Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0128 | 0.1672 | 0.1672 |
Giardia lamblia | Alpha-tubulin | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0123 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0123 | 0.1296 | 0.1296 |
Echinococcus multilocularis | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0179 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0179 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0179 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0179 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0179 | 0.5571 | 0.5571 |
Trypanosoma brucei | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0179 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0179 | 0.5571 | 0.5571 |
Brugia malayi | Tubulin alpha-2 chain | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0128 | 0.1672 | 0.1672 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0123 | 0.1296 | 0.1296 |
Schistosoma mansoni | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0179 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0179 | 0.5571 | 0.5571 |
Brugia malayi | Tubulin alpha-2 chain | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0179 | 0.5571 | 0.5571 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0179 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0128 | 0.1672 | 0.1672 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0179 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0128 | 0.1672 | 0.1672 |
Plasmodium falciparum | alpha tubulin 2 | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0179 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0179 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0179 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0179 | 0.5571 | 0.5571 |
Plasmodium falciparum | alpha tubulin 1 | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0179 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0179 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0179 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0179 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0123 | 0.1296 | 0.1296 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0179 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0123 | 0.1296 | 0.1296 |
Trypanosoma brucei | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0179 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0179 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0179 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0179 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0179 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0179 | 0.5571 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0179 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0179 | 0.5571 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 86.34 uM | Inhibition of human recombinant PARP1 after 1 hr by ELISA | ChEMBL. | 23473053 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.