Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0183 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0183 | 0.6486 | 0.6486 |
Trypanosoma brucei | epsilon tubulin | 0.0131 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0183 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0126 | 0.3094 | 0.1296 |
Trypanosoma brucei | epsilon tubulin | 0.0131 | 0.3392 | 0.3392 |
Schistosoma mansoni | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0126 | 0.3094 | 0.3094 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0109 | 0.2066 | 0.2066 |
Brugia malayi | Tubulin alpha-2 chain | 0.0183 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0183 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin subunit TubB | 0.0183 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0183 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0131 | 0.3392 | 0.3392 |
Echinococcus multilocularis | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0183 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0131 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | alpha-tubulin | 0.0183 | 0.6486 | 0.5571 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0183 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0131 | 0.3392 | 0.3392 |
Brugia malayi | alpha-tubulin | 0.0183 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0183 | 0.6486 | 0.5571 |
Loa Loa (eye worm) | hypothetical protein | 0.0183 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0126 | 0.3094 | 0.1296 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0183 | 0.6486 | 0.5571 |
Giardia lamblia | Alpha-tubulin | 0.0183 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0131 | 0.3392 | 0.1672 |
Echinococcus granulosus | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0183 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0131 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0183 | 0.6486 | 0.6486 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0183 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0183 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0183 | 0.6486 | 0.6486 |
Echinococcus multilocularis | hypothetical protein | 0.0183 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0183 | 0.6486 | 0.6486 |
Schistosoma mansoni | tubulin subunit alpha | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0131 | 0.3392 | 0.3392 |
Brugia malayi | Tubulin alpha-2 chain | 0.0183 | 0.6486 | 0.6486 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0183 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0131 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0126 | 0.3094 | 0.1296 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0126 | 0.3094 | 0.1296 |
Brugia malayi | tubulin alpha chain - mouse | 0.0183 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0183 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0183 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0183 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0183 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0183 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0183 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0183 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0131 | 0.3392 | 0.3392 |
Schistosoma mansoni | tubulin subunit alpha | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0183 | 0.6486 | 0.6486 |
Giardia lamblia | Alpha-tubulin | 0.0183 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0183 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0183 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0183 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0183 | 0.6486 | 0.5571 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0183 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0183 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 6 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.