Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Brugia malayi | Serotonin receptor | 0.0507 | 0.0082 | 0.0082 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Onchocerca volvulus | Putative neuronal RhoA GEF protein | 0.0393 | 0 | 0.5 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.0496 | 0.0074 | 1 |
Entamoeba histolytica | protein kinase 2, putative | 0.9261 | 0.6365 | 0.6365 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.4775 | 0.3145 | 0.3145 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 1.4326 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Echinococcus granulosus | protein kinase c iota type | 0.4775 | 0.3145 | 0.4731 |
Loa Loa (eye worm) | hypothetical protein | 0.0669 | 0.0198 | 0.0198 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.4671 | 0.3071 | 0.3071 |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Echinococcus multilocularis | serine threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.4775 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.4775 | 0.3145 | 0.4731 |
Entamoeba histolytica | protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Echinococcus granulosus | hypothetical protein | 0.1534 | 0.0819 | 0.1232 |
Trichomonas vaginalis | AGC family protein kinase | 0.4775 | 0.3145 | 0.3145 |
Loa Loa (eye worm) | hypothetical protein | 0.4775 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.5168 | 0.3427 | 0.3427 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.0496 | 0.0074 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Echinococcus granulosus | nervana 2 | 0.9158 | 0.6291 | 0.9464 |
Toxoplasma gondii | calcium dependent protein kinase CDPK7 | 0.0496 | 0.0074 | 0.0076 |
Onchocerca volvulus | Protein melted homolog | 0.0393 | 0 | 0.5 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.4775 | 0.3145 | 0.4731 |
Echinococcus multilocularis | serotonin receptor | 0.0669 | 0.0198 | 0.0298 |
Leishmania major | protein kinase, putative | 0.0496 | 0.0074 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | ribosomal protein S6 kinase, 90kD, polypeptide, putative | 0.0496 | 0.0074 | 0.0074 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.4775 | 0.3145 | 0.4731 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0496 | 0.0074 | 0.0112 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.9654 | 0.6647 | 1 |
Echinococcus multilocularis | serotonin receptor | 0.0669 | 0.0198 | 0.0298 |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Echinococcus granulosus | NDR protein kinase | 0.4775 | 0.3145 | 0.4731 |
Entamoeba histolytica | protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.4775 | 0.3145 | 0.4731 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 1.3933 | 0.9718 | 0.9718 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 1.4326 | 1 | 1 |
Brugia malayi | protein kinase C II. | 0.4775 | 0.3145 | 0.3145 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.4775 | 0.3145 | 0.3145 |
Loa Loa (eye worm) | hypothetical protein | 0.0669 | 0.0198 | 0.0198 |
Entamoeba histolytica | hypothetical protein | 0.0496 | 0.0074 | 0.0074 |
Onchocerca volvulus | Putative zinc finger protein | 0.0393 | 0 | 0.5 |
Echinococcus granulosus | protein kinase C gamma type | 0.4775 | 0.3145 | 0.4731 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.9654 | 0.6647 | 1 |
Entamoeba histolytica | protein kinase, putative | 1.4326 | 1 | 1 |
Echinococcus multilocularis | nervana 2 | 0.9158 | 0.6291 | 0.9464 |
Brugia malayi | Protein kinase domain containing protein | 0.4775 | 0.3145 | 0.3145 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.4775 | 0.3145 | 0.4731 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.4775 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.9654 | 0.6647 | 1 |
Trypanosoma brucei | serine/threonine-protein kinase NRKB, putative | 0.0496 | 0.0074 | 0.0074 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.4775 | 0.3145 | 0.4731 |
Trypanosoma brucei | Serine/threonine-protein kinase NEK21, putative | 0.0496 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 1.3933 | 0.9718 | 0.9718 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Onchocerca volvulus | Abnormal cell migration protein 10 homolog | 0.0393 | 0 | 0.5 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Trichomonas vaginalis | AGC family protein kinase | 0.4775 | 0.3145 | 0.3145 |
Trypanosoma cruzi | serine/threonine protein kinase, putative | 0.0496 | 0.0074 | 0.0112 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.4775 | 0.3145 | 0.4731 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.9261 | 0.6365 | 0.9576 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.9261 | 0.6365 | 0.9576 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | 3-phosphoinositide dependent protein kinase-1, putative | 0.0496 | 0.0074 | 0.0074 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.4775 | 0.3145 | 0.4731 |
Brugia malayi | Protein kinase domain containing protein | 0.4775 | 0.3145 | 0.3145 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.4775 | 0.3145 | 0.4731 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0496 | 0.0074 | 0.0112 |
Plasmodium vivax | calcium-dependent protein kinase 7, putative | 0.0496 | 0.0074 | 0.0116 |
Entamoeba histolytica | hypothetical protein | 0.0496 | 0.0074 | 0.0074 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0496 | 0.0074 | 0.0076 |
Echinococcus granulosus | nervana 2 | 0.9158 | 0.6291 | 0.9464 |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Schistosoma mansoni | biogenic amine (5HT) receptor | 0.0669 | 0.0198 | 0.0298 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.9261 | 0.6365 | 0.9576 |
Trypanosoma cruzi | NEK family Serine/threonine-protein kinase, putative | 0.0496 | 0.0074 | 0.0112 |
Leishmania major | protein kinase, putative | 0.0496 | 0.0074 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.9654 | 0.6647 | 0.6647 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.9158 | 0.6291 | 0.9464 |
Entamoeba histolytica | protein kinase, putative | 0.4775 | 0.3145 | 0.3145 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0496 | 0.0074 | 0.0112 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0496 | 0.0074 | 0.0112 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0496 | 0.0074 | 0.0112 |
Trypanosoma brucei | NEK family Serine/threonine-protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0496 | 0.0074 | 0.0112 |
Onchocerca volvulus | outspread protein homolog | 0.0393 | 0 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Giardia lamblia | Kinase, AGC PKA | 0.9261 | 0.6365 | 0.5 |
Echinococcus multilocularis | nervana 2 | 0.9158 | 0.6291 | 0.9464 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.9654 | 0.6647 | 1 |
Entamoeba histolytica | p21-activated kinase | 0.0496 | 0.0074 | 0.0074 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.9158 | 0.6291 | 0.9464 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0496 | 0.0074 | 0.0112 |
Echinococcus granulosus | biogenic amine 5HT receptor | 0.0669 | 0.0198 | 0.0298 |
Toxoplasma gondii | AGC kinase | 1.3933 | 0.9718 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 1.4326 | 1 | 1 |
Echinococcus granulosus | protein kinase c epsilon type | 0.4775 | 0.3145 | 0.4731 |
Echinococcus multilocularis | conserved hypothetical protein | 0.1503 | 0.0797 | 0.1199 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.4775 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.4775 | 0.3145 | 0.3145 |
Trypanosoma cruzi | Protein kinase B | 0.9654 | 0.6647 | 1 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.9261 | 0.6365 | 1 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.9261 | 0.6365 | 0.9576 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0496 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.4775 | 0.3145 | 0.3145 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Schistosoma mansoni | serine/threonine protein kinase | 0.4775 | 0.3145 | 0.4731 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.4775 | 0.3145 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.4775 | 0.3145 | 0.4731 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Echinococcus granulosus | serine/threonine protein kinase | 0.9654 | 0.6647 | 1 |
Brugia malayi | Hr1 repeat family protein | 0.4775 | 0.3145 | 0.3145 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.0496 | 0.0074 | 1 |
Schistosoma mansoni | atypical protein kinase C | 0.4775 | 0.3145 | 0.4731 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.4775 | 0.3145 | 0.4731 |
Schistosoma mansoni | serine/threonine kinase | 0.4775 | 0.3145 | 0.4731 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.9261 | 0.6365 | 1 |
Trypanosoma brucei | protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Trypanosoma brucei | serine/threonine-protein kinase NrkA | 0.0496 | 0.0074 | 0.0074 |
Plasmodium falciparum | calcium-dependent protein kinase 7 | 0.0496 | 0.0074 | 0.0116 |
Entamoeba histolytica | protein kinase, putative | 0.0496 | 0.0074 | 0.0074 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.9158 | 0.6291 | 0.9464 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.9654 | 0.6647 | 0.6647 |
Trichomonas vaginalis | AGC family protein kinase | 1.4326 | 1 | 1 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.4775 | 0.3145 | 0.4731 |
Brugia malayi | p70 ribosomal S6 kinase beta | 1.3933 | 0.9718 | 0.9718 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.9158 | 0.6291 | 0.9464 |
Onchocerca volvulus | 0.0393 | 0 | 0.5 | |
Leishmania major | folate/biopterin transporter, putative | 0.0496 | 0.0074 | 1 |
Trypanosoma cruzi | serine/threonine-protein kinase NRKB, putative | 0.0496 | 0.0074 | 0.0112 |
Echinococcus multilocularis | protein kinase c iota type | 0.4775 | 0.3145 | 0.4731 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
GI50 (functional) | = 2.7 uM | Cytotoxicity against human U251 cells by MTT assay | ChEMBL. | 23538115 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.