Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma brucei | tubulin gamma chain | 0.0029 | 0.0221 | 0.0221 |
Echinococcus granulosus | mitogen activated protein kinase | 0.0585 | 1 | 1 |
Brugia malayi | Tubulin gamma chain | 0.0029 | 0.0221 | 0.0221 |
Leishmania major | mitogen activated protein kinase 4, putative;with=GeneDB:LmxM19.1440 | 0.0585 | 1 | 1 |
Trypanosoma cruzi | mitogen-activated protein kinase 11, putative | 0.0585 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | BEN-1 protein | 0.0029 | 0.0221 | 0.0221 |
Echinococcus multilocularis | mitogen activated protein kinase | 0.0585 | 1 | 1 |
Giardia lamblia | Kinase, CMGC MAPK | 0.0585 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0585 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | alpha-tubulin | 0.0029 | 0.0221 | 0.0221 |
Brugia malayi | Tubulin alpha-2 chain | 0.0029 | 0.0221 | 0.0221 |
Brugia malayi | Tubulin alpha-2 chain | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | epsilon tubulin | 0.0029 | 0.0221 | 0.0221 |
Toxoplasma gondii | CMGC kinase, MAPK family (ERK) MAPK-1 | 0.0585 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0585 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | beta-tubulin | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | beta tubulin | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0585 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0029 | 0.0221 | 0.5 |
Trypanosoma brucei | epsilon tubulin | 0.0029 | 0.0221 | 0.0221 |
Plasmodium falciparum | tubulin gamma chain | 0.0029 | 0.0221 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | epsilon tubulin | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0029 | 0.0221 | 0.0221 |
Brugia malayi | Tubulin beta-1 chain | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | alpha tubulin | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | CMGC/MAPK/ERK1 protein kinase | 0.0585 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma cruzi | mitogen-activated protein kinase 11, putative | 0.0585 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | BEN-1 protein | 0.0029 | 0.0221 | 0.0221 |
Brugia malayi | Tubulin alpha chain | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0029 | 0.0221 | 0.0221 |
Entamoeba histolytica | tubulin family protein | 0.0029 | 0.0221 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | beta tubulin | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Plasmodium vivax | tubulin epsilon chain, putative | 0.0029 | 0.0221 | 0.5 |
Trypanosoma brucei | protein kinase, putative | 0.0585 | 1 | 1 |
Echinococcus multilocularis | mitogen activated protein kinase 3 | 0.0585 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0029 | 0.0221 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0029 | 0.0221 | 0.0221 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0029 | 0.0221 | 0.5 |
Entamoeba histolytica | tubulin gamma chain | 0.0029 | 0.0221 | 0.5 |
Trypanosoma cruzi | mitogen activated protein kinase 2, putative | 0.0585 | 1 | 1 |
Trypanosoma cruzi | mitogen activated protein kinase 4, putative | 0.0585 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Plasmodium falciparum | tubulin epsilon chain, putative | 0.0029 | 0.0221 | 0.5 |
Brugia malayi | tubulin alpha chain - mouse | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | mitogen activated protein kinase 4, putative | 0.0585 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0029 | 0.0221 | 0.0221 |
Plasmodium falciparum | tubulin beta chain | 0.0029 | 0.0221 | 0.5 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0585 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Plasmodium falciparum | alpha tubulin 2 | 0.0029 | 0.0221 | 0.5 |
Trypanosoma brucei | alpha tubulin | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | beta tubulin | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0029 | 0.0221 | 0.0221 |
Plasmodium vivax | tubulin gamma chain, putative | 0.0029 | 0.0221 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0029 | 0.0221 | 0.0221 |
Echinococcus granulosus | mitogen activated protein kinase 3 | 0.0585 | 1 | 1 |
Brugia malayi | tubulin alpha-2 chain | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | alpha tubulin | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0029 | 0.0221 | 0.0221 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0029 | 0.0221 | 0.5 |
Leishmania major | mitogen activated protein kinase, putative,map kinase, putative | 0.0585 | 1 | 1 |
Onchocerca volvulus | 0.0016 | 0 | 0.5 | |
Plasmodium vivax | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.5 |
Plasmodium falciparum | alpha tubulin 1 | 0.0029 | 0.0221 | 0.5 |
Trichomonas vaginalis | tubulin, putative | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | CMGC family protein kinase | 0.0585 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0029 | 0.0221 | 0.0221 |
Trypanosoma brucei | alpha tubulin | 0.0029 | 0.0221 | 0.0221 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0029 | 0.0221 | 0.0221 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0029 | 0.0221 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Activity (functional) | = 26 % | Cytotoxicity against human SKHEP1 cells at 50 uM after 48 hrs by sulforhodamine B assay | ChEMBL. | 23387901 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.