Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0835 | 0.0804 | 0.0804 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0519 | 0.0199 | 0.0199 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0834 | 0.0802 | 0.0802 |
Leishmania major | target of rapamycin (TOR) kinase 2, putative | 0.1547 | 0.2167 | 0.2008 |
Loa Loa (eye worm) | CMGC/MAPK/ERK1 protein kinase | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Echinococcus granulosus | FKBP12 rapamycin complex associated protein | 0.1547 | 0.2167 | 0.2008 |
Echinococcus multilocularis | mitogen activated protein kinase 3 | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1231 | 0.1561 | 0.1561 |
Trypanosoma cruzi | mitogen-activated protein kinase 11, putative | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1231 | 0.1561 | 0.1561 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0519 | 0.0199 | 0.0199 |
Trypanosoma brucei | phosphatidylinositol 3-kinase tor, putative | 0.0732 | 0.0606 | 0.0416 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1231 | 0.1561 | 0.1561 |
Entamoeba histolytica | phosphatidylinositol3-kinaseTor2, putative | 0.1547 | 0.2167 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0834 | 0.0802 | 0.0802 |
Trypanosoma brucei | mitogen activated protein kinase 4, putative | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0924 | 0.0975 | 0.0975 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1321 | 0.1734 | 0.1734 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1038 | 0.1192 | 0.1192 |
Leishmania major | mitogen activated protein kinase 4, putative;with=GeneDB:LmxM19.1440 | 0.5639 | 1 | 1 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.1232 | 0.1563 | 0.1392 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm)-related | 0.1547 | 0.2167 | 0.2008 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0835 | 0.0804 | 0.0804 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor2 | 0.1547 | 0.2167 | 0.2008 |
Trypanosoma cruzi | target of rapamycin kinase 3 | 0.1232 | 0.1563 | 0.1392 |
Toxoplasma gondii | CMGC kinase, MAPK family (ERK) MAPK-1 | 0.5639 | 1 | 1 |
Echinococcus granulosus | mitogen activated protein kinase | 0.5639 | 1 | 1 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor1 | 0.1547 | 0.2167 | 0.2008 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0834 | 0.0802 | 0.0802 |
Trypanosoma brucei | protein kinase, putative | 0.5639 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.5639 | 1 | 1 |
Echinococcus multilocularis | mitogen activated protein kinase | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0915 | 0.0957 | 0.0957 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1004 | 0.1128 | 0.1128 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0519 | 0.0199 | 0.0199 |
Trichomonas vaginalis | CMGC family protein kinase | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.1547 | 0.2167 | 0.2008 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0924 | 0.0975 | 0.0975 |
Echinococcus multilocularis | FKBP12 rapamycin complex associated protein | 0.1547 | 0.2167 | 0.2008 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.1547 | 0.2167 | 0.2008 |
Trypanosoma cruzi | mitogen-activated protein kinase 11, putative | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1547 | 0.2167 | 0.2167 |
Schistosoma mansoni | serine/threonine protein kinase | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0519 | 0.0199 | 0.0199 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0924 | 0.0975 | 0.0975 |
Leishmania major | target of rapamycin kinase (TOR) kinase 3 | 0.1232 | 0.1563 | 0.1392 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0835 | 0.0804 | 0.0804 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0519 | 0.0199 | 0.0199 |
Trypanosoma cruzi | mitogen activated protein kinase 2, putative | 0.5639 | 1 | 1 |
Echinococcus granulosus | mitogen activated protein kinase 3 | 0.5639 | 1 | 1 |
Trypanosoma brucei | FAT domain/Rapamycin binding domain/Phosphatidylinositol 3- and 4-kinase, putative | 0.0643 | 0.0435 | 0.0242 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1231 | 0.1561 | 0.1561 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1547 | 0.2167 | 0.2167 |
Giardia lamblia | Kinase, CMGC MAPK | 0.5639 | 1 | 1 |
Trichomonas vaginalis | CMGC family protein kinase | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0835 | 0.0804 | 0.0804 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0915 | 0.0957 | 0.0957 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.1547 | 0.2167 | 0.2008 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1151 | 0.1408 | 0.1408 |
Leishmania major | target of rapamycin (TOR) kinase 1, putative | 0.1547 | 0.2167 | 0.2008 |
Leishmania major | mitogen activated protein kinase, putative,map kinase, putative | 0.5639 | 1 | 1 |
Trypanosoma cruzi | mitogen activated protein kinase 4, putative | 0.5639 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1231 | 0.1561 | 0.1561 |
Trichomonas vaginalis | CMGC family protein kinase | 0.5639 | 1 | 1 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.1547 | 0.2167 | 0.2008 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.1547 | 0.2167 | 0.2167 |
Entamoeba histolytica | FKBP-rapamycin associated protein (FRAP), putative | 0.1547 | 0.2167 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 200 uM | Inhibition of canine platelet-rich plasma agregation induced by ADP | ChEMBL. | 1920361 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.