Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | alpha-tubulin | 0.0383 | 0.4774 | 0.4774 |
Schistosoma mansoni | tubulin subunit alpha | 0.0383 | 0.4774 | 0.3517 |
Giardia lamblia | Alpha-tubulin | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | tubulin subunit alpha | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | Tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.3517 |
Giardia lamblia | Alpha-tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | hypothetical protein | 0.0383 | 0.4774 | 0.4774 |
Schistosoma mansoni | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin subunit TubB | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.4774 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | hypothetical protein | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0383 | 0.4774 | 0.3517 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Loa Loa (eye worm) | hypothetical protein | 0.0259 | 0.111 | 0.111 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | Tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | tubulin alpha chain - mouse | 0.0383 | 0.4774 | 0.3517 |
Brugia malayi | Tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0259 | 0.111 | 0.111 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0287 | 0.1939 | 0.1939 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0383 | 0.4774 | 0.4774 |
Plasmodium falciparum | alpha tubulin 2 | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0287 | 0.1939 | 0.1939 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0259 | 0.111 | 0.111 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0287 | 0.1939 | 0.1939 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0383 | 0.4774 | 0.4774 |
Plasmodium falciparum | alpha tubulin 1 | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Schistosoma mansoni | tubulin subunit alpha | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0259 | 0.111 | 0.111 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0383 | 0.4774 | 0.4774 |
Brugia malayi | tubulin alpha-2 chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0259 | 0.111 | 0.111 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0287 | 0.1939 | 0.1939 |
Echinococcus multilocularis | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0383 | 0.4774 | 0.4774 |
Brugia malayi | alpha-tubulin | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | tubulin alpha chain | 0.0383 | 0.4774 | 0.3517 |
Trypanosoma brucei | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0383 | 0.4774 | 0.3517 |
Leishmania major | alpha tubulin | 0.0383 | 0.4774 | 0.3517 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0383 | 0.4774 | 0.3517 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0383 | 0.4774 | 0.3517 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Loa Loa (eye worm) | alpha-tubulin | 0.0383 | 0.4774 | 0.4774 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0383 | 0.4774 | 0.3517 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0383 | 0.4774 | 0.3517 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 5 uM | Cytotoxicity against mouse J774 cells assessed as cell viability after 72 hrs by Alamar blue assay | ChEMBL. | 23265887 |
Species name | Source | Reference | Is orphan |
---|---|---|---|
Mus musculus | ChEMBL23 | 23265887 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.