Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Schistosoma mansoni | pol-related | 0.0096 | 1 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0096 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0049 | 0.3011 | 0.3011 |
Toxoplasma gondii | lactate dehydrogenase LDH2 | 0.0049 | 0.3011 | 0.3011 |
Trypanosoma cruzi | aldo/keto reductase, putative | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0096 | 1 | 1 |
Giardia lamblia | Aldose reductase | 0.0096 | 1 | 0.5 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Toxoplasma gondii | lactate dehydrogenase LDH1 | 0.0049 | 0.3011 | 0.3011 |
Onchocerca volvulus | 0.0096 | 1 | 1 | |
Mycobacterium leprae | Conserved hypothetical protein | 0.0068 | 0.5922 | 0.5922 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldehyde reductase | 0.0068 | 0.5922 | 0.5922 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Toxoplasma gondii | aldose reductase, putative | 0.0096 | 1 | 1 |
Leishmania major | prostaglandin f synthase, putative | 0.0096 | 1 | 1 |
Trypanosoma cruzi | aldo-keto reductase | 0.0096 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0096 | 1 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase | 0.003 | 0.0256 | 0.0256 |
Echinococcus multilocularis | aldo keto reductase | 0.0096 | 1 | 1 |
Onchocerca volvulus | 0.0096 | 1 | 1 | |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Onchocerca volvulus | 0.0096 | 1 | 1 | |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Trypanosoma brucei | prostaglandin f synthase | 0.0096 | 1 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.0096 | 1 | 1 |
Brugia malayi | lactate dehydrogenase. | 0.0049 | 0.3011 | 0.3011 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Giardia lamblia | Aldose reductase | 0.0096 | 1 | 0.5 |
Schistosoma mansoni | malate dehydrogenase | 0.0049 | 0.3011 | 0.3011 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0049 | 0.3011 | 0.3011 |
Leishmania major | aldo-keto reductase-like protein | 0.0096 | 1 | 1 |
Echinococcus granulosus | lactate dehydrogenase protein | 0.0049 | 0.3011 | 0.3011 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0096 | 1 | 1 |
Onchocerca volvulus | 0.0096 | 1 | 1 | |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0096 | 1 | 1 |
Echinococcus multilocularis | L lactate dehydrogenase B chain | 0.0049 | 0.3011 | 0.3011 |
Plasmodium falciparum | L-lactate dehydrogenase | 0.0049 | 0.3011 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Schistosoma mansoni | aldo-keto reductase | 0.0096 | 1 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0096 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0096 | 1 | 1 |
Toxoplasma gondii | malate dehydrogenase MDH | 0.0049 | 0.3011 | 0.3011 |
Loa Loa (eye worm) | hypothetical protein | 0.0096 | 1 | 1 |
Schistosoma mansoni | aldo-keto reductase | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Leishmania major | prostaglandin f2-alpha synthase/D-arabinose dehydrogenase | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0096 | 1 | 1 |
Echinococcus granulosus | hypothetical protein | 0.0096 | 1 | 1 |
Plasmodium vivax | lactate dehydrogenase | 0.0049 | 0.3011 | 1 |
Plasmodium falciparum | malate dehydrogenase | 0.0049 | 0.3011 | 1 |
Entamoeba histolytica | aldose reductase, putative | 0.0096 | 1 | 1 |
Onchocerca volvulus | 0.0096 | 1 | 1 | |
Entamoeba histolytica | malate dehydrogenase, putative | 0.0049 | 0.3011 | 0.3011 |
Leishmania major | aldehyde reductase, putative,oxidoreductase, putative | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase | 0.0096 | 1 | 1 |
Mycobacterium ulcerans | oxidoreductase | 0.0096 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase protein | 0.0049 | 0.3011 | 0.3011 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0049 | 0.3011 | 0.3011 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0096 | 1 | 1 |
Plasmodium vivax | malate dehydrogenase, putative | 0.0049 | 0.3011 | 1 |
Trichomonas vaginalis | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Echinococcus multilocularis | lactate dehydrogenase a | 0.0049 | 0.3011 | 0.3011 |
Loa Loa (eye worm) | oxidoreductase | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | L lactate dehydrogenase | 0.003 | 0.0256 | 0.0256 |
Echinococcus granulosus | aldo keto reductase | 0.0096 | 1 | 1 |
Trypanosoma brucei | aldo-keto reductase, putative | 0.0096 | 1 | 1 |
Brugia malayi | oxidoreductase, aldo/keto reductase family protein | 0.0096 | 1 | 1 |
Mycobacterium leprae | PROBABLE OXIDOREDUCTASE | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Trichomonas vaginalis | dihydrodiol dehydrogenase, putative | 0.0096 | 1 | 1 |
Echinococcus granulosus | L lactate dehydrogenase B chain | 0.0049 | 0.3011 | 0.3011 |
Leishmania major | malate dehydrogenase, putative | 0.0049 | 0.3011 | 0.3011 |
Onchocerca volvulus | 0.0096 | 1 | 1 | |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Trichomonas vaginalis | aldo/keto reductase, putative | 0.0096 | 1 | 1 |
Loa Loa (eye worm) | oxidoreductase | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Schistosoma mansoni | L-lactate dehydrogenase | 0.0049 | 0.3011 | 0.3011 |
Echinococcus granulosus | lactate dehydrogenase a | 0.0049 | 0.3011 | 0.3011 |
Wolbachia endosymbiont of Brugia malayi | malate dehydrogenase | 0.0049 | 0.3011 | 0.5 |
Echinococcus multilocularis | aldo keto reductase family 1, member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Echinococcus granulosus | aldo keto reductase family 1 member B4 | 0.0096 | 1 | 1 |
Echinococcus multilocularis | aldehyde reductase | 0.0068 | 0.5922 | 0.5922 |
Loa Loa (eye worm) | hypothetical protein | 0.0049 | 0.3011 | 0.3011 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | = 0.5 ug ml-1 | Inhibitory activity against S. pneumoniae UC9912 | ChEMBL. | 10715160 |
MIC (functional) | = 1 ug ml-1 | Inhibitory activity against Methicillin-resistant S. epidermidis UC12084 | ChEMBL. | 10715160 |
MIC (functional) | = 2 ug ml-1 | Inhibitory activity against E. faecalis UC9217 | ChEMBL. | 10715160 |
MIC (functional) | = 2 ug ml-1 | Inhibitory activity against M. catarrhalis UC30610 | ChEMBL. | 10715160 |
MIC (functional) | = 4 ug ml-1 | Inhibitory activity against Methicillin-susceptible S. aureus UC9213 | ChEMBL. | 10715160 |
MIC (functional) | = 4 ug ml-1 | Inhibitory activity against Methicillin-resistant S. aureus UC6685 | ChEMBL. | 10715160 |
MIC (functional) | > 16 ug ml-1 | Inhibitory activity against H. influenzae UC30063 | ChEMBL. | 10715160 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.