Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | serine/threonine-protein kinase wnk, putative | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | 3'partial|tyrosine protein kinase Fgr | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Onchocerca volvulus | 0.0161 | 1 | 1 | |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Fps85D | 0.0161 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Brugia malayi | Tyrosine-protein kinase abl-1 | 0.0161 | 1 | 1 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase lyn tyrosine protein kinase blk | 0.0161 | 1 | 1 |
Trichomonas vaginalis | STE family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine kinase|tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Echinococcus multilocularis | tyrosine kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Brugia malayi | Protein kinase domain containing protein | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase lyn lyn a protein tyrosine kinase lymphocyte specific protein tyrosine kinase | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Echinococcus granulosus | tyrosine protein kinase Blk | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Plasmodium falciparum | tyrosine kinase-like protein | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase shark | 0.0161 | 1 | 1 |
Echinococcus multilocularis | c src tyrosine kinase | 0.0161 | 1 | 1 |
Trypanosoma brucei | protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Blk | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Onchocerca volvulus | 0.0161 | 1 | 1 | |
Brugia malayi | Protein kinase domain containing protein | 0.0161 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0161 | 1 | 1 |
Toxoplasma gondii | protein kinase | 0.0091 | 0 | 0.5 |
Schistosoma mansoni | tyrosine kinase | 0.0161 | 1 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.0161 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Brugia malayi | protein-tyrosine kinase | 0.0161 | 1 | 1 |
Schistosoma mansoni | proto-oncogene tyrosine-protein kinase src | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Entamoeba histolytica | SH2-protein kinase domain containing protein | 0.0161 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trypanosoma brucei | Pseudokinase, putative | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Fps85D | 0.0161 | 1 | 1 |
Schistosoma mansoni | tyrosine kinase | 0.0161 | 1 | 1 |
Trypanosoma cruzi | protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Toxoplasma gondii | STE kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Echinococcus granulosus | tyrosine protein kinase Lyn | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | CAMK family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Src64B | 0.0161 | 1 | 1 |
Trypanosoma cruzi | protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Schistosoma mansoni | tyrosine kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Plasmodium falciparum | protein kinase, putative | 0.0091 | 0 | 0.5 |
Schistosoma mansoni | tyrosine kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Plasmodium falciparum | protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | ankyrin repeat-containing protein, putative | 0.0091 | 0 | 0.5 |
Trypanosoma brucei | Flagellum attachment zone protein 20 | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | c src tyrosine kinase | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | TK protein kinase | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Onchocerca volvulus | 0.0161 | 1 | 1 | |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Onchocerca volvulus | 0.0161 | 1 | 1 | |
Giardia lamblia | Kinase, NEK | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Abl | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Plasmodium falciparum | protein kinase, putative | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0161 | 1 | 1 |
Giardia lamblia | Protein 21.1 | 0.0091 | 0 | 0.5 |
Onchocerca volvulus | 0.0161 | 1 | 1 | |
Echinococcus granulosus | tyrosine kinase | 0.0161 | 1 | 1 |
Brugia malayi | SRC-1 | 0.0161 | 1 | 1 |
Loa Loa (eye worm) | SRC-1 | 0.0161 | 1 | 1 |
Trichomonas vaginalis | protein kinase atn1, putative | 0.0091 | 0 | 0.5 |
Toxoplasma gondii | Tyrosine kinase-like (TKL) protein | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Btk29A | 0.0161 | 1 | 1 |
Brugia malayi | SH2 domain containing protein | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Toxoplasma gondii | calcium dependent protein kinase CDPK8 | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/ABL protein kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Plasmodium vivax | protein kinase, putative | 0.0091 | 0 | 0.5 |
Trypanosoma cruzi | STE/STE11 serine/threonine-protein kinase, putative | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Fgr | 0.0161 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase ABL1 | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Schistosoma mansoni | tyrosine kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trypanosoma brucei | AGC/RSK family serine/threonine kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | protein tyrosine kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TK family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Srms | 0.0161 | 1 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.0161 | 1 | 1 |
Leishmania major | hypothetical protein, conserved | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Leishmania major | protein kinase, putative | 0.0091 | 0 | 0.5 |
Giardia lamblia | Kinase, NEK | 0.0091 | 0 | 0.5 |
Leishmania major | protein kinase, putative | 0.0091 | 0 | 0.5 |
Plasmodium vivax | tyrosine kinase-like protein, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Plasmodium falciparum | tyrosine kinase-like protein | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Plasmodium vivax | tyrosine kinase-like protein, putative | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine kinase | 0.0161 | 1 | 1 |
Schistosoma mansoni | tyrosine kinase | 0.0161 | 1 | 1 |
Echinococcus granulosus | tyrosine protein kinase ABL1 | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Srms | 0.0161 | 1 | 1 |
Trichomonas vaginalis | br serine/threonine-protein kinase, putative | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | proto oncogene tyrosine protein kinase LCK | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0161 | 1 | 1 |
Onchocerca volvulus | 0.0161 | 1 | 1 | |
Giardia lamblia | Kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Src64B | 0.0161 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase shark | 0.0161 | 1 | 1 |
Trypanosoma cruzi | STE/STE11 serine/threonine-protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trypanosoma brucei | STE/STE11 serine/threonine-protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | serine-threonine protein kinase, putative | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Brugia malayi | hypothetical protein | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | proto oncogene tyrosine protein kinase LCK | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0091 | 0 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Btk29A | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Loa Loa (eye worm) | TK/FER protein kinase | 0.0161 | 1 | 1 |
Toxoplasma gondii | Tyrosine kinase-like (TKL) protein | 0.0091 | 0 | 0.5 |
Brugia malayi | SH2 domain containing protein | 0.0161 | 1 | 1 |
Trichomonas vaginalis | TKL family protein kinase | 0.0091 | 0 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
CC50 (ADMET) | = 35.3 uM | Cytotoxicity against human HeLa cells expressing CD4, CCR5 after 3 days | ChEMBL. | 23200254 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.