Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | melanocortin 4 receptor | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Plasmodium falciparum | tubulin beta chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Plasmodium vivax | tubulin beta chain, putative | 0.0027 | 0.5 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0027 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Toxoplasma gondii | beta-tubulin, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta chain | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0027 | 0.5 | 0.5 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.5 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0027 | 0.5 | 0.5 |
Loa Loa (eye worm) | beta-tubulin | 0.0027 | 0.5 | 0.5 |
Toxoplasma gondii | beta tubulin | 0.0027 | 0.5 | 0.5 |
Brugia malayi | beta-tubulin, identical | 0.0027 | 0.5 | 0.5 |
Leishmania major | beta tubulin | 0.0027 | 0.5 | 0.5 |
Schistosoma mansoni | tubulin subunit beta | 0.0027 | 0.5 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0027 | 0.5 | 0.5 |
Echinococcus multilocularis | beta tubulin | 0.0027 | 0.5 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Ki (binding) | = 3 nM | Competitive Binding Assay Using Eu-NDP-a-MSH | BINDINGDB. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.