Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Vaccinia virus (strain Copenhagen) (VACV) | Uracil-DNA glycosylase | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.019 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0131 | 0.3094 | 0.3094 |
Echinococcus granulosus | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.019 | 0.6486 | 0.5571 |
Trypanosoma brucei | epsilon tubulin | 0.0136 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.019 | 0.6486 | 0.6486 |
Plasmodium vivax | tubulin alpha chain, putative | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0136 | 0.3392 | 0.1672 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.019 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0113 | 0.2066 | 0.2066 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.019 | 0.6486 | 0.6486 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.019 | 0.6486 | 0.5571 |
Brugia malayi | tubulin alpha chain - mouse | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.019 | 0.6486 | 0.5571 |
Brugia malayi | alpha-tubulin | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0131 | 0.3094 | 0.1296 |
Schistosoma mansoni | tubulin subunit alpha | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.019 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0131 | 0.3094 | 0.1296 |
Trypanosoma brucei | epsilon tubulin | 0.0136 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0136 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0131 | 0.3094 | 0.1296 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.019 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.019 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.019 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0136 | 0.3392 | 0.3392 |
Brugia malayi | Tubulin gamma chain | 0.0136 | 0.3392 | 0.3392 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.019 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.019 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0136 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | hypothetical protein | 0.0131 | 0.3094 | 0.1296 |
Trypanosoma cruzi | alpha tubulin, putative | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.019 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.019 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0136 | 0.3392 | 0.3392 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.019 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.019 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.019 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.019 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.019 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 10000 nM | Viral Plaque Reduction Assay | BINDINGDB. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.