Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | lipoxygenase | 0.0083 | 0.3777 | 0.2611 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0132 | 0.7288 | 0.7093 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0052 | 0.1578 | 0.2166 |
Echinococcus multilocularis | tubulin gamma 1 chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | aldehyde dehydrogenase, mitochondrial precursor | 0.0062 | 0.2344 | 0.2569 |
Loa Loa (eye worm) | glutathione reductase | 0.0038 | 0.0635 | 0.0871 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0052 | 0.1578 | 0.2166 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Trypanosoma brucei | tubulin gamma chain | 0.0052 | 0.1578 | 0.2166 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.0089 | 0.4254 | 0.5837 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0052 | 0.1578 | 0.1418 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0052 | 0.1578 | 0.2166 |
Giardia lamblia | Beta tubulin | 0.0132 | 0.7288 | 1 |
Mycobacterium tuberculosis | Probable membrane NADH dehydrogenase NdhA | 0.0087 | 0.4083 | 0.8342 |
Echinococcus multilocularis | arachidonate 5 lipoxygenase | 0.0118 | 0.6288 | 0.6021 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0132 | 0.7288 | 0.7093 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0052 | 0.1578 | 0.0973 |
Loa Loa (eye worm) | alpha-tubulin | 0.0052 | 0.1578 | 0.2166 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Trypanosoma brucei | beta tubulin | 0.0132 | 0.7288 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0052 | 0.1578 | 0.1418 |
Trypanosoma cruzi | cytochrome P450, putative | 0.0089 | 0.4254 | 0.544 |
Loa Loa (eye worm) | hypothetical protein | 0.0064 | 0.2438 | 0.3345 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0132 | 0.7288 | 1 |
Mycobacterium tuberculosis | Probable nitrite reductase [NAD(P)H] large subunit [FAD flavoprotein] NirB | 0.0087 | 0.4083 | 0.8342 |
Trypanosoma brucei | beta tubulin | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | beta tubulin | 0.0132 | 0.7288 | 0.7093 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0132 | 0.7288 | 0.7093 |
Mycobacterium tuberculosis | Dihydrolipoamide dehydrogenase LpdC (lipoamide reductase (NADH)) (lipoyl dehydrogenase) (dihydrolipoyl dehydrogenase) (diaphoras | 0.0097 | 0.4768 | 1 |
Mycobacterium tuberculosis | Putative ferredoxin reductase | 0.0087 | 0.4083 | 0.8342 |
Mycobacterium ulcerans | cytochrome P450 185A4 Cyp185A4 | 0.0089 | 0.4254 | 1 |
Toxoplasma gondii | beta tubulin | 0.0132 | 0.7288 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0132 | 0.7288 | 1 |
Brugia malayi | glutathione reductase | 0.0038 | 0.0635 | 0.0871 |
Schistosoma mansoni | tubulin subunit beta | 0.0132 | 0.7288 | 0.678 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0052 | 0.1578 | 0.1418 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0132 | 0.7288 | 1 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0052 | 0.1578 | 0.1418 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0052 | 0.1578 | 0.0973 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0052 | 0.1578 | 0.1418 |
Plasmodium vivax | tubulin beta chain, putative | 0.0132 | 0.7288 | 1 |
Loa Loa (eye worm) | CYP4Cod1 | 0.0089 | 0.4254 | 0.5837 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus multilocularis | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0052 | 0.1578 | 0.0973 |
Loa Loa (eye worm) | BEN-1 protein | 0.0132 | 0.7288 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Trypanosoma brucei | alpha tubulin | 0.0052 | 0.1578 | 0.2166 |
Echinococcus granulosus | tubulin subunit TubB | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | tubulin subunit beta | 0.0132 | 0.7288 | 0.7093 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0052 | 0.1578 | 0.0973 |
Brugia malayi | Thioredoxin reductase | 0.0038 | 0.0635 | 0.0871 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Trypanosoma cruzi | tubulin gamma chain | 0.0052 | 0.1578 | 0.1418 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0052 | 0.1578 | 0.1418 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0132 | 0.7288 | 0.7093 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0052 | 0.1578 | 0.2166 |
Schistosoma mansoni | aldehyde dehydrogenase | 0.0062 | 0.2344 | 0.0909 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0052 | 0.1578 | 0.0973 |
Mycobacterium leprae | DIHYDROLIPOAMIDE DEHYDROGENASE LPD (LIPOAMIDE REDUCTASE (NADH)) (LIPOYL DEHYDROGENASE) (DIHYDROLIPOYL DEHYDROGENASE) (DIAPHORASE | 0.0097 | 0.4768 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0132 | 0.7288 | 0.7093 |
Schistosoma mansoni | tubulin subunit beta | 0.0132 | 0.7288 | 0.678 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0052 | 0.1578 | 0.0973 |
Trypanosoma brucei | trypanothione reductase | 0.0038 | 0.0635 | 0.0871 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0132 | 0.7288 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0132 | 0.7288 | 1 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0052 | 0.1578 | 0.2166 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Brugia malayi | Cytochrome P450 family protein | 0.0089 | 0.4254 | 0.5837 |
Trypanosoma brucei | epsilon tubulin | 0.0052 | 0.1578 | 0.2166 |
Schistosoma mansoni | hypothetical protein | 0.0171 | 1 | 1 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0052 | 0.1578 | 0.1418 |
Mycobacterium tuberculosis | Probable dehydrogenase | 0.0087 | 0.4083 | 0.8342 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Plasmodium vivax | tubulin epsilon chain, putative | 0.0052 | 0.1578 | 0.1418 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | tubulin alpha | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Leishmania major | epsilon tubulin, putative | 0.0052 | 0.1578 | 0.1418 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Echinococcus granulosus | arachidonate 5 lipoxygenase | 0.0118 | 0.6288 | 0.6021 |
Brugia malayi | Cytochrome P450 family protein | 0.0089 | 0.4254 | 0.5837 |
Trypanosoma cruzi | beta tubulin, putative | 0.0132 | 0.7288 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0052 | 0.1578 | 0.2166 |
Echinococcus granulosus | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Brugia malayi | Tubulin beta-1 chain | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | alpha tubulin | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | beta tubulin | 0.0132 | 0.7288 | 0.7093 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0052 | 0.1578 | 0.0973 |
Entamoeba histolytica | tubulin family protein | 0.0132 | 0.7288 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.0052 | 0.1578 | 0.2166 |
Toxoplasma gondii | aldehyde dehydrogenase | 0.0062 | 0.2344 | 0.2569 |
Echinococcus multilocularis | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Loa Loa (eye worm) | thioredoxin reductase | 0.0038 | 0.0635 | 0.0871 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0052 | 0.1578 | 0.2166 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0052 | 0.1578 | 0.2166 |
Loa Loa (eye worm) | alpha-tubulin | 0.0052 | 0.1578 | 0.2166 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0052 | 0.1578 | 0.2166 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus multilocularis | aldehyde dehydrogenase, mitochondrial | 0.0062 | 0.2344 | 0.1793 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0132 | 0.7288 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0132 | 0.7288 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Schistosoma mansoni | hypothetical protein | 0.0171 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0052 | 0.1578 | 0.0973 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0052 | 0.1578 | 0.1418 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0052 | 0.1578 | 0.2166 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0052 | 0.1578 | 0.0973 |
Schistosoma mansoni | tubulin subunit beta | 0.0132 | 0.7288 | 0.678 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0052 | 0.1578 | 0.0973 |
Mycobacterium tuberculosis | Probable reductase | 0.0087 | 0.4083 | 0.8342 |
Loa Loa (eye worm) | cytochrome P450 family protein | 0.0089 | 0.4254 | 0.5837 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Leishmania major | gamma-tubulin | 0.0052 | 0.1578 | 0.1418 |
Giardia lamblia | Beta tubulin | 0.0132 | 0.7288 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0052 | 0.1578 | 0.2166 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0052 | 0.1578 | 0.2166 |
Trypanosoma brucei | alpha tubulin | 0.0052 | 0.1578 | 0.2166 |
Plasmodium falciparum | tubulin gamma chain | 0.0052 | 0.1578 | 0.1418 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0052 | 0.1578 | 0.2166 |
Echinococcus multilocularis | beta tubulin | 0.0132 | 0.7288 | 0.7093 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0052 | 0.1578 | 0.2166 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0052 | 0.1578 | 0.2166 |
Trypanosoma brucei | beta tubulin | 0.0052 | 0.1578 | 0.2166 |
Schistosoma mansoni | lipoxygenase | 0.0118 | 0.6288 | 0.5593 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0052 | 0.1578 | 0.2166 |
Echinococcus granulosus | aldehyde dehydrogenase mitochondrial | 0.0062 | 0.2344 | 0.1793 |
Schistosoma mansoni | tubulin subunit beta | 0.0132 | 0.7288 | 0.678 |
Toxoplasma gondii | tubulin/FtsZ family, GTPase domain-containing protein | 0.0052 | 0.1578 | 0.1418 |
Loa Loa (eye worm) | BEN-1 protein | 0.0132 | 0.7288 | 1 |
Brugia malayi | Tubulin alpha-2 chain | 0.0052 | 0.1578 | 0.2166 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0052 | 0.1578 | 0.0973 |
Giardia lamblia | Beta tubulin | 0.0132 | 0.7288 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0132 | 0.7288 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0132 | 0.7288 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0052 | 0.1578 | 0.2166 |
Plasmodium falciparum | tubulin epsilon chain, putative | 0.0052 | 0.1578 | 0.1418 |
Loa Loa (eye worm) | hypothetical protein | 0.0052 | 0.1578 | 0.2166 |
Echinococcus multilocularis | tubulin epsilon chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Mycobacterium tuberculosis | NAD(P)H quinone reductase LpdA | 0.0097 | 0.4768 | 1 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Mycobacterium tuberculosis | Probable oxidoreductase | 0.0097 | 0.4768 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0052 | 0.1578 | 0.2166 |
Brugia malayi | Tubulin gamma chain | 0.0052 | 0.1578 | 0.2166 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0052 | 0.1578 | 0.1418 |
Brugia malayi | Tubulin alpha-2 chain | 0.0052 | 0.1578 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0132 | 0.7288 | 0.678 |
Echinococcus granulosus | tubulin epsilon chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Echinococcus multilocularis | geminin | 0.0171 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0052 | 0.1578 | 0.2166 |
Brugia malayi | tubulin alpha-2 chain | 0.0052 | 0.1578 | 0.2166 |
Trypanosoma brucei | beta tubulin | 0.0132 | 0.7288 | 1 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0132 | 0.7288 | 0.7093 |
Mycobacterium tuberculosis | Probable aldehyde dehydrogenase | 0.0062 | 0.2344 | 0.4135 |
Trypanosoma cruzi | cytochrome P450, putative | 0.0089 | 0.4254 | 0.544 |
Schistosoma mansoni | tubulin subunit beta | 0.0132 | 0.7288 | 0.678 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0132 | 0.7288 | 1 |
Leishmania major | beta tubulin | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Schistosoma mansoni | aldehyde dehydrogenase | 0.0062 | 0.2344 | 0.0909 |
Brugia malayi | Tubulin alpha chain | 0.0052 | 0.1578 | 0.2166 |
Loa Loa (eye worm) | beta-tubulin | 0.0132 | 0.7288 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0132 | 0.7288 | 0.7093 |
Brugia malayi | alpha-tubulin | 0.0052 | 0.1578 | 0.2166 |
Plasmodium vivax | tubulin gamma chain, putative | 0.0052 | 0.1578 | 0.1418 |
Trypanosoma brucei | beta tubulin | 0.0132 | 0.7288 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0132 | 0.7288 | 1 |
Onchocerca volvulus | 0.0029 | 0 | 0.5 | |
Echinococcus granulosus | tubulin gamma 1 chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus multilocularis | tubulin alpha | 0.0052 | 0.1578 | 0.0973 |
Toxoplasma gondii | beta-tubulin, putative | 0.0132 | 0.7288 | 1 |
Trypanosoma brucei | cytochrome P450, putative | 0.0089 | 0.4254 | 0.5837 |
Plasmodium falciparum | tubulin beta chain | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0132 | 0.7288 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0052 | 0.1578 | 0.2166 |
Echinococcus multilocularis | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | cytochrome p450-like protein | 0.0089 | 0.4254 | 0.544 |
Mycobacterium tuberculosis | Probable NADH dehydrogenase Ndh | 0.0087 | 0.4083 | 0.8342 |
Entamoeba histolytica | tubulin family protein | 0.0132 | 0.7288 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0052 | 0.1578 | 0.0973 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0052 | 0.1578 | 0.0973 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Leishmania major | alpha tubulin | 0.0052 | 0.1578 | 0.1418 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
K bind (binding) | = 0.0000001 M | Vasopressin V2 receptor binding affinity measured by competition with tritiated LVP lysine vasopressin in pig renal medullary preparation | ChEMBL. | 2965243 |
Ki (binding) | = 0.00000001 M | Inhibition of LVP-sensitive adenylate cyclase in a pig renal medullary preparation | ChEMBL. | 2965243 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.