Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | aldo keto reductase | 0.1677 | 1 | 1 |
Trichomonas vaginalis | chromodomain helicase DNA binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Echinococcus granulosus | neuropeptide receptor A26 | 0.0541 | 0.3206 | 0.3189 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Trichomonas vaginalis | chromodomain-helicase-DNA-binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Leishmania major | aldo-keto reductase-like protein | 0.1677 | 1 | 1 |
Toxoplasma gondii | oxidoreductase, aldo/keto reductase family protein | 0.0486 | 0.2879 | 0.2617 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Plasmodium falciparum | aldehyde reductase, putative | 0.0486 | 0.2879 | 1 |
Toxoplasma gondii | aldehyde dehydrogenase | 0.0071 | 0.04 | 0.0046 |
Loa Loa (eye worm) | N-myristoyltransferase 2 | 0.0375 | 0.2214 | 0.2184 |
Mycobacterium ulcerans | hypothetical protein | 0.0486 | 0.2879 | 0.2583 |
Schistosoma mansoni | pol-related | 0.1677 | 1 | 1 |
Trypanosoma cruzi | aldo/keto reductase, putative | 0.0486 | 0.2879 | 0.0855 |
Loa Loa (eye worm) | hypothetical protein | 0.1677 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.1677 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.1677 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.1677 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Schistosoma mansoni | cpg binding protein | 0.0035 | 0.0188 | 0.0183 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Schistosoma mansoni | potassium channel beta | 0.0486 | 0.2879 | 0.2876 |
Trichomonas vaginalis | chromodomain helicase DNA binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Echinococcus multilocularis | aldo keto reductase | 0.1677 | 1 | 1 |
Trichomonas vaginalis | chromodomain-helicase-DNA-binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Brugia malayi | CXXC zinc finger family protein | 0.0034 | 0.0176 | 0.014 |
Trypanosoma brucei | aldo/keto reductase, putative | 0.0486 | 0.2879 | 0.0855 |
Onchocerca volvulus | 0.1677 | 1 | 1 | |
Loa Loa (eye worm) | oxidoreductase | 0.1677 | 1 | 1 |
Leishmania major | N-myristoyl transferase, putative | 0.0375 | 0.2214 | 0.1889 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Schistosoma mansoni | hypothetical protein | 0.0478 | 0.2833 | 0.283 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Echinococcus granulosus | glycylpeptide N tetradecanoyltransferase | 0.0375 | 0.2214 | 0.2194 |
Plasmodium vivax | aldehyde reductase, putative | 0.0486 | 0.2879 | 1 |
Echinococcus granulosus | hypothetical protein | 0.1677 | 1 | 1 |
Echinococcus multilocularis | glycylpeptide N tetradecanoyltransferase | 0.0375 | 0.2214 | 0.2194 |
Toxoplasma gondii | aldose reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Echinococcus multilocularis | microtubule associated protein 2 | 0.0807 | 0.4796 | 0.4783 |
Onchocerca volvulus | 0.1677 | 1 | 1 | |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.1677 | 1 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.1677 | 1 | 1 |
Echinococcus granulosus | microtubule associated protein 2 | 0.0807 | 0.4796 | 0.4783 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Loa Loa (eye worm) | oxidoreductase | 0.1677 | 1 | 1 |
Mycobacterium leprae | PROBABLE OXIDOREDUCTASE | 0.1677 | 1 | 1 |
Echinococcus granulosus | dnaJ subfamily B | 0.0478 | 0.2833 | 0.2815 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.1677 | 1 | 1 |
Leishmania major | aldehyde reductase, putative,oxidoreductase, putative | 0.1677 | 1 | 1 |
Schistosoma mansoni | mixed-lineage leukemia protein mll | 0.0008 | 0.0025 | 0.0021 |
Loa Loa (eye worm) | oxidoreductase | 0.1677 | 1 | 1 |
Trypanosoma brucei | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | chromodomain helicase DNA binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Schistosoma mansoni | aldehyde dehydrogenase | 0.0071 | 0.04 | 0.0396 |
Echinococcus multilocularis | aldo keto reductase | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0486 | 0.2879 | 0.2879 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Echinococcus granulosus | aldehyde reductase | 0.1192 | 0.7096 | 0.7089 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Trypanosoma cruzi | aldo-keto reductase | 0.1677 | 1 | 1 |
Plasmodium vivax | oxidoreductase, aldo/keto reductase domain containing protein | 0.0486 | 0.2879 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Leishmania major | prostaglandin f synthase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0486 | 0.2879 | 0.2879 |
Schistosoma mansoni | cpg binding protein | 0.0035 | 0.0188 | 0.0183 |
Echinococcus granulosus | neuropeptide s receptor | 0.0541 | 0.3206 | 0.3189 |
Toxoplasma gondii | aldo-keto reductase | 0.0486 | 0.2879 | 0.2617 |
Echinococcus granulosus | cpg binding protein | 0.0035 | 0.0188 | 0.0163 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.1677 | 1 | 1 |
Schistosoma mansoni | cpg binding protein | 0.0034 | 0.0176 | 0.0172 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Schistosoma mansoni | microtubule-associated protein tau | 0.0807 | 0.4796 | 0.4794 |
Plasmodium falciparum | aldo-keto reductase, putative | 0.0486 | 0.2879 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Trypanosoma cruzi | aldo/keto reductase, putative | 0.1677 | 1 | 1 |
Brugia malayi | glutamate-cysteine ligase modifier subunit | 0.0486 | 0.2879 | 0.2853 |
Entamoeba histolytica | aldose reductase, putative | 0.1677 | 1 | 1 |
Schistosoma mansoni | N-myristoyltransferase | 0.0375 | 0.2214 | 0.221 |
Echinococcus granulosus | histone lysine N methyltransferase MLL3 | 0.001 | 0.0038 | 0.0012 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0486 | 0.2879 | 0.2879 |
Trichomonas vaginalis | helicase, putative | 0.0008 | 0.0021 | 0.0021 |
Mycobacterium tuberculosis | Conserved protein | 0.0486 | 0.2879 | 0.2583 |
Toxoplasma gondii | aldo/keto reductase family oxidoreductase | 0.0486 | 0.2879 | 0.2617 |
Echinococcus multilocularis | neuropeptide s receptor | 0.0541 | 0.3206 | 0.3189 |
Trichomonas vaginalis | alcohol dehydrogenase, putative | 0.0486 | 0.2879 | 0.2879 |
Onchocerca volvulus | 0.0486 | 0.2879 | 0.2751 | |
Entamoeba histolytica | alcohol dehydrogenase, putative | 0.0486 | 0.2879 | 0.0855 |
Echinococcus granulosus | aldo keto reductase family 1, member B4 | 0.0486 | 0.2879 | 0.2861 |
Schistosoma mansoni | aldo-keto reductase | 0.1677 | 1 | 1 |
Trichomonas vaginalis | chromodomain helicase DNA binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Leishmania major | prostaglandin f2-alpha synthase/D-arabinose dehydrogenase | 0.1677 | 1 | 1 |
Mycobacterium ulcerans | oxidoreductase | 0.1677 | 1 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.1677 | 1 | 1 |
Echinococcus granulosus | aldehyde dehydrogenase mitochondrial | 0.0071 | 0.04 | 0.0375 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Giardia lamblia | Aldose reductase | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Trichomonas vaginalis | N-myristoyl transferase, putative | 0.0246 | 0.1446 | 0.1446 |
Echinococcus multilocularis | aldehyde reductase | 0.1192 | 0.7096 | 0.7089 |
Echinococcus multilocularis | aldo keto reductase | 0.1677 | 1 | 1 |
Schistosoma mansoni | mixed-lineage leukemia protein mll | 0.0071 | 0.0401 | 0.0397 |
Schistosoma mansoni | aldo-keto reductase | 0.1677 | 1 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.1677 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Echinococcus granulosus | voltage gated potassium channel subunit | 0.0486 | 0.2879 | 0.2861 |
Brugia malayi | NADH-dependent xylose reductase | 0.0486 | 0.2879 | 0.2853 |
Entamoeba histolytica | alcohol dehydrogenase, putative | 0.0486 | 0.2879 | 0.0855 |
Mycobacterium leprae | Conserved hypothetical protein | 0.1192 | 0.7096 | 0.5922 |
Onchocerca volvulus | 0.1677 | 1 | 1 | |
Loa Loa (eye worm) | oxidoreductase | 0.1677 | 1 | 1 |
Echinococcus multilocularis | voltage gated potassium channel subunit | 0.0486 | 0.2879 | 0.2861 |
Brugia malayi | N-myristoyltransferase 2 | 0.0375 | 0.2214 | 0.2185 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0486 | 0.2879 | 0.2879 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.1677 | 1 | 1 |
Onchocerca volvulus | 0.1677 | 1 | 1 | |
Loa Loa (eye worm) | CXXC zinc finger family protein | 0.0034 | 0.0176 | 0.0139 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Echinococcus multilocularis | histone lysine N methyltransferase MLL3 | 0.001 | 0.0038 | 0.0012 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Onchocerca volvulus | 0.1677 | 1 | 1 | |
Trichomonas vaginalis | chromodomain helicase DNA binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Entamoeba histolytica | aldose reductase, putative | 0.1677 | 1 | 1 |
Trichomonas vaginalis | N-myristoyl transferase, putative | 0.0375 | 0.2214 | 0.2214 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0008 | 0.0021 | 0.0021 |
Loa Loa (eye worm) | glutamate-cysteine ligase modifier subunit | 0.0486 | 0.2879 | 0.2852 |
Echinococcus multilocularis | dnaJ subfamily B | 0.0478 | 0.2833 | 0.2815 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.1677 | 1 | 1 |
Onchocerca volvulus | 0.1677 | 1 | 1 | |
Giardia lamblia | Aldose reductase | 0.1677 | 1 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.1677 | 1 | 1 |
Echinococcus multilocularis | neuropeptide receptor A26 | 0.0541 | 0.3206 | 0.3189 |
Echinococcus multilocularis | aldehyde dehydrogenase, mitochondrial | 0.0071 | 0.04 | 0.0375 |
Schistosoma mansoni | aldehyde dehydrogenase | 0.0071 | 0.04 | 0.0396 |
Leishmania major | aldo/keto reductase, putative,aldo/keto reductase family-like protein | 0.0486 | 0.2879 | 0.2583 |
Trichomonas vaginalis | chromodomain helicase DNA binding protein, putative | 0.0008 | 0.0021 | 0.0021 |
Trypanosoma brucei | prostaglandin f synthase | 0.1677 | 1 | 1 |
Echinococcus multilocularis | cpg binding protein | 0.0035 | 0.0188 | 0.0163 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.1677 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 0 % | Inhibitory activity against partially purified rat liver HMG CoA reductase at 2 ug/ml concentration | ChEMBL. | 3973903 |
Inhibition (binding) | = 2 % | Inhibitory activity against partially purified rat liver HMG CoA reductase at 4 ug/ml concentration | ChEMBL. | 3973903 |
Inhibition (binding) | = 4 % | Inhibitory activity of the compound against partially purified rat liver HMG CoA reductase at 6 ug/ml concentration | ChEMBL. | 3973903 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.