Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | tubulin subunit beta | 0.0033 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0033 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0019 | 0.1484 | 0.1484 |
Brugia malayi | Tubulin alpha-2 chain | 0.0027 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | BEN-1 protein | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | beta tubulin | 0.0033 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin subunit TubB | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.6136 | 0.6136 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0027 | 0.6136 | 0.6136 |
Schistosoma mansoni | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | hypothetical protein | 0.0019 | 0.1427 | 0.1427 |
Schistosoma mansoni | tubulin subunit beta | 0.0033 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0027 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin beta chain | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0033 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.6136 | 0.6136 |
Schistosoma mansoni | tubulin subunit beta | 0.0033 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0027 | 0.6136 | 0.5463 |
Giardia lamblia | Alpha-tubulin | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0019 | 0.1484 | 0.1484 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0027 | 0.6136 | 0.6136 |
Toxoplasma gondii | beta-tubulin, putative | 0.0033 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0033 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0027 | 0.6136 | 0.5463 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0033 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0019 | 0.1427 | 0.1427 |
Brugia malayi | tubulin alpha-2 chain | 0.0027 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit beta | 0.0033 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0027 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit beta | 0.0033 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | alpha-tubulin | 0.0027 | 0.6136 | 0.6136 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0033 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0033 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0033 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0033 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Trypanosoma brucei | beta tubulin | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0019 | 0.1427 | 0.1427 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0027 | 0.6136 | 0.6136 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0027 | 0.6136 | 0.5463 |
Giardia lamblia | Beta tubulin | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0019 | 0.1484 | 0.1484 |
Trypanosoma brucei | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0027 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0033 | 1 | 1 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0033 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0019 | 0.1427 | 0.1427 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.6136 | 0.6136 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0033 | 1 | 1 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.6136 | 0.6136 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0027 | 0.6136 | 0.5463 |
Trypanosoma brucei | beta tubulin | 0.0033 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0027 | 0.6136 | 0.6136 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0027 | 0.6136 | 0.6136 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin subunit beta | 0.0033 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Schistosoma mansoni | tubulin subunit alpha | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Plasmodium falciparum | alpha tubulin 1 | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0033 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0033 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0019 | 0.1484 | 0.1484 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0033 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Brugia malayi | Tubulin alpha-2 chain | 0.0027 | 0.6136 | 0.5463 |
Brugia malayi | tubulin alpha chain - mouse | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0033 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | tubulin alpha chain | 0.0027 | 0.6136 | 0.5463 |
Trypanosoma brucei | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.6136 | 0.6136 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0033 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0027 | 0.6136 | 0.5463 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0027 | 0.6136 | 0.6136 |
Leishmania major | beta tubulin | 0.0033 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0033 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0033 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0027 | 0.6136 | 0.5463 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0027 | 0.6136 | 0.5463 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0019 | 0.1427 | 0.1427 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0033 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0033 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Leishmania major | alpha tubulin | 0.0027 | 0.6136 | 0.5463 |
Trypanosoma brucei | beta tubulin | 0.0033 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0027 | 0.6136 | 0.5463 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0027 | 0.6136 | 0.6136 |
Loa Loa (eye worm) | hypothetical protein | 0.0027 | 0.6136 | 0.6136 |
Schistosoma mansoni | tubulin subunit beta | 0.0033 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 55 % | Tested for the inhibition of Candida GGTase I in Candida albicans at concentration of 3 microM | ChEMBL. | 11844687 |
Inhibition (binding) | = 55 % | Tested for the inhibition of Candida GGTase I in Candida albicans at concentration of 3 microM | ChEMBL. | 11844687 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.