Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0082 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0082 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0075 | 0.8206 | 0.8206 |
Echinococcus granulosus | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Plasmodium falciparum | alpha tubulin 1 | 0.0075 | 0.8206 | 0.8051 |
Schistosoma mansoni | tubulin subunit beta | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0075 | 0.8206 | 0.8206 |
Brugia malayi | tubulin alpha-2 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0082 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Loa Loa (eye worm) | tubulin beta chain | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.005 | 0.0792 | 0.0792 |
Loa Loa (eye worm) | beta-tubulin | 0.0082 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.005 | 0.0792 | 0.0792 |
Schistosoma mansoni | tubulin subunit beta | 0.0082 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0075 | 0.8206 | 0.8206 |
Loa Loa (eye worm) | BEN-1 protein | 0.0082 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0075 | 0.8206 | 0.8051 |
Toxoplasma gondii | beta-tubulin, putative | 0.0082 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0054 | 0.1909 | 0.1909 |
Trypanosoma brucei | beta tubulin | 0.0082 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0082 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Loa Loa (eye worm) | hypothetical protein | 0.0075 | 0.8206 | 0.8206 |
Trypanosoma brucei | beta tubulin | 0.0082 | 1 | 1 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Brugia malayi | Tubulin alpha-2 chain | 0.0075 | 0.8206 | 0.8051 |
Trichomonas vaginalis | tubulin, putative | 0.0082 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0075 | 0.8206 | 0.8051 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.005 | 0.0792 | 0.0792 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0075 | 0.8206 | 0.8206 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0075 | 0.8206 | 0.8051 |
Trypanosoma brucei | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0075 | 0.8206 | 0.8051 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0075 | 0.8206 | 0.8206 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0075 | 0.8206 | 0.8206 |
Giardia lamblia | Alpha-tubulin | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0082 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0075 | 0.8206 | 0.8206 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0082 | 1 | 1 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0082 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0082 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.005 | 0.0792 | 0.0792 |
Plasmodium vivax | tubulin beta chain, putative | 0.0082 | 1 | 1 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0075 | 0.8206 | 0.8206 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0075 | 0.8206 | 0.8206 |
Echinococcus multilocularis | beta tubulin | 0.0082 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Brugia malayi | alpha-tubulin | 0.0075 | 0.8206 | 0.8051 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0075 | 0.8206 | 0.8051 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0082 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0082 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0054 | 0.1909 | 0.1909 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0082 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0082 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0075 | 0.8206 | 0.8206 |
Plasmodium falciparum | alpha tubulin 2 | 0.0075 | 0.8206 | 0.8051 |
Loa Loa (eye worm) | hypothetical protein | 0.0054 | 0.1909 | 0.1909 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Trypanosoma brucei | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0075 | 0.8206 | 0.8051 |
Toxoplasma gondii | beta tubulin | 0.0082 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | beta tubulin | 0.0082 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0082 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0082 | 1 | 1 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0054 | 0.1909 | 0.1909 |
Echinococcus granulosus | beta tubulin | 0.0082 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0082 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0075 | 0.8206 | 0.8206 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0054 | 0.1909 | 0.1909 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0075 | 0.8206 | 0.8051 |
Giardia lamblia | Beta tubulin | 0.0082 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0082 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0082 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Schistosoma mansoni | tubulin subunit beta | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0082 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0082 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Brugia malayi | tubulin alpha chain - mouse | 0.0075 | 0.8206 | 0.8051 |
Echinococcus granulosus | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0075 | 0.8206 | 0.8206 |
Echinococcus granulosus | tubulin alpha chain | 0.0075 | 0.8206 | 0.8051 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0082 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0075 | 0.8206 | 0.8051 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0075 | 0.8206 | 0.8051 |
Schistosoma mansoni | tubulin subunit beta | 0.0082 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0075 | 0.8206 | 0.8051 |
Schistosoma mansoni | tubulin subunit alpha | 0.0075 | 0.8206 | 0.8051 |
Schistosoma mansoni | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Leishmania major | beta tubulin | 0.0082 | 1 | 1 |
Brugia malayi | Tubulin alpha-2 chain | 0.0075 | 0.8206 | 0.8051 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0075 | 0.8206 | 0.8206 |
Echinococcus granulosus | tubulin subunit TubB | 0.0075 | 0.8206 | 0.8051 |
Schistosoma mansoni | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0082 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0075 | 0.8206 | 0.8206 |
Plasmodium falciparum | tubulin beta chain | 0.0082 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0075 | 0.8206 | 0.8051 |
Loa Loa (eye worm) | BEN-1 protein | 0.0082 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
C50 (binding) | = 4 uM | Inhibitory concentration against ethidium bromide binding to [poly(dA-dT)] [poly(dA-dT)] | ChEMBL. | 8126699 |
IC50 (functional) | = 22 uM | Inhibition of P388 leukemia cells growth in culture | ChEMBL. | 8126699 |
IC50 (functional) | = 22 uM | Inhibition of P388 leukemia cells growth in culture | ChEMBL. | 8126699 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.