Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Onchocerca volvulus | 0.0031 | 1 | 0.5 | |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Trypanosoma brucei | unspecified product | 0.0021 | 0.4091 | 0.4091 |
Giardia lamblia | Aldose reductase | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0031 | 1 | 1 |
Leishmania major | prostaglandin f2-alpha synthase/D-arabinose dehydrogenase | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Schistosoma mansoni | aldo-keto reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase IV, putative | 0.0021 | 0.4091 | 0.4091 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0031 | 1 | 1 |
Schistosoma mansoni | aldo-keto reductase | 0.0031 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0031 | 1 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.0031 | 1 | 1 |
Leishmania major | aldo-keto reductase-like protein | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Entamoeba histolytica | aldose reductase, putative | 0.0031 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldehyde reductase | 0.0022 | 0.4471 | 0.0643 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Leishmania major | prostaglandin f synthase, putative | 0.0031 | 1 | 1 |
Mycobacterium leprae | PROBABLE OXIDOREDUCTASE | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldehyde reductase | 0.0022 | 0.4471 | 0.0643 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Onchocerca volvulus | 0.0031 | 1 | 0.5 | |
Onchocerca volvulus | 0.0031 | 1 | 0.5 | |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Onchocerca volvulus | 0.0031 | 1 | 0.5 | |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0031 | 1 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0031 | 1 | 1 |
Trypanosoma cruzi | aldo/keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Leishmania major | aldehyde reductase, putative,oxidoreductase, putative | 0.0031 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Onchocerca volvulus | 0.0031 | 1 | 0.5 | |
Schistosoma mansoni | pol-related | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase eta, putative | 0.0021 | 0.4091 | 0.4091 |
Giardia lamblia | Aldose reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Echinococcus multilocularis | aldo keto reductase | 0.0031 | 1 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase kappa, putative | 0.0021 | 0.4091 | 0.4091 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0031 | 1 | 1 |
Mycobacterium ulcerans | oxidoreductase | 0.0031 | 1 | 1 |
Trypanosoma cruzi | aldo-keto reductase | 0.0031 | 1 | 1 |
Trypanosoma brucei | prostaglandin f synthase | 0.0031 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0031 | 1 | 1 |
Trypanosoma brucei | DNA polymerase IV, putative | 0.0021 | 0.4091 | 0.4091 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Toxoplasma gondii | aldose reductase, putative | 0.0031 | 1 | 0.5 |
Trypanosoma brucei | DNA polymerase IV, putative | 0.0021 | 0.4091 | 0.4091 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0031 | 1 | 1 |
Onchocerca volvulus | 0.0031 | 1 | 0.5 | |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0031 | 1 | 1 |
Echinococcus granulosus | hypothetical protein | 0.0031 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
GI50 (functional) | > 1 10'-4M | Cytotoxicity against Homo sapiens (human) G361 cells by SRB assay | ChEMBL. | No reference |
IZ (functional) | = 1.3 mm | Antibacterial activity against Escherichia coli NCIM 2803 at 20 ug/ml after 24 hr by agar diffusion method | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.