Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0053 | 1 | 1 |
Giardia lamblia | GTOR | 0.0053 | 1 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Onchocerca volvulus | Transient receptor potential cation channel trpm homolog | 0.002 | 0 | 0.5 |
Trypanosoma brucei | phosphatidylinositol 3-kinase tor, putative | 0.0025 | 0.1544 | 0.1544 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.6717 | 0.6717 |
Onchocerca volvulus | Transient receptor potential cation channel trpm homolog | 0.002 | 0 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor2 | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Leishmania major | target of rapamycin (TOR) kinase 1, putative | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.3448 | 0.3448 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.2606 | 0.2606 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.6717 | 0.6717 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0034 | 0.4372 | 0.4372 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.262 | 0.262 |
Echinococcus multilocularis | Basic leucine zipper (bZIP) transcription | 0.0042 | 0.68 | 0.68 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.2606 | 0.2606 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.6717 | 0.6717 |
Trypanosoma cruzi | target of rapamycin kinase 3 | 0.0042 | 0.6731 | 0.6731 |
Schistosoma mansoni | hypothetical protein | 0.0042 | 0.68 | 0.68 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0035 | 0.4718 | 0.4718 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.3448 | 0.3448 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Entamoeba histolytica | phosphatidylinositol3-kinaseTor2, putative | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.6717 | 0.6717 |
Toxoplasma gondii | target of rapamycin (TOR), putative | 0.0039 | 0.5889 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0045 | 0.7654 | 0.7654 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.262 | 0.262 |
Echinococcus multilocularis | FKBP12 rapamycin complex associated protein | 0.0053 | 1 | 1 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.0042 | 0.6731 | 0.6731 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm)-related | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.262 | 0.262 |
Trypanosoma brucei | FAT domain/Rapamycin binding domain/Phosphatidylinositol 3- and 4-kinase, putative | 0.0022 | 0.062 | 0.062 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.262 | 0.262 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0039 | 0.5889 | 0.5889 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.3543 | 0.3543 |
Entamoeba histolytica | FKBP-rapamycin associated protein (FRAP), putative | 0.0053 | 1 | 1 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor1 | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.2606 | 0.2606 |
Echinococcus granulosus | FKBP12 rapamycin complex associated protein | 0.0053 | 1 | 1 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0053 | 1 | 1 |
Leishmania major | target of rapamycin (TOR) kinase 2, putative | 0.0053 | 1 | 1 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.0053 | 1 | 1 |
Echinococcus granulosus | Basic leucine zipper bZIP transcription | 0.0042 | 0.68 | 0.68 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.3543 | 0.3543 |
Leishmania major | target of rapamycin kinase (TOR) kinase 3 | 0.0042 | 0.6731 | 0.6731 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0053 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0042 | 0.6717 | 0.6717 |
Onchocerca volvulus | 0.002 | 0 | 0.5 | |
Schistosoma mansoni | transcription factor LCR-F1 | 0.0042 | 0.68 | 0.68 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0031 | 0.3543 | 0.3543 |
Brugia malayi | hypothetical protein | 0.0042 | 0.68 | 0.68 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (ADMET) | = 0.51 uM | Cytotoxicity against human MRC5 cells after 72 hrs by MTS assay | ChEMBL. | 24273633 |
Species name | Source | Reference | Is orphan |
---|---|---|---|
Homo sapiens | ChEMBL23 | 24273633 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.