Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | tubulin family protein | 0.049 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.049 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0361 | 0.5357 | 0.5357 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.049 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0262 | 0.1744 | 0.1744 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0361 | 0.5357 | 0.4376 |
Giardia lamblia | Alpha-tubulin | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0361 | 0.5357 | 0.4376 |
Schistosoma mansoni | tubulin subunit beta | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0361 | 0.5357 | 0.5357 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0361 | 0.5357 | 0.4376 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0361 | 0.5357 | 0.4376 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | beta tubulin | 0.049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0361 | 0.5357 | 0.5357 |
Trypanosoma brucei | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.049 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0361 | 0.5357 | 0.4376 |
Schistosoma mansoni | tubulin subunit beta | 0.049 | 1 | 1 |
Brugia malayi | tubulin alpha-2 chain | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | hypothetical protein | 0.0248 | 0.1246 | 0.1246 |
Echinococcus multilocularis | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | tubulin subunit beta | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | beta tubulin | 0.049 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | BEN-1 protein | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0262 | 0.1744 | 0.1744 |
Brugia malayi | Tubulin alpha-2 chain | 0.0361 | 0.5357 | 0.4376 |
Entamoeba histolytica | tubulin family protein | 0.049 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0262 | 0.1744 | 0.1744 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0361 | 0.5357 | 0.5357 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0361 | 0.5357 | 0.5357 |
Echinococcus granulosus | tubulin subunit TubB | 0.0361 | 0.5357 | 0.4376 |
Plasmodium falciparum | alpha tubulin 2 | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0361 | 0.5357 | 0.4376 |
Schistosoma mansoni | tubulin subunit alpha | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | tubulin beta 1 chain | 0.049 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | tubulin beta chain | 0.049 | 1 | 1 |
Echinococcus granulosus | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.049 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Brugia malayi | tubulin alpha chain - mouse | 0.0361 | 0.5357 | 0.4376 |
Brugia malayi | Tubulin alpha-2 chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.049 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0248 | 0.1246 | 0.1246 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.049 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0361 | 0.5357 | 0.5357 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.049 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.049 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0361 | 0.5357 | 0.4376 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0361 | 0.5357 | 0.5357 |
Trichomonas vaginalis | tubulin, putative | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0361 | 0.5357 | 0.5357 |
Schistosoma mansoni | tubulin subunit beta | 0.049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0361 | 0.5357 | 0.4376 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0361 | 0.5357 | 0.5357 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | beta tubulin | 0.049 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.049 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Giardia lamblia | Alpha-tubulin | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0248 | 0.1246 | 0.1246 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0248 | 0.1246 | 0.1246 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Giardia lamblia | Beta tubulin | 0.049 | 1 | 1 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0361 | 0.5357 | 0.5357 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0248 | 0.1246 | 0.1246 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.049 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0262 | 0.1744 | 0.1744 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0361 | 0.5357 | 0.5357 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0361 | 0.5357 | 0.5357 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.049 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.049 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Echinococcus granulosus | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0361 | 0.5357 | 0.4376 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0361 | 0.5357 | 0.5357 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0361 | 0.5357 | 0.4376 |
Toxoplasma gondii | beta tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.049 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.049 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | alpha tubulin | 0.0361 | 0.5357 | 0.4376 |
Schistosoma mansoni | tubulin subunit alpha | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0361 | 0.5357 | 0.5357 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0361 | 0.5357 | 0.4376 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0361 | 0.5357 | 0.4376 |
Echinococcus multilocularis | tubulin subunit beta | 0.049 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0361 | 0.5357 | 0.4376 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0361 | 0.5357 | 0.5357 |
Giardia lamblia | Beta tubulin | 0.049 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0361 | 0.5357 | 0.4376 |
Trypanosoma brucei | beta tubulin | 0.049 | 1 | 1 |
Leishmania major | beta tubulin | 0.049 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Dose (functional) | = 5 mg kg-1 | Dose required in phototherapy for twelve days in tumor size detected in male Fischer CDF (F-344)/CrlBr rats | ChEMBL. | 2319568 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.