Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | protein kinase, putative | 0.1704 | 1 | 1 |
Schistosoma mansoni | serine/threonine kinase | 0.0573 | 0.3239 | 0.4858 |
Echinococcus multilocularis | oxysterol binding protein 9 | 0.0033 | 0.0015 | 0.0023 |
Entamoeba histolytica | p21-activated kinase | 0.0045 | 0.0089 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.0573 | 0.3239 | 0.3229 |
Mycobacterium leprae | Probable pyruvate kinase PykA | 0.0039 | 0.0049 | 0.5 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.1099 | 0.6381 | 0.9592 |
Echinococcus granulosus | protein kinase c epsilon type | 0.0573 | 0.3239 | 0.4858 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.1144 | 0.6652 | 0.6647 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.0573 | 0.3239 | 0.487 |
Trypanosoma cruzi | Protein kinase B | 0.1144 | 0.6652 | 1 |
Echinococcus multilocularis | pdz domain containing protein | 0.0033 | 0.0015 | 0.0023 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.0573 | 0.3239 | 0.3229 |
Trichomonas vaginalis | pyruvate kinase, putative | 0.0039 | 0.0049 | 0.0034 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | Pleckstrin y | 0.0033 | 0.0015 | 0.0023 |
Trichomonas vaginalis | ribosomal protein S6 kinase, 90kD, polypeptide, putative | 0.0045 | 0.0089 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0045 | 0.0089 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma cruzi | NEK family Serine/threonine-protein kinase, putative | 0.0045 | 0.0089 | 0.0111 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma brucei | Serine/threonine-protein kinase NEK21, putative | 0.0045 | 0.0089 | 0.0074 |
Onchocerca volvulus | Pyruvate kinase homolog | 0.0039 | 0.0049 | 1 |
Plasmodium vivax | pyruvate kinase, putative | 0.0039 | 0.0049 | 0.0052 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0045 | 0.0089 | 0.0111 |
Entamoeba histolytica | protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.0573 | 0.3239 | 0.3229 |
Trichomonas vaginalis | pyruvate kinase, putative | 0.0039 | 0.0049 | 0.0034 |
Echinococcus multilocularis | Rho GTPase activating protein 24 | 0.0033 | 0.0015 | 0.0023 |
Echinococcus multilocularis | arf GAP with coiled coil, ANK repeat and PH | 0.0033 | 0.0015 | 0.0023 |
Leishmania major | pyruvate kinase | 0.0039 | 0.0049 | 0.4563 |
Echinococcus multilocularis | FERM and pleckstrin domain containing protein | 0.0033 | 0.0015 | 0.0023 |
Loa Loa (eye worm) | pyruvate kinase | 0.0039 | 0.0049 | 0.0034 |
Echinococcus multilocularis | nervana 2 | 0.1099 | 0.6381 | 0.9592 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | calcium dependent secretion activator 1 | 0.0033 | 0.0015 | 0.0023 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.0573 | 0.3239 | 0.4858 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0045 | 0.0089 | 0.0075 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.1099 | 0.6381 | 0.9592 |
Echinococcus granulosus | pyruvate kinase | 0.0039 | 0.0049 | 0.0051 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0045 | 0.0089 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.1671 | 0.9803 | 0.9802 |
Echinococcus multilocularis | type II inositol 3,4 bisphosphate 4 phosphatase | 0.0033 | 0.0015 | 0.0023 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.0573 | 0.3239 | 0.487 |
Entamoeba histolytica | protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | GRB2 associated binding protein 3 | 0.0033 | 0.0015 | 0.0023 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Entamoeba histolytica | hypothetical protein | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma cruzi | pyruvate kinase 2, putative | 0.0039 | 0.0049 | 0.0051 |
Entamoeba histolytica | protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma brucei | serine/threonine-protein kinase NRKB, putative | 0.0045 | 0.0089 | 0.0074 |
Echinococcus granulosus | nervana 2 | 0.1099 | 0.6381 | 0.9591 |
Echinococcus granulosus | protein kinase C gamma type | 0.0573 | 0.3239 | 0.4858 |
Loa Loa (eye worm) | hypothetical protein | 0.0573 | 0.3239 | 0.3229 |
Leishmania major | protein kinase, putative | 0.0045 | 0.0089 | 1 |
Echinococcus multilocularis | Pleckstrin y | 0.0033 | 0.0015 | 0.0023 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Giardia lamblia | Kinase, AGC PKA | 0.1111 | 0.6455 | 1 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.0045 | 0.0089 | 1 |
Brugia malayi | Pyruvate kinase, M2 isozyme | 0.0039 | 0.0049 | 0.0034 |
Echinococcus granulosus | serine/threonine protein kinase | 0.1144 | 0.6652 | 1 |
Mycobacterium tuberculosis | Probable pyruvate kinase PykA | 0.0039 | 0.0049 | 0.5 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.0573 | 0.3239 | 0.4858 |
Loa Loa (eye worm) | pyruvate kinase | 0.0039 | 0.0049 | 0.0034 |
Onchocerca volvulus | Pyruvate kinase homolog | 0.0039 | 0.0049 | 1 |
Echinococcus multilocularis | Pleckstrin domain containing protein, family B | 0.0033 | 0.0015 | 0.0023 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.1099 | 0.6381 | 0.9591 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.1111 | 0.6455 | 1 |
Plasmodium falciparum | calcium-dependent protein kinase 7 | 0.0045 | 0.0089 | 0.0115 |
Echinococcus multilocularis | oxysterol binding protein 1 | 0.0033 | 0.0015 | 0.0023 |
Echinococcus multilocularis | ras specific guanine nucleotide releasing factor | 0.0033 | 0.0015 | 0.0023 |
Echinococcus granulosus | pyruvate kinase | 0.0039 | 0.0049 | 0.0051 |
Trypanosoma brucei | protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0045 | 0.0089 | 0.0111 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.0573 | 0.3239 | 0.487 |
Echinococcus granulosus | NDR protein kinase | 0.0573 | 0.3239 | 0.4858 |
Entamoeba histolytica | protein kinase, putative | 0.1704 | 1 | 1 |
Echinococcus multilocularis | oxysterol binding protein 3 | 0.0033 | 0.0015 | 0.0023 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | myotubularin protein 13 | 0.0033 | 0.0015 | 0.0023 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.0573 | 0.3239 | 0.487 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.0573 | 0.3239 | 0.487 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0045 | 0.0089 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.0573 | 0.3239 | 0.3229 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Echinococcus granulosus | protein kinase c iota type | 0.0573 | 0.3239 | 0.4858 |
Echinococcus multilocularis | Oxysterol binding protein 11 | 0.0033 | 0.0015 | 0.0023 |
Trichomonas vaginalis | AGC family protein kinase | 0.0573 | 0.3239 | 0.3229 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.0573 | 0.3239 | 0.487 |
Entamoeba histolytica | protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.1111 | 0.6455 | 0.9703 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.1099 | 0.6381 | 0.9591 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.1144 | 0.6652 | 1 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.0045 | 0.0089 | 1 |
Leishmania major | protein kinase, putative | 0.0045 | 0.0089 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.1144 | 0.6652 | 0.6647 |
Toxoplasma gondii | calcium dependent protein kinase CDPK7 | 0.0045 | 0.0089 | 0.0075 |
Schistosoma mansoni | atypical protein kinase C | 0.0573 | 0.3239 | 0.4858 |
Brugia malayi | Pyruvate kinase, muscle isozyme | 0.0039 | 0.0049 | 0.0034 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Brugia malayi | Protein kinase domain containing protein | 0.0573 | 0.3239 | 0.3229 |
Echinococcus multilocularis | cytohesin 1 | 0.0033 | 0.0015 | 0.0023 |
Onchocerca volvulus | Pyruvate kinase homolog | 0.0039 | 0.0049 | 1 |
Trypanosoma cruzi | serine/threonine-protein kinase NRKB, putative | 0.0045 | 0.0089 | 0.0111 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.0573 | 0.3239 | 0.3229 |
Trypanosoma cruzi | pyruvate kinase 2, putative | 0.0039 | 0.0049 | 0.0051 |
Entamoeba histolytica | protein kinase 2, putative | 0.1111 | 0.6455 | 0.6449 |
Schistosoma mansoni | pyruvate kinase | 0.0039 | 0.0049 | 0.0051 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.1111 | 0.6455 | 0.9703 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.1704 | 1 | 1 |
Echinococcus multilocularis | arf GAP with SH3 domain, ANK repeat and PH | 0.0033 | 0.0015 | 0.0023 |
Echinococcus multilocularis | collagen type iv alpha 3 binding protein | 0.0033 | 0.0015 | 0.0023 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0045 | 0.0089 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | pleckstrin y domain containing family A | 0.0033 | 0.0015 | 0.0023 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.1144 | 0.6652 | 1 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0045 | 0.0089 | 0.0111 |
Echinococcus multilocularis | dynamin 1 | 0.0033 | 0.0015 | 0.0023 |
Plasmodium vivax | calcium-dependent protein kinase 7, putative | 0.0045 | 0.0089 | 0.0115 |
Entamoeba histolytica | protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0573 | 0.3239 | 0.3229 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Leishmania major | pyruvate kinase | 0.0039 | 0.0049 | 0.4563 |
Echinococcus multilocularis | Arf GAP and Pleckstrin domain containing protein | 0.0033 | 0.0015 | 0.0023 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.0573 | 0.3239 | 0.487 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Trichomonas vaginalis | 3-phosphoinositide dependent protein kinase-1, putative | 0.0045 | 0.0089 | 0.0074 |
Echinococcus multilocularis | DCC interacting protein 13 beta | 0.0033 | 0.0015 | 0.0023 |
Brugia malayi | Hr1 repeat family protein | 0.0573 | 0.3239 | 0.3229 |
Chlamydia trachomatis | pyruvate kinase | 0.0039 | 0.0049 | 0.5 |
Schistosoma mansoni | pyruvate kinase | 0.0039 | 0.0049 | 0.0051 |
Trypanosoma brucei | pyruvate kinase 1 | 0.0039 | 0.0049 | 0.0034 |
Echinococcus multilocularis | serine threonine protein kinase | 0.0573 | 0.3239 | 0.487 |
Echinococcus multilocularis | Pleckstrin y | 0.0033 | 0.0015 | 0.0023 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.1111 | 0.6455 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0606 | 0.3437 | 0.3427 |
Brugia malayi | protein kinase C II. | 0.0573 | 0.3239 | 0.3229 |
Echinococcus multilocularis | actin binding protein anillin | 0.0033 | 0.0015 | 0.0023 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.0573 | 0.3239 | 0.3229 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.1144 | 0.6652 | 1 |
Trypanosoma cruzi | serine/threonine protein kinase, putative | 0.0045 | 0.0089 | 0.0111 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.1111 | 0.6455 | 0.9703 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.0573 | 0.3239 | 0.3229 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.056 | 0.3166 | 0.3155 |
Echinococcus multilocularis | beta 1 syntrophin | 0.0033 | 0.0015 | 0.0023 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.0573 | 0.3239 | 0.4858 |
Brugia malayi | Protein kinase domain containing protein | 0.0573 | 0.3239 | 0.3229 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.0573 | 0.3239 | 0.4858 |
Echinococcus multilocularis | Ras associated and pleckstrin y | 0.0033 | 0.0015 | 0.0023 |
Mycobacterium ulcerans | pyruvate kinase | 0.0039 | 0.0049 | 0.5 |
Toxoplasma gondii | pyruvate kinase PyK1 | 0.0039 | 0.0049 | 0.0034 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Loa Loa (eye worm) | pyruvate kinase | 0.0039 | 0.0049 | 0.0034 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Echinococcus multilocularis | pyruvate kinase | 0.0039 | 0.0049 | 0.0073 |
Entamoeba histolytica | hypothetical protein | 0.0045 | 0.0089 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.1671 | 0.9803 | 0.9802 |
Loa Loa (eye worm) | hypothetical protein | 0.0039 | 0.0049 | 0.0034 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Echinococcus granulosus | nervana 2 | 0.1099 | 0.6381 | 0.9591 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0573 | 0.3239 | 0.4858 |
Trypanosoma brucei | pyruvate kinase 1, putative | 0.0039 | 0.0049 | 0.0034 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0573 | 0.3239 | 0.3229 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.0573 | 0.3239 | 0.4858 |
Trypanosoma brucei | serine/threonine-protein kinase NrkA | 0.0045 | 0.0089 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.1111 | 0.6455 | 0.9703 |
Trichomonas vaginalis | AGC family protein kinase | 0.1704 | 1 | 1 |
Plasmodium falciparum | pyruvate kinase | 0.0039 | 0.0049 | 0.0052 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.1704 | 1 | 1 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.0573 | 0.3239 | 0.487 |
Echinococcus multilocularis | nervana 2 | 0.1099 | 0.6381 | 0.9592 |
Trichomonas vaginalis | AGC family protein kinase | 0.0045 | 0.0089 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.1144 | 0.6652 | 1 |
Echinococcus multilocularis | pyruvate kinase | 0.0039 | 0.0049 | 0.0073 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.0045 | 0.0089 | 1 |
Echinococcus multilocularis | protein kinase c iota type | 0.0573 | 0.3239 | 0.487 |
Trypanosoma brucei | NEK family Serine/threonine-protein kinase, putative | 0.0045 | 0.0089 | 0.0074 |
Leishmania major | folate/biopterin transporter, putative | 0.0045 | 0.0089 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.1671 | 0.9803 | 0.9802 |
Toxoplasma gondii | AGC kinase | 0.1671 | 0.9803 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 8 % | Antagonist activity human EP1 receptor assessed as inhibition of PGE2-induced effect at 1 uM by reporter gene assay relative to control | ChEMBL. | 24252546 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.