Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | adenosine A3 receptor | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | alpha-tubulin | 0.0194 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0194 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0194 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0194 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0194 | 0.5571 | 0.5571 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0194 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0194 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0194 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.5571 | 0.5571 |
Schistosoma mansoni | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0194 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.5571 | 0.5571 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0139 | 0.1672 | 0.1672 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | hypothetical protein | 0.0134 | 0.1296 | 0.1296 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.1296 | 0.1296 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0134 | 0.1296 | 0.1296 |
Echinococcus multilocularis | hypothetical protein | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0194 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0139 | 0.1672 | 0.1672 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0194 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0139 | 0.1672 | 0.1672 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0194 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0194 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0139 | 0.1672 | 0.1672 |
Brugia malayi | Tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0194 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0194 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0134 | 0.1296 | 0.1296 |
Giardia lamblia | Alpha-tubulin | 0.0194 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0194 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0194 | 0.5571 | 0.5571 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0194 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0194 | 0.5571 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0194 | 0.5571 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 1 % | Inhibition of human A2B adenosine receptor transfected in CHO cells assessed as inhibition of NECA-induced cyclic AMP production at 1 uM after 10 mins by competitive protein binding assay | ChEMBL. | 23427825 |
Inhibition (binding) | = 1 % | Displacement of [3H]ZM241385 from human A2A adenosine receptor expressed in CHO cells at 1 uM after 60 mins by scintillation counting analysis | ChEMBL. | 23427825 |
Inhibition (binding) | = 12 % | Displacement of [3H]DPCPX from human A1 adenosine receptor expressed in CHO cells at 1 uM after 120 mins by scintillation counting analysis | ChEMBL. | 23427825 |
Ki (binding) | = 5.3 nM | Displacement of [125I]AB-MECA from human A3 adenosine receptor expressed in CHO cells after 60 mins by scintillation counting analysis | ChEMBL. | 23427825 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.