Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | tubulin, putative | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0019 | 0.249 | 0.2166 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0019 | 0.249 | 0.2166 |
Echinococcus granulosus | beta tubulin | 0.0049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0049 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0019 | 0.249 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0019 | 0.249 | 0.249 |
Trypanosoma brucei | tubulin gamma chain | 0.0019 | 0.249 | 0.2166 |
Echinococcus multilocularis | beta tubulin | 0.0049 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0019 | 0.249 | 0.2166 |
Brugia malayi | Tubulin alpha-2 chain | 0.0019 | 0.249 | 0.249 |
Schistosoma mansoni | tubulin subunit beta | 0.0049 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0049 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0049 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0049 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0019 | 0.249 | 0.2166 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0019 | 0.249 | 0.249 |
Onchocerca volvulus | 0.0011 | 0.0414 | 1 | |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0019 | 0.249 | 0.249 |
Plasmodium falciparum | tubulin beta chain | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0019 | 0.249 | 0.249 |
Plasmodium vivax | tubulin beta chain, putative | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0011 | 0.0414 | 0.0414 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0011 | 0.0414 | 0.0414 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0049 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin subunit TubB | 0.0019 | 0.249 | 0.249 |
Schistosoma mansoni | tubulin subunit beta | 0.0049 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0019 | 0.249 | 0.2166 |
Trypanosoma brucei | beta tubulin | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0049 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0049 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0049 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0049 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0019 | 0.249 | 0.249 |
Schistosoma mansoni | tubulin subunit alpha | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.0019 | 0.249 | 0.249 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0019 | 0.249 | 0.2166 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0019 | 0.249 | 0.249 |
Brugia malayi | Tubulin beta chain | 0.0011 | 0.0414 | 0.0414 |
Schistosoma mansoni | tubulin subunit epsilon | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0019 | 0.249 | 0.249 |
Entamoeba histolytica | tubulin family protein | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0049 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0019 | 0.249 | 0.2166 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0019 | 0.249 | 0.2166 |
Entamoeba histolytica | tubulin family protein | 0.0049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0019 | 0.249 | 0.2166 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0019 | 0.249 | 0.2166 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0019 | 0.249 | 0.2166 |
Echinococcus multilocularis | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0019 | 0.249 | 0.2166 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0019 | 0.249 | 0.2166 |
Brugia malayi | alpha-tubulin | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0019 | 0.249 | 0.249 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0019 | 0.249 | 0.2166 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0019 | 0.249 | 0.249 |
Brugia malayi | tubulin alpha-2 chain | 0.0019 | 0.249 | 0.249 |
Giardia lamblia | Beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0019 | 0.249 | 0.249 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin epsilon chain | 0.0019 | 0.249 | 0.249 |
Schistosoma mansoni | tubulin subunit beta | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin gamma 1 chain | 0.0019 | 0.249 | 0.249 |
Trypanosoma brucei | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Loa Loa (eye worm) | hypothetical protein | 0.0011 | 0.0414 | 0.0414 |
Brugia malayi | Tubulin gamma chain | 0.0019 | 0.249 | 0.249 |
Giardia lamblia | Beta tubulin | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0049 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0019 | 0.249 | 0.2166 |
Loa Loa (eye worm) | alpha-tubulin | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | hypothetical protein | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | tubulin alpha | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0019 | 0.249 | 0.249 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0019 | 0.249 | 0.2166 |
Schistosoma mansoni | alpha tubulin | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0049 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0019 | 0.249 | 0.249 |
Echinococcus granulosus | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Loa Loa (eye worm) | beta-tubulin | 0.0049 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Brugia malayi | Tubulin alpha-2 chain | 0.0019 | 0.249 | 0.249 |
Trypanosoma brucei | beta tubulin | 0.0049 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0019 | 0.249 | 0.2166 |
Loa Loa (eye worm) | tubulin beta chain | 0.0049 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Schistosoma mansoni | tubulin subunit gamma | 0.0019 | 0.249 | 0.249 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin gamma 1 chain | 0.0019 | 0.249 | 0.249 |
Trypanosoma brucei | epsilon tubulin | 0.0019 | 0.249 | 0.2166 |
Echinococcus granulosus | alpha tubulin | 0.0019 | 0.249 | 0.249 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0011 | 0.0414 | 0.0414 |
Echinococcus multilocularis | tubulin epsilon chain | 0.0019 | 0.249 | 0.249 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0019 | 0.249 | 0.2166 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0019 | 0.249 | 0.249 |
Loa Loa (eye worm) | BEN-1 protein | 0.0049 | 1 | 1 |
Leishmania major | beta tubulin | 0.0049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0019 | 0.249 | 0.249 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0049 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0049 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
PFA (functional) | 0 mg kg-1 | Oral antiallergy activity in the passive foot anaphylaxis (PFA) model of rat, at a dose of 10 (mg/kg); Activity between positive and negative control groups | ChEMBL. | 2562852 |
PFA (functional) | 0 mg kg-1 | Oral antiallergy activity in the passive foot anaphylaxis (PFA) model of rat, at a dose of 3.16 (mg/kg); not significantly different from negative control group | ChEMBL. | 2562852 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.