Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | uridine phosphorylase | 0.0358 | 0.1248 | 0.1618 |
Leishmania major | nucleoside phosphorylase-like protein | 0.0358 | 0.1248 | 1 |
Schistosoma mansoni | methylthioadenosine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Giardia lamblia | Purine nucleoside phosphorylase lateral transfer candidate | 0.173 | 1 | 1 |
Chlamydia trachomatis | AMP nucleosidase | 0.0358 | 0.1248 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Trichomonas vaginalis | purine nucleoside phosphorylase I, putative | 0.173 | 1 | 1 |
Schistosoma mansoni | methylthioadenosine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1372 | 0.7714 | 0.7714 |
Giardia lamblia | 5-methylthioadenosine nucleosidase, S-adenosylhomocysteine nucleosidase | 0.0358 | 0.1248 | 0.1248 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Toxoplasma gondii | phosphorylase family protein | 0.0358 | 0.1248 | 0.5 |
Plasmodium falciparum | purine nucleoside phosphorylase | 0.0358 | 0.1248 | 0.5 |
Trypanosoma cruzi | nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0358 | 0.1248 | 0.1248 |
Echinococcus granulosus | uridine phosphorylase 1 | 0.0358 | 0.1248 | 0.1248 |
Toxoplasma gondii | phosphorylase family protein | 0.0358 | 0.1248 | 0.5 |
Trypanosoma brucei | methylthioadenosine phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Giardia lamblia | 5-methylthioadenosine nucleosidase, S-adenosylhomocysteine nucleosidase | 0.0358 | 0.1248 | 0.1248 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Loa Loa (eye worm) | hypothetical protein | 0.1372 | 0.7714 | 1 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Mycobacterium ulcerans | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Treponema pallidum | uridine phosphorylase (udp) | 0.0358 | 0.1248 | 0.5 |
Giardia lamblia | UPL-1 | 0.0358 | 0.1248 | 0.1248 |
Leishmania major | methylthioadenosine phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Schistosoma mansoni | uridine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Trypanosoma brucei | uridine phosphorylase | 0.0358 | 0.1248 | 1 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Treponema pallidum | purine nucleoside phosphorylase (deoD) | 0.0358 | 0.1248 | 0.5 |
Trypanosoma cruzi | methylthioadenosine phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0358 | 0.1248 | 0.5 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.5 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.1372 | 0.7714 | 0.7714 |
Schistosoma mansoni | methylthioadenosine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Trichomonas vaginalis | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.1248 |
Schistosoma mansoni | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Brugia malayi | MTAP | 0.0358 | 0.1248 | 0.1248 |
Schistosoma mansoni | uridine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Onchocerca volvulus | Purine nucleoside phosphorylase homolog | 0.173 | 1 | 0.5 |
Echinococcus multilocularis | methylthioadenosine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Toxoplasma gondii | Purine nucleoside phosphorylase | 0.0358 | 0.1248 | 0.5 |
Brugia malayi | uridine phosphorylase family protein | 0.0358 | 0.1248 | 0.1248 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.5 |
Trypanosoma cruzi | methylthioadenosine phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Plasmodium vivax | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.5 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus granulosus | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Schistosoma mansoni | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Loa Loa (eye worm) | S-methyl-5'-thioadenosine phosphorylase MTAP | 0.0358 | 0.1248 | 0.1618 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.5 |
Trypanosoma cruzi | nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Echinococcus granulosus | inosine guanosine and xanthosine phosphorylase | 0.1372 | 0.7714 | 0.7714 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.5 |
Trypanosoma cruzi | nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 1 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus multilocularis | uridine phosphorylase 1 | 0.0358 | 0.1248 | 0.1248 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0358 | 0.1248 | 0.1248 |
Treponema pallidum | pfs protein (pfs) | 0.0358 | 0.1248 | 0.5 |
Mycobacterium tuberculosis | Probable purine nucleoside phosphorylase DeoD (inosine phosphorylase) (PNP) | 0.173 | 1 | 1 |
Entamoeba histolytica | purine nucleoside phosphorylase, putative | 0.0358 | 0.1248 | 0.5 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Echinococcus granulosus | methylthioadenosine phosphorylase | 0.0358 | 0.1248 | 0.1248 |
Entamoeba histolytica | MTA/SAH nucleosidase, putative | 0.0358 | 0.1248 | 0.5 |
Mycobacterium leprae | Probable purine nucleoside phosphorylase DeoD (INOSINE PHOSPHORYLASE) (PNP) | 0.173 | 1 | 1 |
Echinococcus multilocularis | purine nucleoside phosphorylase | 0.173 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
-Log KB (functional) | = 4.67 | In vitro Histamine H2 receptor antagonist activity in the histamine-stimulated guinea pig right atrium | ChEMBL. | 2894467 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.