Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | dihydroorotate dehydrogenase | 0.3306 | 1 | 0.5 |
Trypanosoma brucei | dihydroorotate dehydrogenase (fumarate) | 0.3306 | 1 | 0.5 |
Echinococcus granulosus | dihydropyrimidine dehydrogenase NADP | 0.1291 | 0.2156 | 0.5 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Echinococcus multilocularis | dihydropyrimidine dehydrogenase (NADP+) | 0.1291 | 0.2156 | 0.5 |
Echinococcus granulosus | dihydropyrimidine dehydrogenase NADP | 0.1291 | 0.2156 | 0.5 |
Schistosoma mansoni | dihydroorotate dehydrogenase | 0.3306 | 1 | 1 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Plasmodium vivax | dihydroorotate dehydrogenase, mitochondrial precursor, putative | 0.3306 | 1 | 0.5 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Mycobacterium leprae | Probable dihydroorotate dehydrogenase PyrD | 0.3306 | 1 | 0.5 |
Toxoplasma gondii | dihydroorotate dehydrogenase reveal, putative | 0.3306 | 1 | 0.5 |
Wolbachia endosymbiont of Brugia malayi | dihydroorotate dehydrogenase 2 | 0.3306 | 1 | 0.5 |
Plasmodium falciparum | dihydroorotate dehydrogenase | 0.3306 | 1 | 0.5 |
Mycobacterium tuberculosis | Probable dihydroorotate dehydrogenase PyrD | 0.3306 | 1 | 0.5 |
Trypanosoma cruzi | dihydroorotate dehydrogenase, putative | 0.3306 | 1 | 1 |
Trichomonas vaginalis | dihydropyrimidine dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Echinococcus multilocularis | dihydropyrimidine dehydrogenase (NADP+) | 0.1291 | 0.2156 | 0.5 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Trypanosoma cruzi | dihydroorotate dehydrogenase, putative | 0.3306 | 1 | 1 |
Trypanosoma cruzi | dihydroorotate dehydrogenase (fumarate), putative | 0.3306 | 1 | 1 |
Mycobacterium ulcerans | dihydroorotate dehydrogenase 2 | 0.3306 | 1 | 0.5 |
Brugia malayi | Dihydroorotate dehydrogenase, mitochondrial precursor, putative | 0.3306 | 1 | 1 |
Entamoeba histolytica | dihydropyrimidine dehydrogenase, putative | 0.1291 | 0.2156 | 0.5 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Log SP (functional) | = 0.88 | Sweet potency as logarithm of sweet potency (log SP) relative to sucrose | ChEMBL. | 7241515 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.