Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0174 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.012 | 0.3094 | 0.1296 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0174 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0125 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0174 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0125 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0125 | 0.3392 | 0.3392 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0174 | 0.6486 | 0.6486 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0174 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0125 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0174 | 0.6486 | 0.5571 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0125 | 0.3392 | 0.1672 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0174 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0125 | 0.3392 | 0.3392 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0174 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0174 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0174 | 0.6486 | 0.6486 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0174 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0125 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0174 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0174 | 0.6486 | 0.5571 |
Trypanosoma brucei | epsilon tubulin | 0.0125 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0174 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0174 | 0.6486 | 0.6486 |
Brugia malayi | tubulin alpha-2 chain | 0.0174 | 0.6486 | 0.6486 |
Trypanosoma brucei | tubulin gamma chain | 0.0125 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0174 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | hypothetical protein | 0.012 | 0.3094 | 0.1296 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0174 | 0.6486 | 0.6486 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0174 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0174 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | alpha-tubulin | 0.0174 | 0.6486 | 0.5571 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0174 | 0.6486 | 0.6486 |
Plasmodium falciparum | alpha tubulin 2 | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0103 | 0.2066 | 0.2066 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0174 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0174 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0174 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.012 | 0.3094 | 0.1296 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0174 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0174 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0174 | 0.6486 | 0.6486 |
Schistosoma mansoni | tubulin subunit alpha | 0.0174 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0174 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0174 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0174 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0125 | 0.3392 | 0.3392 |
Trypanosoma brucei | alpha tubulin | 0.0174 | 0.6486 | 0.6486 |
Brugia malayi | Tubulin alpha chain | 0.0174 | 0.6486 | 0.6486 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0174 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0174 | 0.6486 | 0.6486 |
Echinococcus granulosus | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0174 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.012 | 0.3094 | 0.1296 |
Brugia malayi | alpha-tubulin | 0.0174 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0174 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0174 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0174 | 0.6486 | 0.5571 |
Plasmodium falciparum | alpha tubulin 1 | 0.0174 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0174 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.012 | 0.3094 | 0.3094 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0174 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 6 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.