Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | sodium channel, voltage-gated, type IX, alpha subunit | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.3094 | 0.1296 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0194 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0134 | 0.3094 | 0.1296 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0139 | 0.3392 | 0.3392 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.6486 | 0.6486 |
Brugia malayi | Tubulin alpha-2 chain | 0.0194 | 0.6486 | 0.6486 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0194 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin gamma chain | 0.0139 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0194 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.6486 | 0.6486 |
Brugia malayi | tubulin alpha-2 chain | 0.0194 | 0.6486 | 0.6486 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0194 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0194 | 0.6486 | 0.6486 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0139 | 0.3392 | 0.1672 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0139 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0194 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0194 | 0.6486 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.6486 | 0.6486 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0194 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.6486 | 0.6486 |
Giardia lamblia | Alpha-tubulin | 0.0194 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0194 | 0.6486 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0194 | 0.6486 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0139 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0194 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0194 | 0.6486 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0194 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0194 | 0.6486 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0194 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0194 | 0.6486 | 0.4682 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0194 | 0.6486 | 0.6486 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0139 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.6486 | 0.6486 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0194 | 0.6486 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0194 | 0.6486 | 0.6486 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0194 | 0.6486 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0194 | 0.6486 | 0.6486 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0134 | 0.3094 | 0.3094 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0116 | 0.2066 | 0.2066 |
Echinococcus multilocularis | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0139 | 0.3392 | 0.3392 |
Loa Loa (eye worm) | hypothetical protein | 0.0134 | 0.3094 | 0.1296 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0194 | 0.6486 | 0.4682 |
Trypanosoma brucei | epsilon tubulin | 0.0139 | 0.3392 | 0.3392 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0194 | 0.6486 | 0.6486 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0194 | 0.6486 | 0.6486 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0194 | 0.6486 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.3094 | 0.1296 |
Plasmodium falciparum | alpha tubulin 1 | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0194 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0194 | 0.6486 | 0.5571 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0194 | 0.6486 | 0.6486 |
Echinococcus granulosus | tubulin alpha chain | 0.0194 | 0.6486 | 0.4682 |
Trypanosoma brucei | tubulin gamma chain | 0.0139 | 0.3392 | 0.3392 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0194 | 0.6486 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0194 | 0.6486 | 0.4682 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0194 | 0.6486 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0194 | 0.6486 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0194 | 0.6486 | 0.5571 |
Trypanosoma brucei | epsilon tubulin | 0.0139 | 0.3392 | 0.3392 |
Leishmania major | alpha tubulin | 0.0194 | 0.6486 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 7.8239 | Inhibition of NaV1.7 ion channel (unknown origin) | ChEMBL. | 23177785 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.