Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6136 | 0.6136 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6136 | 0.6136 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0131 | 0.1484 | 0.1484 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.013 | 0.1427 | 0.1427 |
Echinococcus granulosus | tubulin subunit TubB | 0.0187 | 0.6136 | 0.5463 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | hypothetical protein | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | hypothetical protein | 0.013 | 0.1427 | 0.1427 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.013 | 0.1427 | 0.1427 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0131 | 0.1484 | 0.1484 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0187 | 0.6136 | 0.6136 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | alpha-tubulin | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.013 | 0.1427 | 0.1427 |
Trypanosoma brucei | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.013 | 0.1427 | 0.1427 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | hypothetical protein | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin | 0.0187 | 0.6136 | 0.6136 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Brugia malayi | tubulin alpha chain - mouse | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0187 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0187 | 0.6136 | 0.6136 |
Plasmodium falciparum | alpha tubulin 1 | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0187 | 0.6136 | 0.6136 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0187 | 0.6136 | 0.5463 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0187 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0187 | 0.6136 | 0.5463 |
Giardia lamblia | Alpha-tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0187 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0131 | 0.1484 | 0.1484 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0187 | 0.6136 | 0.6136 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0131 | 0.1484 | 0.1484 |
Plasmodium falciparum | alpha tubulin 2 | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0187 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0187 | 0.6136 | 0.5463 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
CC50 (ADMET) | > 100 uM | Cytotoxicity against Homo sapiens (human) MT4 cells containing integrated HTLV-1 genome after 96 hr by MTT assay | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.