Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | Ran family GTPase | 0.0022 | 0.0392 | 0.1371 |
Giardia lamblia | NADH oxidase lateral transfer candidate | 0.0047 | 0.1171 | 0.1488 |
Schistosoma mansoni | Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein) | 0.0048 | 0.1214 | 0.1214 |
Giardia lamblia | NADPH oxidoreductase, putative | 0.0242 | 0.7432 | 1 |
Entamoeba histolytica | iron-sulfur flavoprotein, putative | 0.0061 | 0.1618 | 0.565 |
Wolbachia endosymbiont of Brugia malayi | dihydrolipoamide dehydrogenase E3 component | 0.0047 | 0.1171 | 1 |
Plasmodium falciparum | flap endonuclease 1 | 0.0027 | 0.0554 | 0.1223 |
Plasmodium vivax | dihydrolipoyl dehydrogenase, mitochondrial, putative | 0.0047 | 0.1171 | 0.2803 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trypanosoma brucei | NADPH:adrenodoxin oxidoreductase, mitochondrial, putative | 0.0012 | 0.0076 | 0.0192 |
Onchocerca volvulus | Serine\/threonine kinase homolog | 0.01 | 0.2863 | 0.2918 |
Schistosoma mansoni | glutamate synthase | 0.0012 | 0.0076 | 0.0076 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trypanosoma brucei | importin beta-1 subunit, putative | 0.003 | 0.0648 | 0.1627 |
Trichomonas vaginalis | disulfide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0008 |
Leishmania major | 2-oxoglutarate dehydrogenase, e3 component, lipoamidedehydrogenase-like protein | 0.0047 | 0.1171 | 0.2942 |
Entamoeba histolytica | glutamate synthase beta subunit, putative | 0.0012 | 0.0076 | 0.0267 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Echinococcus granulosus | dihydrolipoamide dehydrogenase | 0.0047 | 0.1171 | 0.1171 |
Trichomonas vaginalis | apoptosis inducing factor, putative | 0.0012 | 0.0076 | 0.0008 |
Toxoplasma gondii | GTP-binding nuclear protein ran/tc4 | 0.0022 | 0.0392 | 0.0986 |
Brugia malayi | RNA, U transporter 1 | 0.0086 | 0.243 | 0.2476 |
Trypanosoma cruzi | trypanothione reductase, putative | 0.0047 | 0.1171 | 0.2942 |
Trichomonas vaginalis | flap endonuclease-1, putative | 0.0027 | 0.0554 | 0.0656 |
Echinococcus granulosus | serine:threonine protein kinase PLK1 | 0.01 | 0.2863 | 0.2863 |
Echinococcus granulosus | dual specificity | 0.0094 | 0.2683 | 0.2683 |
Trichomonas vaginalis | NAD(P)H dehydrogenase, putative | 0.0242 | 0.7432 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0038 | 0.0887 | 0.3098 |
Trypanosoma brucei | dihydrolipoamide dehydrogenase | 0.0047 | 0.1171 | 0.2942 |
Entamoeba histolytica | hypothetical protein | 0.0012 | 0.0071 | 0.0248 |
Echinococcus multilocularis | sulfide:quinone oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0182 | 0.5496 | 0.7369 |
Echinococcus multilocularis | serine:threonine protein kinase PLK1 | 0.01 | 0.2863 | 0.2863 |
Toxoplasma gondii | flap structure-specific endonuclease 1, putative | 0.0027 | 0.0554 | 0.1392 |
Schistosoma mansoni | importin beta-1 | 0.003 | 0.0648 | 0.0648 |
Echinococcus multilocularis | glutamate synthase | 0.0012 | 0.0076 | 0.0076 |
Echinococcus granulosus | histone lysine N methyltransferase H3 lysine 36 | 0.0011 | 0.0037 | 0.0037 |
Brugia malayi | MH2 domain containing protein | 0.0125 | 0.3683 | 0.3754 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Schistosoma mansoni | hypothetical protein | 0.0178 | 0.5361 | 0.5361 |
Trypanosoma cruzi | 2,4-dienoyl-coa reductase-like protein, putative | 0.0012 | 0.0076 | 0.0192 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0012 | 0.0071 | 0.0178 |
Entamoeba histolytica | serine/threonine protein kinase, putative | 0.01 | 0.2863 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0012 | 0.0071 | 0.0248 |
Onchocerca volvulus | 0.0012 | 0.0076 | 0.0078 | |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Brugia malayi | hypothetical protein | 0.0073 | 0.2012 | 0.2051 |
Mycobacterium tuberculosis | NADPH-dependent mycothiol reductase Mtr | 0.0134 | 0.3981 | 1 |
Leishmania major | protein kinase, putative,polo-like protein kinase, putative | 0.01 | 0.2863 | 0.7192 |
Entamoeba histolytica | hypothetical protein | 0.0061 | 0.1618 | 0.565 |
Loa Loa (eye worm) | programmed cell death 8 | 0.0012 | 0.0076 | 0.0076 |
Giardia lamblia | GTP-binding nuclear protein RAN/TC4 | 0.0022 | 0.0392 | 0.0429 |
Entamoeba histolytica | NAD(FAD)-dependent dehydrogenase, putative | 0.0012 | 0.0076 | 0.0267 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Echinococcus granulosus | flap endonuclease 1 | 0.0027 | 0.0554 | 0.0554 |
Brugia malayi | hypothetical protein | 0.0317 | 0.9812 | 1 |
Mycobacterium tuberculosis | NAD(P)H quinone reductase LpdA | 0.0047 | 0.1171 | 0.2803 |
Echinococcus multilocularis | thioredoxin glutathione reductase | 0.0134 | 0.3981 | 0.3981 |
Leishmania major | hypothetical protein, conserved | 0.0012 | 0.0076 | 0.0192 |
Trypanosoma cruzi | trypanothione reductase, putative | 0.0134 | 0.3981 | 1 |
Trichomonas vaginalis | importin beta-1, putative | 0.0025 | 0.0465 | 0.0535 |
Schistosoma mansoni | hypothetical protein | 0.0012 | 0.0076 | 0.0076 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Brugia malayi | Pyridine nucleotide-disulphide oxidoreductase family protein | 0.0012 | 0.0076 | 0.0078 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Loa Loa (eye worm) | hypothetical protein | 0.0073 | 0.2012 | 0.2012 |
Mycobacterium ulcerans | dihydrolipoamide dehydrogenase | 0.0047 | 0.1171 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.003 | 0.0648 | 0.0648 |
Trichomonas vaginalis | dihydrolipoamide dehydrogenase, putative | 0.0012 | 0.0076 | 0.0008 |
Trypanosoma brucei | dihydrolipoyl dehydrogenase | 0.0047 | 0.1171 | 0.2942 |
Entamoeba histolytica | protein kinase, putative | 0.0094 | 0.2683 | 0.9372 |
Plasmodium falciparum | thioredoxin reductase | 0.0047 | 0.1171 | 0.2803 |
Trichomonas vaginalis | glutamate synthase, putative | 0.0012 | 0.0076 | 0.0008 |
Echinococcus granulosus | dihydropyrimidine dehydrogenase NADP | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma cruzi | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Toxoplasma gondii | pyruvate dehydrogenase complex subunit PDH-E3II | 0.0047 | 0.1171 | 0.2942 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Trypanosoma brucei | polo-like protein kinase | 0.01 | 0.2863 | 0.7192 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Entamoeba histolytica | glutamate synthase beta subunit, putative | 0.0012 | 0.0076 | 0.0267 |
Leishmania major | acetoin dehydrogenase e3 component-like protein | 0.0047 | 0.1171 | 0.2942 |
Treponema pallidum | NADH oxidase | 0.0047 | 0.1171 | 1 |
Leishmania major | 2,4-dienoyl-coa reductase fadh1, putative | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trypanosoma cruzi | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Entamoeba histolytica | hypothetical protein | 0.0025 | 0.0465 | 0.1623 |
Echinococcus granulosus | geminin | 0.0178 | 0.5361 | 0.5361 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.0047 | 0.1171 | 0.2803 |
Brugia malayi | alpha keto acid dehydrogenase complex, E3 component, lipoamide dehydrogenase | 0.0034 | 0.0776 | 0.079 |
Trypanosoma cruzi | CMGC/DYRK protein kinase, putative | 0.0094 | 0.2683 | 0.674 |
Echinococcus granulosus | Basic leucine zipper bZIP transcription | 0.0038 | 0.0887 | 0.0887 |
Trichomonas vaginalis | disulfide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0008 |
Giardia lamblia | NADPH oxidoreductase, putative | 0.0242 | 0.7432 | 1 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Brugia malayi | serine/threonine-protein kinase plk-2 | 0.01 | 0.2863 | 0.2918 |
Brugia malayi | Importin beta-1 subunit | 0.003 | 0.0648 | 0.066 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0094 | 0.2683 | 0.2683 |
Onchocerca volvulus | 0.0317 | 0.9812 | 1 | |
Trichomonas vaginalis | Importin beta-1 subunit, putative | 0.0025 | 0.0465 | 0.0535 |
Trichomonas vaginalis | hypothetical protein | 0.0036 | 0.0816 | 0.1013 |
Mycobacterium ulcerans | dihydrolipoamide dehydrogenase, LpdB | 0.0047 | 0.1171 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0038 | 0.0887 | 0.3098 |
Trypanosoma cruzi | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Wolbachia endosymbiont of Brugia malayi | dihydrolipoamide dehydrogenase E3 component | 0.0047 | 0.1171 | 1 |
Toxoplasma gondii | NADPH-glutathione reductase | 0.0047 | 0.1171 | 0.2942 |
Toxoplasma gondii | non-proton pumping type-II NADH dehydrogenase I | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Loa Loa (eye worm) | nucleolar RNA-associated protein alpha | 0.0323 | 1 | 1 |
Echinococcus granulosus | guanine nucleotide binding protein Gs subunit | 0.0048 | 0.1214 | 0.1214 |
Trypanosoma brucei | dihydrolipoamide dehydrogenase, point mutation | 0.0047 | 0.1171 | 0.2942 |
Brugia malayi | dihydrolipoyl dehydrogenase, mitochondrial precursor, putative | 0.0047 | 0.1171 | 0.1193 |
Loa Loa (eye worm) | CMGC/DYRK/DYRK1 protein kinase | 0.0094 | 0.2683 | 0.2683 |
Trypanosoma cruzi | dihydrolipoyl dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Entamoeba histolytica | Flap nuclease, putative | 0.0027 | 0.0554 | 0.1935 |
Schistosoma mansoni | ran | 0.0022 | 0.0392 | 0.0392 |
Brugia malayi | Thioredoxin reductase | 0.0134 | 0.3981 | 0.4057 |
Plasmodium vivax | thioredoxin reductase, putative | 0.0134 | 0.3981 | 1 |
Schistosoma mansoni | kinase | 0.0051 | 0.1306 | 0.1306 |
Loa Loa (eye worm) | pyridine nucleotide-disufhide oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Schistosoma mansoni | SET domain protein | 0.0011 | 0.0037 | 0.0037 |
Trichomonas vaginalis | disulfide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0008 |
Trypanosoma brucei | CMGC/DYRK protein kinase, putative | 0.0094 | 0.2683 | 0.674 |
Loa Loa (eye worm) | hypothetical protein | 0.0093 | 0.2657 | 0.2657 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Trypanosoma brucei | hypothetical protein, conserved | 0.0012 | 0.0076 | 0.0192 |
Loa Loa (eye worm) | hypothetical protein | 0.0093 | 0.2657 | 0.2657 |
Echinococcus multilocularis | apoptosis inducing factor 1 mitochondrial | 0.0012 | 0.0076 | 0.0076 |
Schistosoma mansoni | tsg101-related | 0.005 | 0.1267 | 0.1267 |
Trichomonas vaginalis | CAMK family protein kinase | 0.005 | 0.1264 | 0.1621 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Brugia malayi | NADPH:adrenodoxin oxidoreductase, mitochondrial precursor | 0.0012 | 0.0076 | 0.0078 |
Echinococcus granulosus | dihydropyrimidine dehydrogenase NADP | 0.0012 | 0.0076 | 0.0076 |
Echinococcus multilocularis | geminin | 0.0178 | 0.5361 | 0.5361 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | NAD(P)H dehydrogenase, putative | 0.0061 | 0.1618 | 0.2101 |
Mycobacterium tuberculosis | Probable soluble pyridine nucleotide transhydrogenase SthA (STH) (NAD(P)(+) transhydrogenase [B-specific]) (nicotinamide nucleot | 0.0047 | 0.1171 | 0.2803 |
Echinococcus granulosus | apoptosis inducing factor 1 mitochondrial | 0.0012 | 0.0076 | 0.0076 |
Schistosoma mansoni | Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein) | 0.0048 | 0.1214 | 0.1214 |
Entamoeba histolytica | protein kinase, putative | 0.0094 | 0.2683 | 0.9372 |
Toxoplasma gondii | NADH dehydrogenase (NDH2-II) | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Schistosoma mansoni | flap endonuclease-1 | 0.0025 | 0.047 | 0.047 |
Trypanosoma brucei | pyridine nucleotide-disulphide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0192 |
Entamoeba histolytica | dihydropyrimidine dehydrogenase, putative | 0.0012 | 0.0076 | 0.0267 |
Brugia malayi | hypothetical protein | 0.0038 | 0.0887 | 0.0904 |
Schistosoma mansoni | hypothetical protein | 0.0178 | 0.5361 | 0.5361 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Trypanosoma cruzi | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Plasmodium vivax | glutathione reductase, putative | 0.0134 | 0.3981 | 1 |
Schistosoma mansoni | dihydrolipoamide dehydrogenase | 0.0047 | 0.1171 | 0.1171 |
Toxoplasma gondii | pyridine nucleotide-disulfide oxidoreductase domain-containing protein | 0.0012 | 0.0076 | 0.0192 |
Echinococcus multilocularis | guanine nucleotide binding protein G(s) subunit | 0.0048 | 0.1214 | 0.1214 |
Trichomonas vaginalis | NAD(P)H dehydrogenase, putative | 0.0061 | 0.1618 | 0.2101 |
Brugia malayi | Pyridine nucleotide-disulphide oxidoreductase family protein | 0.0012 | 0.0076 | 0.0078 |
Schistosoma mansoni | hypothetical protein | 0.0038 | 0.0887 | 0.0887 |
Trichomonas vaginalis | glutamate synthase, putative | 0.0012 | 0.0076 | 0.0008 |
Plasmodium falciparum | GTP-binding nuclear protein RAN/TC4 | 0.0022 | 0.0392 | 0.0809 |
Mycobacterium tuberculosis | Dihydrolipoamide dehydrogenase LpdC (lipoamide reductase (NADH)) (lipoyl dehydrogenase) (dihydrolipoyl dehydrogenase) (diaphoras | 0.0047 | 0.1171 | 0.2803 |
Loa Loa (eye worm) | GTP-binding nuclear protein RAN/TC4 | 0.0022 | 0.0392 | 0.0392 |
Trypanosoma cruzi | NADH dehydrogenase, putative | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Leishmania major | hypothetical protein, conserved | 0.0012 | 0.0076 | 0.0192 |
Schistosoma mansoni | hypothetical protein | 0.0323 | 1 | 1 |
Plasmodium falciparum | importin beta, putative | 0.003 | 0.0648 | 0.1463 |
Trypanosoma cruzi | GTP-binding nuclear protein rtb2, putative | 0.0022 | 0.0392 | 0.0986 |
Trypanosoma cruzi | NADH dehydrogenase, putative | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | NAD(P)H dehydrogenase, putative | 0.0242 | 0.7432 | 1 |
Echinococcus granulosus | guanine nucleotide binding protein Gs subunit | 0.0048 | 0.1214 | 0.1214 |
Leishmania major | trypanothione reductase | 0.0134 | 0.3981 | 1 |
Schistosoma mansoni | tsg101-related | 0.0061 | 0.1622 | 0.1622 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Brugia malayi | Pyridine nucleotide-disulphide oxidoreductase, dimerisation domain containing protein | 0.0034 | 0.0776 | 0.079 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Entamoeba histolytica | disulphide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0267 |
Leishmania major | GTP-binding protein, putative | 0.0022 | 0.0392 | 0.0986 |
Brugia malayi | Flap endonuclease-1 | 0.0027 | 0.0554 | 0.0565 |
Entamoeba histolytica | hypothetical protein | 0.0012 | 0.0071 | 0.0248 |
Trichomonas vaginalis | disulfide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0008 |
Entamoeba histolytica | hypothetical protein | 0.0038 | 0.0887 | 0.3098 |
Plasmodium falciparum | glutathione reductase | 0.0047 | 0.1171 | 0.2803 |
Echinococcus granulosus | importin subunit beta 1 | 0.003 | 0.0648 | 0.0648 |
Loa Loa (eye worm) | MH2 domain-containing protein | 0.0125 | 0.3683 | 0.3683 |
Loa Loa (eye worm) | PLK/PLK1 protein kinase | 0.01 | 0.2863 | 0.2863 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trypanosoma cruzi | GTP-binding nuclear protein rtb2, putative | 0.0022 | 0.0392 | 0.0986 |
Entamoeba histolytica | protein kinase domain containing protein | 0.0094 | 0.2683 | 0.9372 |
Schistosoma mansoni | disulfide oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Echinococcus multilocularis | snurportin 1 | 0.0323 | 1 | 1 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Loa Loa (eye worm) | flap endonuclease-1 | 0.0027 | 0.0554 | 0.0554 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Echinococcus multilocularis | importin subunit beta 1 | 0.003 | 0.0648 | 0.0648 |
Schistosoma mansoni | tsg101-related | 0.0061 | 0.1622 | 0.1622 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | disulfide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0008 |
Toxoplasma gondii | HEAT repeat-containing protein | 0.003 | 0.0648 | 0.1627 |
Giardia lamblia | NADPH oxidoreductase, putative | 0.0242 | 0.7432 | 1 |
Loa Loa (eye worm) | GTP-binding regulatory protein Gs alpha-S chain | 0.0048 | 0.1214 | 0.1214 |
Leishmania major | serine/threonine-protein kinase, putative,protein kinase, putative | 0.0094 | 0.2683 | 0.674 |
Trypanosoma cruzi | pyridine nucleotide-disulphide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0192 |
Plasmodium falciparum | glutathione reductase | 0.0134 | 0.3981 | 1 |
Schistosoma mansoni | sulfide quinone reductase | 0.0012 | 0.0076 | 0.0076 |
Schistosoma mansoni | glutamate synthase | 0.0012 | 0.0076 | 0.0076 |
Trichomonas vaginalis | dihydropyrimidine dehydrogenase, putative | 0.0012 | 0.0076 | 0.0008 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Schistosoma mansoni | ran | 0.0022 | 0.0392 | 0.0392 |
Echinococcus multilocularis | dihydropyrimidine dehydrogenase (NADP+) | 0.0012 | 0.0076 | 0.0076 |
Trichomonas vaginalis | glutathione reductase, putative | 0.0047 | 0.1171 | 0.1494 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Leishmania major | importin beta-1 subunit, putative | 0.0025 | 0.0465 | 0.1168 |
Brugia malayi | glutamate synthase | 0.0012 | 0.0076 | 0.0078 |
Echinococcus granulosus | NADPH:adrenodoxin oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma cruzi | flap endonuclease-1 (FEN-1), putative | 0.0027 | 0.0554 | 0.1392 |
Mycobacterium ulcerans | flavoprotein disulfide reductase | 0.0047 | 0.1171 | 1 |
Trichomonas vaginalis | mercuric reductase, putative | 0.0047 | 0.1171 | 0.1494 |
Trypanosoma cruzi | 2,4-dienoyl-coa reductase fadh1, putative | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Echinococcus multilocularis | histone lysine N methyltransferase, H3 lysine 36 | 0.0011 | 0.0037 | 0.0037 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0012 | 0.0071 | 0.0178 |
Plasmodium vivax | importin-beta 2, putative | 0.003 | 0.0648 | 0.1463 |
Toxoplasma gondii | pyridine nucleotide-disulfide oxidoreductase domain-containing protein | 0.0012 | 0.0076 | 0.0192 |
Schistosoma mansoni | glutamate synthase | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma cruzi | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Mycobacterium leprae | DIHYDROLIPOAMIDE DEHYDROGENASE LPD (LIPOAMIDE REDUCTASE (NADH)) (LIPOYL DEHYDROGENASE) (DIHYDROLIPOYL DEHYDROGENASE) (DIAPHORASE | 0.0047 | 0.1171 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0038 | 0.0887 | 0.3098 |
Entamoeba histolytica | pyridine nucleotide-disulfide oxidoreductase family protein | 0.0012 | 0.0076 | 0.0267 |
Loa Loa (eye worm) | glutathione reductase | 0.0134 | 0.3981 | 0.3981 |
Trichomonas vaginalis | Importin beta-1 subunit, putative | 0.0025 | 0.0465 | 0.0535 |
Schistosoma mansoni | serine/threonine protein kinase | 0.01 | 0.2863 | 0.2863 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trypanosoma cruzi | CMGC/DYRK protein kinase, putative | 0.0094 | 0.2683 | 0.674 |
Trypanosoma cruzi | Vps23 core domain containing protein, putative | 0.0023 | 0.0427 | 0.1071 |
Echinococcus granulosus | GTP binding nuclear protein Ran | 0.0022 | 0.0392 | 0.0392 |
Trypanosoma brucei | 2,4-dienoyl-coa reductase-like protein | 0.0012 | 0.0076 | 0.0192 |
Trypanosoma brucei | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Trichomonas vaginalis | NAD(P)H dehydrogenase, putative | 0.0242 | 0.7432 | 1 |
Plasmodium falciparum | thioredoxin reductase | 0.0134 | 0.3981 | 1 |
Entamoeba histolytica | thioredoxin reductase, putative | 0.0012 | 0.0076 | 0.0267 |
Echinococcus multilocularis | dual specificity | 0.0094 | 0.2683 | 0.2683 |
Entamoeba histolytica | tumor susceptibility gene 101 protein, putative | 0.005 | 0.1267 | 0.4424 |
Trypanosoma cruzi | polo-like protein kinase, putative | 0.01 | 0.2863 | 0.7192 |
Plasmodium falciparum | dihydrolipoyl dehydrogenase, apicoplast | 0.0047 | 0.1171 | 0.2803 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Trypanosoma brucei | flap endonuclease-1 (FEN-1), putative | 0.0027 | 0.0554 | 0.1392 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Trypanosoma cruzi | pyridine nucleotide-disulphide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0192 |
Entamoeba histolytica | modulator of drug activity B homolog, putative | 0.0061 | 0.1618 | 0.565 |
Plasmodium vivax | flap endonuclease 1, putative | 0.0027 | 0.0554 | 0.1223 |
Brugia malayi | GTP-binding regulatory protein Gs alpha-S chain, putative | 0.0048 | 0.1214 | 0.1238 |
Leishmania major | hypothetical protein, conserved | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Echinococcus multilocularis | tumor susceptibility gene 101 protein | 0.0073 | 0.2012 | 0.2012 |
Echinococcus multilocularis | dihydropyrimidine dehydrogenase (NADP+) | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0012 | 0.0076 | 0.0192 |
Leishmania major | 2,4-dienoyl-coa reductase-like protein | 0.0012 | 0.0076 | 0.0192 |
Loa Loa (eye worm) | hypothetical protein | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma cruzi | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Schistosoma mansoni | transcription factor LCR-F1 | 0.0038 | 0.0887 | 0.0887 |
Echinococcus multilocularis | Basic leucine zipper (bZIP) transcription | 0.0038 | 0.0887 | 0.0887 |
Toxoplasma gondii | thioredoxin reductase | 0.0134 | 0.3981 | 1 |
Echinococcus granulosus | histone lysine N methyltransferase NSD3 | 0.0034 | 0.078 | 0.078 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trichomonas vaginalis | FMN-dependent NADH-azoreductase, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | ran, putative | 0.0022 | 0.0392 | 0.0437 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Echinococcus granulosus | glutamate synthase | 0.0012 | 0.0076 | 0.0076 |
Echinococcus multilocularis | dihydrolipoamide dehydrogenase | 0.0047 | 0.1171 | 0.1171 |
Leishmania major | flap endonuclease-1 (FEN-1), putative | 0.0027 | 0.0554 | 0.1392 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Echinococcus multilocularis | pyridine nucleotide disulfide oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Echinococcus granulosus | tumor susceptibility gene 101 protein | 0.0073 | 0.2012 | 0.2012 |
Trypanosoma brucei | trypanothione reductase | 0.0134 | 0.3981 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Trypanosoma brucei | pyridine nucleotide-disulphide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0192 |
Plasmodium vivax | dihydrolipoyl dehydrogenase, apicoplast, putative | 0.0047 | 0.1171 | 0.2803 |
Leishmania major | NADH dehydrogenase, putative | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | CAMK family protein kinase | 0.01 | 0.2863 | 0.3793 |
Brugia malayi | Protein kinase domain containing protein | 0.0094 | 0.2683 | 0.2735 |
Trypanosoma cruzi | dihydrolipoyl dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Schistosoma mansoni | sulfide quinone reductase | 0.0012 | 0.0076 | 0.0076 |
Brugia malayi | GTP-binding nuclear protein RAN/TC4 | 0.0022 | 0.0392 | 0.04 |
Trypanosoma brucei | importin beta-1 subunit, putative | 0.003 | 0.0648 | 0.1627 |
Loa Loa (eye worm) | hypothetical protein | 0.0317 | 0.9812 | 0.9812 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Loa Loa (eye worm) | thioredoxin reductase | 0.0134 | 0.3981 | 0.3981 |
Trypanosoma brucei | dihydrolipoamide dehydrogenase | 0.0047 | 0.1171 | 0.2942 |
Echinococcus multilocularis | histone lysine N methyltransferase NSD3 | 0.0034 | 0.078 | 0.078 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0242 | 0.7432 | 1 |
Giardia lamblia | Flap structure-specific endonuclease | 0.0027 | 0.0554 | 0.0649 |
Echinococcus granulosus | pyridine nucleotide disulfide oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma brucei | NADH dehydrogenase | 0.0012 | 0.0076 | 0.0192 |
Trypanosoma cruzi | polo-like protein kinase, putative | 0.01 | 0.2863 | 0.7192 |
Trichomonas vaginalis | CAMK family protein kinase | 0.005 | 0.1264 | 0.1621 |
Chlamydia trachomatis | dihydrolipoyl dehydrogenase | 0.0047 | 0.1171 | 1 |
Trypanosoma brucei | GTP-binding nuclear protein rtb2, putative | 0.0022 | 0.0392 | 0.0986 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Leishmania major | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Schistosoma mansoni | SET domain protein | 0.0034 | 0.078 | 0.078 |
Schistosoma mansoni | Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein) | 0.0048 | 0.1214 | 0.1214 |
Plasmodium vivax | GTP-binding nuclear protein RAN/TC4, putative | 0.0022 | 0.0392 | 0.0809 |
Echinococcus multilocularis | guanine nucleotide binding protein G(s) subunit | 0.0048 | 0.1214 | 0.1214 |
Giardia lamblia | Kinase, PLK | 0.01 | 0.2863 | 0.3788 |
Echinococcus multilocularis | flap endonuclease 1 | 0.0027 | 0.0554 | 0.0554 |
Toxoplasma gondii | selenide, water dikinase | 0.0012 | 0.0076 | 0.0192 |
Entamoeba histolytica | hypothetical protein | 0.0094 | 0.2683 | 0.9372 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0012 | 0.0076 | 0.0008 |
Toxoplasma gondii | pyridine nucleotide-disulfide oxidoreductase domain-containing protein | 0.0012 | 0.0076 | 0.0192 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Echinococcus multilocularis | GTP binding nuclear protein Ran | 0.0022 | 0.0392 | 0.0392 |
Trichomonas vaginalis | dihydroorotate dehydrogenase, putative | 0.0012 | 0.0076 | 0.0008 |
Echinococcus granulosus | sulfide:quinone oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Loa Loa (eye worm) | transcription factor SMAD2 | 0.0125 | 0.3683 | 0.3683 |
Leishmania major | hypothetical protein, conserved | 0.0023 | 0.0427 | 0.1071 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0061 | 0.1618 | 0.2101 |
Trichomonas vaginalis | disulfide oxidoreductase, putative | 0.0012 | 0.0076 | 0.0008 |
Entamoeba histolytica | hypothetical protein | 0.0012 | 0.0071 | 0.0248 |
Trichomonas vaginalis | modulator of drug activity B, putative | 0.0061 | 0.1618 | 0.2101 |
Brugia malayi | glutathione reductase | 0.0134 | 0.3981 | 0.4057 |
Trypanosoma brucei | Vps23 core domain containing protein, putative | 0.0023 | 0.0427 | 0.1071 |
Leishmania major | dihydrolipoamide dehydrogenase, putative | 0.0047 | 0.1171 | 0.2942 |
Plasmodium falciparum | dihydrolipoyl dehydrogenase, mitochondrial | 0.0047 | 0.1171 | 0.2803 |
Echinococcus granulosus | thioredoxin glutathione reductase | 0.0134 | 0.3981 | 0.3981 |
Trypanosoma cruzi | importin beta-1 subunit, putative | 0.0025 | 0.0465 | 0.1168 |
Trypanosoma cruzi | NADPH:adrenodoxin oxidoreductase, mitochondrial, putative | 0.0012 | 0.0076 | 0.0192 |
Echinococcus multilocularis | NADPH:adrenodoxin oxidoreductase | 0.0012 | 0.0076 | 0.0076 |
Trypanosoma cruzi | UEV domain/Zinc finger, C3HC4 type (RING finger), putative | 0.0012 | 0.0071 | 0.0178 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 25 nM | Inhibitory activity against VEGF stimulated autophosphorylation of VEGFR2 expressed in KDR15 cells | ChEMBL. | 16302797 |
IC50 (binding) | = 240.9 nM | Inhibition of poly(Glu4-Tyr)peptide phosphorylation by recombinant VEGFR2 at 10 uM ATP | ChEMBL. | 16302797 |
IC50 (binding) | = 436.3 nM | Inhibition of poly(Glu4-Tyr)peptide phosphorylation by recombinant VEGFR2 at 1 mm ATP | ChEMBL. | 16302797 |
IC50 (binding) | = 558.6 nM | Inhibition of poly(Glu4-Tyr)peptide phosphorylation by recombinant VEGFR2 at 10 uM ATP and in presence of 100 uM glutathione | ChEMBL. | 16302797 |
IC50 (binding) | > 1000 nM | Inhibition of poly(Glu4-Tyr)peptide phosphorylation by recombinant VEGFR2 at 10 uM ATP and in presence of 5% mouse plasma | ChEMBL. | 16302797 |
T1/2 (ADMET) | = 68 hr | Half life at 1uM in the presence of 100 uM reduced glutathione in H2O-Acetonitrile (1:1) | ChEMBL. | 16302797 |
T1/2 (ADMET) | = 80 hr | Half life at 10uM in the presence of 100 uM reduced glutathione in H2O-Acetonitrile (1:1) | ChEMBL. | 16302797 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.