Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | P-glycoprotein 5, putative | 0.0025 | 0.4631 | 0.1711 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0025 | 0.4631 | 0.4631 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0025 | 0.4631 | 0.4631 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0025 | 0.4631 | 0.1711 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.004 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4631 | 0.4631 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Entamoeba histolytica | P-glycoprotein-5 | 0.0025 | 0.4631 | 0.1711 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0015 | 0.1231 | 0.1231 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.4631 | 0.4564 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Entamoeba histolytica | P-glyco protein 6, putative | 0.0025 | 0.4631 | 0.1711 |
Echinococcus granulosus | multidrug resistance associated protein 1 | 0.0021 | 0.3522 | 0.3522 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4631 | 0.4631 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6594 | 0.6594 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0021 | 0.3522 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0025 | 0.4631 | 0.1711 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma brucei | ubiquitin-protein ligase, putative | 0.004 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6594 | 0.6594 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0021 | 0.3522 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6593 | 0.6593 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0015 | 0.1231 | 0.1231 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0021 | 0.3522 | 0.3522 |
Leishmania major | ubiquitin-conjugating enzyme e2, putative | 0.004 | 1 | 1 |
Entamoeba histolytica | P-glycoprotein-2, putative | 0.0025 | 0.4631 | 0.1711 |
Trypanosoma brucei | trans-sialidase, putative | 0.003 | 0.6594 | 0.4742 |
Leishmania major | p-glycoprotein | 0.0025 | 0.4631 | 0.1711 |
Echinococcus multilocularis | multidrug resistance associated protein 1 | 0.0021 | 0.3522 | 0.3522 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Schistosoma mansoni | multidrug resistance protein | 0.0025 | 0.4631 | 0.1711 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.4631 | 0.4564 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6593 | 0.6593 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4631 | 0.4631 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma brucei | trans-sialidase, putative | 0.003 | 0.6594 | 0.4742 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0025 | 0.4631 | 0.4631 |
Chlamydia trachomatis | ABC transporter ATP binding protein/permease | 0.0025 | 0.4631 | 0.5 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0015 | 0.1231 | 0.1231 |
Plasmodium falciparum | ubiquitin-conjugating enzyme E2 N, putative | 0.004 | 1 | 1 |
Trichomonas vaginalis | taga, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma cruzi | multidrug resistance protein E, putative | 0.0021 | 0.3522 | 0.3522 |
Brugia malayi | ABC transporter family protein | 0.0025 | 0.4631 | 0.1711 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0025 | 0.4631 | 0.1711 |
Schistosoma mansoni | multidrug resistance protein | 0.0025 | 0.4631 | 0.1711 |
Echinococcus granulosus | 5'partial|ATP binding cassette sub family B | 0.0024 | 0.4508 | 0.4508 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | abcb9, putative | 0.0025 | 0.4631 | 0.3877 |
Echinococcus granulosus | multidrug resistance associated protein 7 | 0.0021 | 0.3522 | 0.3522 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Brugia malayi | ubiquitin conjugating enzyme protein 13 | 0.004 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.004 | 1 | 1 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.004 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.3522 | 0.3442 |
Giardia lamblia | ABC transporter, putative | 0.0021 | 0.3522 | 1 |
Giardia lamblia | MRP-like ABC transporter | 0.0021 | 0.3522 | 1 |
Mycobacterium tuberculosis | Probable transmembrane multidrug efflux pump | 0.0025 | 0.4631 | 0.5 |
Entamoeba histolytica | ubiquitin-conjugating enzyme family protein | 0.004 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4631 | 0.4631 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6594 | 0.6594 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4631 | 0.4631 |
Echinococcus granulosus | ubiquitin conjugating enzyme E2 N | 0.004 | 1 | 1 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.004 | 1 | 1 |
Trypanosoma brucei | trans-sialidase | 0.003 | 0.6594 | 0.4742 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4631 | 0.4631 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4631 | 0.3877 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0025 | 0.4631 | 0.4631 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Trichomonas vaginalis | abcb9, putative | 0.0025 | 0.4631 | 0.3877 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0021 | 0.3522 | 0.3522 |
Onchocerca volvulus | 0.0025 | 0.4631 | 0.5 | |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Trypanosoma brucei | trans-sialidase, putative | 0.003 | 0.6594 | 0.4742 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0025 | 0.4631 | 0.4631 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.004 | 1 | 1 |
Loa Loa (eye worm) | multidrug resistance protein 3 | 0.0025 | 0.4631 | 0.4564 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Leishmania major | ATP-binding cassette protein subfamily B, member 2, putative | 0.0025 | 0.4631 | 0.1711 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0025 | 0.4631 | 0.1711 |
Loa Loa (eye worm) | ABC transporter transmembrane region family protein | 0.0021 | 0.3522 | 0.3442 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Loa Loa (eye worm) | hypothetical protein | 0.0024 | 0.4508 | 0.444 |
Toxoplasma gondii | ATP-binding cassette transporter ABC.B1 | 0.0025 | 0.4631 | 0.1711 |
Echinococcus multilocularis | ATP binding cassette sub family B | 0.0024 | 0.4508 | 0.4508 |
Trichomonas vaginalis | abcb9, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.004 | 1 | 1 |
Toxoplasma gondii | ubiquitin-conjugating enzyme subfamily protein | 0.004 | 1 | 1 |
Plasmodium vivax | ubiquitin-conjugating enzyme E2 N, putative | 0.004 | 1 | 1 |
Schistosoma mansoni | ubiquitin conjugating enzyme 13 | 0.004 | 1 | 1 |
Brugia malayi | multidrug resistance protein 3 | 0.0025 | 0.4631 | 0.1711 |
Schistosoma mansoni | smdr2 | 0.0025 | 0.4631 | 0.1711 |
Echinococcus multilocularis | ubiquitin conjugating enzyme E2 N | 0.004 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4631 | 0.4631 |
Entamoeba histolytica | P-glycoprotein-1 | 0.0025 | 0.4631 | 0.1711 |
Loa Loa (eye worm) | ATP-binding cassette sub-family B member 2 | 0.0025 | 0.4631 | 0.4564 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4631 | 0.4631 |
Echinococcus multilocularis | multidrug resistance associated protein 7 | 0.0021 | 0.3522 | 0.3522 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6593 | 0.6593 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.3522 | 0.3442 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.34 | 0.3317 |
Trypanosoma cruzi | trans-sialidase, putative | 0.003 | 0.6593 | 0.6593 |
Trypanosoma brucei | trans-sialidase, putative | 0.003 | 0.6594 | 0.4742 |
Trypanosoma brucei | trans-sialidase, putative | 0.003 | 0.6594 | 0.4742 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.003 | 0.6594 | 0.6594 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0025 | 0.4631 | 0.3877 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4631 | 0.3877 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4631 | 0.4631 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | > 64 ug ml-1 | Antibacterial activity against Escherichia coli ATCC 25922 assessed as growth inhibition after 16 to 18 hr NCCLS agar dilution method | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.