Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma brucei | serine/threonine-protein kinase NrkA | 0.0194 | 0.0074 | 0.0074 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.1863 | 0.3145 | 0.4731 |
Echinococcus granulosus | NDR protein kinase | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma brucei | NEK family Serine/threonine-protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.3614 | 0.6365 | 0.9576 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.1863 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Echinococcus granulosus | protein kinase C gamma type | 0.1863 | 0.3145 | 0.4731 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.1863 | 0.3145 | 0.4731 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0194 | 0.0074 | 0.0111 |
Trypanosoma brucei | protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0194 | 0.0074 | 0.0111 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.5591 | 1 | 1 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.0194 | 0.0074 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.3768 | 0.6647 | 1 |
Onchocerca volvulus | Abnormal cell migration protein 10 homolog | 0.0153 | 0 | 0.5 |
Entamoeba histolytica | p21-activated kinase | 0.0194 | 0.0074 | 0.0074 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.3574 | 0.6291 | 0.9465 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.3614 | 0.6365 | 0.9576 |
Plasmodium falciparum | calcium-dependent protein kinase 7 | 0.0194 | 0.0074 | 0.0116 |
Loa Loa (eye worm) | hypothetical protein | 0.1863 | 0.3145 | 0.3145 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.1863 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | 3-phosphoinositide dependent protein kinase-1, putative | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0194 | 0.0074 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.5438 | 0.9718 | 0.9718 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.3614 | 0.6365 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | ribosomal protein S6 kinase, 90kD, polypeptide, putative | 0.0194 | 0.0074 | 0.0074 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.3574 | 0.6291 | 0.9465 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.1863 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.1863 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.1863 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Echinococcus multilocularis | serine threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma cruzi | serine/threonine-protein kinase NRKB, putative | 0.0194 | 0.0074 | 0.0111 |
Trypanosoma cruzi | NEK family Serine/threonine-protein kinase, putative | 0.0194 | 0.0074 | 0.0111 |
Echinococcus multilocularis | nervana 2 | 0.3574 | 0.6291 | 0.9465 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0194 | 0.0074 | 0.0111 |
Entamoeba histolytica | protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Leishmania major | folate/biopterin transporter, putative | 0.0194 | 0.0074 | 1 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.1863 | 0.3145 | 0.4731 |
Entamoeba histolytica | protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.5591 | 1 | 1 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Echinococcus granulosus | nervana 2 | 0.3574 | 0.6291 | 0.9465 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0194 | 0.0074 | 0.0076 |
Entamoeba histolytica | protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0194 | 0.0074 | 0.0111 |
Trypanosoma cruzi | serine/threonine protein kinase, putative | 0.0194 | 0.0074 | 0.0111 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative | 0.0194 | 0.0074 | 1 |
Trypanosoma brucei | Serine/threonine-protein kinase NEK21, putative | 0.0194 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative | 0.0194 | 0.0074 | 1 |
Onchocerca volvulus | Protein melted homolog | 0.0153 | 0 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.3574 | 0.6291 | 0.9465 |
Onchocerca volvulus | Putative neuronal RhoA GEF protein | 0.0153 | 0 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.1863 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.1863 | 0.3145 | 0.4731 |
Entamoeba histolytica | protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Brugia malayi | Hr1 repeat family protein | 0.1863 | 0.3145 | 0.3145 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.3768 | 0.6647 | 0.6647 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma cruzi | Protein kinase B | 0.3768 | 0.6647 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Echinococcus multilocularis | nervana 2 | 0.3574 | 0.6291 | 0.9465 |
Trichomonas vaginalis | AGC family protein kinase | 0.1863 | 0.3145 | 0.3145 |
Toxoplasma gondii | calcium dependent protein kinase CDPK7 | 0.0194 | 0.0074 | 0.0076 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0194 | 0.0074 | 0.0111 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.3614 | 0.6365 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Toxoplasma gondii | AGC kinase | 0.5438 | 0.9718 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.5438 | 0.9718 | 0.9718 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.3768 | 0.6647 | 0.6647 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Entamoeba histolytica | hypothetical protein | 0.0194 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.1863 | 0.3145 | 0.3145 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.1863 | 0.3145 | 0.4731 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.3574 | 0.6291 | 0.9465 |
Echinococcus multilocularis | protein kinase c iota type | 0.1863 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.1863 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.1863 | 0.3145 | 0.3145 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.5438 | 0.9718 | 0.9718 |
Onchocerca volvulus | outspread protein homolog | 0.0153 | 0 | 0.5 |
Echinococcus granulosus | protein kinase c iota type | 0.1863 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Brugia malayi | Protein kinase domain containing protein | 0.1863 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.2017 | 0.3427 | 0.3427 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.3614 | 0.6365 | 0.9576 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.1823 | 0.3071 | 0.3071 |
Brugia malayi | Protein kinase domain containing protein | 0.1863 | 0.3145 | 0.3145 |
Schistosoma mansoni | serine/threonine kinase | 0.1863 | 0.3145 | 0.4731 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.1863 | 0.3145 | 0.3145 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.1863 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.3768 | 0.6647 | 1 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.3614 | 0.6365 | 0.9576 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.1863 | 0.3145 | 0.3145 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.5591 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Echinococcus granulosus | protein kinase c epsilon type | 0.1863 | 0.3145 | 0.4731 |
Trypanosoma brucei | serine/threonine-protein kinase NRKB, putative | 0.0194 | 0.0074 | 0.0074 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.1863 | 0.3145 | 0.4731 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.5591 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.5591 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.0194 | 0.0074 | 1 |
Echinococcus granulosus | serine/threonine protein kinase | 0.3768 | 0.6647 | 1 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0194 | 0.0074 | 0.0111 |
Brugia malayi | protein kinase C II. | 0.1863 | 0.3145 | 0.3145 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Onchocerca volvulus | Putative zinc finger protein | 0.0153 | 0 | 0.5 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.0194 | 0.0074 | 1 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.1863 | 0.3145 | 0.4731 |
Entamoeba histolytica | protein kinase, putative | 0.0194 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase 2, putative | 0.3614 | 0.6365 | 0.6365 |
Giardia lamblia | Kinase, AGC PKA | 0.3614 | 0.6365 | 0.5 |
Schistosoma mansoni | atypical protein kinase C | 0.1863 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Echinococcus granulosus | nervana 2 | 0.3574 | 0.6291 | 0.9465 |
Entamoeba histolytica | hypothetical protein | 0.0194 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.3768 | 0.6647 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1863 | 0.3145 | 0.4731 |
Plasmodium vivax | calcium-dependent protein kinase 7, putative | 0.0194 | 0.0074 | 0.0116 |
Trichomonas vaginalis | AGC family protein kinase | 0.0194 | 0.0074 | 0.0074 |
Onchocerca volvulus | 0.0153 | 0 | 0.5 | |
Echinococcus multilocularis | rac serine:threonine kinase | 0.3768 | 0.6647 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | 39.8107 uM | PubChem BioAssay. qHTS for Antagonist of cAMP-regulated guanine nucleotide exchange factor 2 (EPAC2): primary screen. (Class of assay: confirmatory) | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.