Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | chemokine (C-C motif) receptor 1 | Starlite/ChEMBL | References |
Species | Potential target | Known druggable target | Length | Alignment span | Identity |
---|---|---|---|---|---|
Brugia malayi | hypothetical protein | chemokine (C-C motif) receptor 1 | 355 aa | 289 aa | 21.8 % |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Brugia malayi | tubulin alpha chain - mouse | 0.0195 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0195 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | hypothetical protein | 0.0134 | 0.1296 | 0.1296 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0195 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0195 | 0.5571 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0195 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0195 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0195 | 0.5571 | 0.5571 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0195 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0195 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0195 | 0.5571 | 0.5571 |
Trypanosoma brucei | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0195 | 0.5571 | 0.5571 |
Giardia lamblia | Alpha-tubulin | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0195 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0195 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0195 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0195 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0195 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0195 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0195 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0195 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0195 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0195 | 0.5571 | 0.5571 |
Brugia malayi | alpha-tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0134 | 0.1296 | 0.1296 |
Schistosoma mansoni | tubulin subunit alpha | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0195 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0134 | 0.1296 | 0.1296 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0195 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0195 | 0.5571 | 0.5571 |
Brugia malayi | tubulin alpha-2 chain | 0.0195 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0139 | 0.1672 | 0.1672 |
Plasmodium falciparum | alpha tubulin 1 | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0195 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0139 | 0.1672 | 0.1672 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0195 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0195 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0195 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0195 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.1296 | 0.1296 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0195 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0195 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0195 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0139 | 0.1672 | 0.1672 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0195 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0139 | 0.1672 | 0.1672 |
Leishmania major | alpha tubulin | 0.0195 | 0.5571 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 3650 nM | Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cells | ChEMBL. | 23374868 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.