Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | opioid receptor, mu 1 | No references |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | AGC family protein kinase | 0.1676 | 0.214 | 1 |
Trypanosoma brucei | 3-methylcrotonyl-CoA carboxylase alpha subunit, putative | 0.1891 | 0.2653 | 0.183 |
Schistosoma mansoni | methylcrotonyl-CoA carboxylase | 0.1891 | 0.2653 | 0.2613 |
Plasmodium vivax | serine/threonine protein kinase 6, putative | 0.1676 | 0.214 | 0.3129 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0804 | 0.0054 | 0.0054 |
Leishmania major | acetyl-CoA carboxylase, putative | 0.4963 | 1 | 1 |
Brugia malayi | serine/threonine-protein kinase 6 | 0.1676 | 0.214 | 0.1321 |
Brugia malayi | serine/threonine protein kinase 6 | 0.1676 | 0.214 | 0.1321 |
Echinococcus granulosus | serine:threonine protein kinase 12 B | 0.1676 | 0.214 | 0.214 |
Schistosoma mansoni | pyruvate carboxylase | 0.1891 | 0.2653 | 0.2613 |
Echinococcus multilocularis | acetyl coenzyme A carboxylase 1 | 0.4963 | 1 | 1 |
Trypanosoma brucei | unspecified product | 0.1243 | 0.1104 | 0.0108 |
Leishmania major | methylcrotonoyl-coa carboxylase biotinylated subunitprotein-like protein | 0.1891 | 0.2653 | 0.0652 |
Loa Loa (eye worm) | carboxyl transferase domain-containing protein | 0.4789 | 0.9584 | 1 |
Chlamydia trachomatis | biotin carboxylase | 0.1717 | 0.2237 | 0.5 |
Plasmodium vivax | biotin carboxylase subunit of acetyl CoA carboxylase, putative | 0.3592 | 0.672 | 1 |
Trypanosoma cruzi | 3-methylcrotonyl-CoA carboxylase, putative | 0.1891 | 0.2653 | 0.479 |
Wolbachia endosymbiont of Brugia malayi | Acetyl/propionyl-CoA carboxylase, alpha subunit | 0.1891 | 0.2653 | 0.5 |
Entamoeba histolytica | protein kinase domain containing protein | 0.1676 | 0.214 | 1 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0804 | 0.0054 | 0.0054 |
Trypanosoma brucei | acetyl-CoA carboxylase | 0.4963 | 1 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.365 | 0.6861 | 1 |
Echinococcus multilocularis | aurora kinase A | 0.1676 | 0.214 | 0.214 |
Entamoeba histolytica | protein kinase, putative | 0.1202 | 0.1006 | 0.4568 |
Entamoeba histolytica | protein kinase , putative | 0.1676 | 0.214 | 1 |
Trypanosoma cruzi | acetyl-CoA carboxylase | 0.3073 | 0.5479 | 1 |
Schistosoma mansoni | methylcrotonyl-CoA carboxylase | 0.1891 | 0.2653 | 0.2613 |
Trypanosoma cruzi | 3-methylcrotonyl-CoA carboxylase, putative | 0.1891 | 0.2653 | 0.479 |
Loa Loa (eye worm) | AUR protein kinase | 0.1676 | 0.214 | 0.1321 |
Schistosoma mansoni | protein kinase | 0.1676 | 0.214 | 0.2097 |
Giardia lamblia | Aurora kinase | 0.1676 | 0.214 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.1202 | 0.1006 | 0.4568 |
Trypanosoma cruzi | aurora B kinase, putative | 0.1676 | 0.214 | 0.3845 |
Giardia lamblia | Acetyl-CoA carboxylase/pyruvate carboxylase fusion protein, putative | 0.0846 | 0.0156 | 0.049 |
Echinococcus multilocularis | propionyl coenzyme A carboxylase alpha chain | 0.1891 | 0.2653 | 0.2653 |
Trypanosoma brucei | 3-methylcrotonyl-CoA carboxylase alpha subunit, putative | 0.1891 | 0.2653 | 0.183 |
Toxoplasma gondii | acetyl-coA carboxylase ACC2 | 0.4963 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1676 | 0.214 | 1 |
Leishmania major | carboxylase, putative | 0.1891 | 0.2653 | 0.0652 |
Plasmodium falciparum | biotin carboxylase subunit of acetyl CoA carboxylase, putative | 0.3592 | 0.672 | 1 |
Entamoeba histolytica | serine/threonine- protein kinase 6, putative | 0.1676 | 0.214 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1676 | 0.214 | 1 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0804 | 0.0054 | 0.0054 |
Entamoeba histolytica | protein kinase, putative | 0.1202 | 0.1006 | 0.4568 |
Brugia malayi | serine/threonine kinase 12 | 0.1676 | 0.214 | 0.1321 |
Brugia malayi | Carboxyl transferase domain containing protein | 0.4789 | 0.9584 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.1676 | 0.214 | 1 |
Mycobacterium ulcerans | short chain dehydrogenase | 0.365 | 0.6861 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1676 | 0.214 | 0.2097 |
Toxoplasma gondii | acetyl-CoA carboxylase ACC1 | 0.4963 | 1 | 1 |
Plasmodium falciparum | serine/threonine protein kinase, putative | 0.1676 | 0.214 | 0.3129 |
Entamoeba histolytica | protein kinase, putative | 0.1676 | 0.214 | 1 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0804 | 0.0054 | 0.0054 |
Mycobacterium leprae | Probable bifunctional protein acetyl-/propionyl-coenzyme A carboxylase, alpha chain AccA3 (BccP) | 0.1891 | 0.2653 | 0.5 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0804 | 0.0054 | 0.0054 |
Trypanosoma brucei | aurora B kinase | 0.1676 | 0.214 | 0.126 |
Echinococcus granulosus | propionyl coenzyme A carboxylase alpha chain | 0.1891 | 0.2653 | 0.2653 |
Echinococcus granulosus | aurora kinase A | 0.1676 | 0.214 | 0.214 |
Entamoeba histolytica | serine/threonine protein kinase 6, putative | 0.1676 | 0.214 | 1 |
Loa Loa (eye worm) | AUR protein kinase | 0.1676 | 0.214 | 0.1321 |
Schistosoma mansoni | acetyl-CoA carboxylase | 0.4963 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.1676 | 0.214 | 1 |
Toxoplasma gondii | aurora kinase | 0.1676 | 0.214 | 0.126 |
Echinococcus multilocularis | serine:threonine protein kinase 12 B | 0.1676 | 0.214 | 0.214 |
Entamoeba histolytica | acetyl-coA carboxylase, putative | 0.0846 | 0.0156 | 0.049 |
Toxoplasma gondii | pyruvate carboxylase | 0.1891 | 0.2653 | 0.183 |
Entamoeba histolytica | serine/threonine- protein kinase 6 , putative | 0.1676 | 0.214 | 1 |
Loa Loa (eye worm) | AUR protein kinase | 0.1676 | 0.214 | 0.1321 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (binding) | = 3162 nM | HiRange Homogenous Time-Resolved Fluorescence (HTRF) Assay | BINDINGDB. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.