288 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0266 | 0.3635 | 0.3628 |
Loa Loa (eye worm) | alpha-tubulin | 0.0266 | 0.3635 | 0.3635 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.012 | 0.12 | 0.0156 |
Echinococcus multilocularis | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Echinococcus multilocularis | tubulin epsilon chain | 0.0258 | 0.3496 | 0.3488 |
Echinococcus granulosus | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Brugia malayi | alpha-tubulin | 0.0266 | 0.3635 | 0.3635 |
Echinococcus multilocularis | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Echinococcus granulosus | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0146 | 0.1627 | 0.0634 |
Trypanosoma brucei | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Echinococcus multilocularis | hypothetical protein | 0.0266 | 0.3635 | 0.3628 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0266 | 0.3635 | 0.3341 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0266 | 0.3635 | 0.3341 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0266 | 0.3635 | 0.3628 |
Loa Loa (eye worm) | hypothetical protein | 0.0075 | 0.0442 | 0.0442 |
Mycobacterium leprae | PROBABLE ATP-DEPENDENT CLP PROTEASE PROTEOLYTIC SUBUNIT 2 CLPP2 (ENDOPEPTIDASE CLP 2) | 0.0075 | 0.0442 | 0.4103 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0266 | 0.3635 | 0.0214 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0266 | 0.3635 | 0.3628 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0266 | 0.3635 | 0.288 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Echinococcus multilocularis | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Giardia lamblia | Alpha-tubulin | 0.0266 | 0.3635 | 0.288 |
Echinococcus granulosus | tubulin delta chain | 0.0112 | 0.1061 | 0.1051 |
Giardia lamblia | Gamma tubulin | 0.0258 | 0.3496 | 0.2724 |
Loa Loa (eye worm) | tubulin alpha-3 chain | 0.012 | 0.12 | 0.12 |
Brugia malayi | tubulin alpha chain - mouse | 0.0266 | 0.3635 | 0.3635 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Brugia malayi | Cell division protein ftsZ | 0.0112 | 0.1061 | 0.1061 |
Echinococcus granulosus | alpha tubulin | 0.0266 | 0.3635 | 0.3628 |
Echinococcus granulosus | tubulin alpha | 0.0258 | 0.3496 | 0.3488 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Loa Loa (eye worm) | alpha-tubulin | 0.0266 | 0.3635 | 0.3635 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0258 | 0.3496 | 0.2724 |
Toxoplasma gondii | tubulin/FtsZ family, GTPase domain-containing protein | 0.0112 | 0.1061 | 0.0647 |
Trichomonas vaginalis | tubulin, putative | 0.0146 | 0.1627 | 0.0634 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0266 | 0.3635 | 0.3628 |
Trypanosoma brucei | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0266 | 0.3635 | 0.288 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0146 | 0.1627 | 0.0634 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0266 | 0.3635 | 0.288 |
Echinococcus granulosus | tubulin epsilon chain | 0.0258 | 0.3496 | 0.3488 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Brugia malayi | Probable ClpP-like protease | 0.0075 | 0.0442 | 0.0442 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0266 | 0.3635 | 0.288 |
Trypanosoma brucei | epsilon tubulin | 0.0258 | 0.3496 | 0.2724 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0266 | 0.3635 | 0.3628 |
Wolbachia endosymbiont of Brugia malayi | cell division protein FtsZ | 0.0112 | 0.1061 | 1 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0258 | 0.3496 | 0.2724 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0266 | 0.3635 | 0.3635 |
Schistosoma mansoni | tubulin subunit delta | 0.0112 | 0.1061 | 0.0647 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0146 | 0.1627 | 0.0634 |
Mycobacterium tuberculosis | Cell division protein FtsZ | 0.0112 | 0.1061 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0146 | 0.1627 | 0.0634 |
Echinococcus granulosus | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0266 | 0.3635 | 0.3628 |
Trypanosoma brucei | beta tubulin | 0.0258 | 0.3496 | 0.2724 |
Trypanosoma brucei | tubulin gamma chain | 0.0258 | 0.3496 | 0.2724 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0154 | 0.1767 | 0.079 |
Schistosoma mansoni | tubulin subunit alpha | 0.0266 | 0.3635 | 0.3341 |
Brugia malayi | Tubulin beta chain | 0.0146 | 0.1627 | 0.1627 |
Brugia malayi | Tubulin alpha chain | 0.0266 | 0.3635 | 0.3635 |
Treponema pallidum | cell division protein FtsZ | 0.0112 | 0.1061 | 1 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0258 | 0.3496 | 0.2724 |
Schistosoma mansoni | alpha tubulin | 0.0266 | 0.3635 | 0.3341 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0266 | 0.3635 | 0.3628 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0258 | 0.3496 | 0.2724 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0266 | 0.3635 | 0.0214 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0266 | 0.3635 | 0.3628 |
Loa Loa (eye worm) | hypothetical protein | 0.012 | 0.12 | 0.12 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0258 | 0.3496 | 0.2724 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0266 | 0.3635 | 0.3628 |
Chlamydia trachomatis | ATP-dependent Clp protease proteolytic subunit | 0.0075 | 0.0442 | 0.5 |
Plasmodium vivax | tubulin gamma chain, putative | 0.0258 | 0.3496 | 0.3195 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0266 | 0.3635 | 0.288 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0266 | 0.3635 | 0.3628 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0266 | 0.3635 | 0.288 |
Mycobacterium leprae | cell division protein FtsZ | 0.0112 | 0.1061 | 1 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Schistosoma mansoni | tubulin subunit beta | 0.0112 | 0.1061 | 0.0647 |
Echinococcus granulosus | tubulin subunit TubB | 0.0266 | 0.3635 | 0.3628 |
Toxoplasma gondii | tubulin/FtsZ family, GTPase domain-containing protein | 0.0112 | 0.1061 | 0.0647 |
Echinococcus granulosus | tubulin gamma 1 chain | 0.0258 | 0.3496 | 0.3488 |
Trypanosoma brucei | epsilon tubulin | 0.0258 | 0.3496 | 0.2724 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0266 | 0.3635 | 0.3628 |
Plasmodium falciparum | tubulin gamma chain | 0.0258 | 0.3496 | 0.3195 |
Echinococcus multilocularis | tubulin alpha | 0.0258 | 0.3496 | 0.3488 |
Plasmodium falciparum | tubulin epsilon chain, putative | 0.0258 | 0.3496 | 0.3195 |
Mycobacterium ulcerans | cell division protein FtsZ | 0.0112 | 0.1061 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Trypanosoma cruzi | tubulin gamma chain | 0.0258 | 0.3496 | 0.2724 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0266 | 0.3635 | 0.3341 |
Loa Loa (eye worm) | hypothetical protein | 0.0154 | 0.1767 | 0.1767 |
Trypanosoma brucei | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Echinococcus multilocularis | ATP dependent Clp protease proteolytic subunit | 0.0075 | 0.0442 | 0.0431 |
Plasmodium vivax | delta tubulin, putative | 0.0112 | 0.1061 | 0.0647 |
Brugia malayi | Tubulin alpha-2 chain | 0.0266 | 0.3635 | 0.3635 |
Brugia malayi | Tubulin alpha-2 chain | 0.0266 | 0.3635 | 0.3635 |
Schistosoma mansoni | alpha tubulin | 0.0266 | 0.3635 | 0.3341 |
Giardia lamblia | Alpha-tubulin | 0.0266 | 0.3635 | 0.288 |
Schistosoma mansoni | tubulin subunit alpha | 0.0266 | 0.3635 | 0.3341 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Leishmania major | gamma-tubulin | 0.0258 | 0.3496 | 0.2724 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Plasmodium vivax | tubulin epsilon chain, putative | 0.0258 | 0.3496 | 0.3195 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0266 | 0.3635 | 0.3628 |
Trypanosoma brucei | alpha tubulin, putative | 0.0146 | 0.1627 | 0.0634 |
Brugia malayi | tubulin alpha-2 chain | 0.0266 | 0.3635 | 0.3635 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0266 | 0.3635 | 0.288 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0266 | 0.3635 | 0.3628 |
Trypanosoma brucei | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0266 | 0.3635 | 0.3635 |
Onchocerca volvulus | 0.0146 | 0.1627 | 0.5 | |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0266 | 0.3635 | 0.288 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0154 | 0.1767 | 0.1767 |
Echinococcus granulosus | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0154 | 0.1767 | 0.1767 |
Echinococcus multilocularis | tubulin alpha chain | 0.0266 | 0.3635 | 0.3628 |
Chlamydia trachomatis | ATP-dependent Clp protease proteolytic subunit | 0.0075 | 0.0442 | 0.5 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0258 | 0.3496 | 0.3496 |
Echinococcus granulosus | ATP dependent Clp protease proteolytic subunit | 0.0075 | 0.0442 | 0.0431 |
Echinococcus multilocularis | tubulin delta chain | 0.0112 | 0.1061 | 0.1051 |
Plasmodium falciparum | alpha tubulin 2 | 0.0266 | 0.3635 | 0.3341 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0266 | 0.3635 | 0.3628 |
Leishmania major | alpha tubulin | 0.0266 | 0.3635 | 0.288 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | = 50 ug ml-1 | Antibacterial activity against Escherichia coli MTCC 443 after 24 hrs by serial broth dilution method | ChEMBL. | 23058887 |
MIC (functional) | = 500 ug ml-1 | Antifungal activity against Candida albicans MTCC 227 after 48 hrs by serial broth dilution method | ChEMBL. | 23058887 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.