Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.538 | 0.6387 | 0.9576 |
Trichomonas vaginalis | 3-phosphoinositide dependent protein kinase-1, putative | 0.0288 | 0.0133 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.037 | 0.0233 | 0.0263 |
Entamoeba histolytica | protein kinase, putative | 0.2774 | 0.3185 | 0.3145 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.2774 | 0.3185 | 0.4731 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.037 | 0.0233 | 0.0263 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Echinococcus granulosus | tyrosine protein kinase Src64B | 0.037 | 0.0233 | 0.0263 |
Echinococcus multilocularis | serine threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.2774 | 0.3185 | 0.3185 |
Loa Loa (eye worm) | hypothetical protein | 0.027 | 0.0111 | 0.0111 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.2774 | 0.3185 | 0.3185 |
Brugia malayi | Protein kinase domain containing protein | 0.2774 | 0.3185 | 0.3145 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Trypanosoma brucei | protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Schistosoma mansoni | tyrosine kinase | 0.037 | 0.0233 | 0.0263 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.037 | 0.0233 | 0.0263 |
Loa Loa (eye worm) | variant SH3 domain-containing protein | 0.027 | 0.0111 | 0.0111 |
Entamoeba histolytica | protein kinase, putative | 0.8322 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | uncoordinated protein 104 | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | tyrosine protein kinase HCK | 0.0287 | 0.0131 | 0.0109 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Brugia malayi | Tyrosine-protein kinase abl-1 | 0.0263 | 0.0102 | 0.0043 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.532 | 0.6313 | 0.9465 |
Leishmania major | folate/biopterin transporter, putative | 0.0288 | 0.0133 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.538 | 0.6387 | 0.9576 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0288 | 0.0133 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.2774 | 0.3185 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.5608 | 0.6667 | 1 |
Plasmodium falciparum | calcium-dependent protein kinase 7 | 0.0288 | 0.0133 | 0.0116 |
Entamoeba histolytica | hypothetical protein | 0.0288 | 0.0133 | 0.0074 |
Trypanosoma brucei | serine/threonine-protein kinase NRKB, putative | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | syntrophin-1 | 0.0228 | 0.0059 | 0.0059 |
Onchocerca volvulus | outspread protein homolog | 0.0228 | 0.0059 | 0.5 |
Loa Loa (eye worm) | SRC-1 | 0.037 | 0.0233 | 0.0233 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0288 | 0.0133 | 0.0111 |
Entamoeba histolytica | protein kinase 2, putative | 0.538 | 0.6387 | 0.6365 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.532 | 0.6313 | 0.9465 |
Echinococcus granulosus | protein kinase c iota type | 0.2774 | 0.3185 | 0.4731 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.2774 | 0.3185 | 0.4731 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0288 | 0.0133 | 0.0111 |
Brugia malayi | protein kinase C II. | 0.2774 | 0.3185 | 0.3145 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0317 | 0.0168 | 0.0165 |
Trypanosoma cruzi | serine/threonine protein kinase, putative | 0.0288 | 0.0133 | 0.0111 |
Entamoeba histolytica | protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Toxoplasma gondii | calcium dependent protein kinase CDPK7 | 0.0288 | 0.0133 | 0.0076 |
Echinococcus granulosus | tyrosine protein kinase Lyn | 0.0429 | 0.0306 | 0.0374 |
Loa Loa (eye worm) | rho-GTPase-activating | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | arf GAP with SH3 domain, ANK repeat and PH | 0.0269 | 0.0109 | 0.0076 |
Entamoeba histolytica | protein kinase, putative | 0.8094 | 0.972 | 0.9718 |
Loa Loa (eye worm) | Plekhf2 protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.532 | 0.6313 | 0.9465 |
Trypanosoma cruzi | serine/threonine-protein kinase NRKB, putative | 0.0288 | 0.0133 | 0.0111 |
Echinococcus multilocularis | tyrosine protein kinase lyn tyrosine protein kinase blk | 0.037 | 0.0233 | 0.0263 |
Echinococcus granulosus | tyrosine kinase|tyrosine protein kinase Fyn | 0.0329 | 0.0182 | 0.0187 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.0288 | 0.0133 | 1 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.037 | 0.0233 | 0.0263 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.2774 | 0.3185 | 0.4731 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.0288 | 0.0133 | 1 |
Echinococcus granulosus | protein kinase C gamma type | 0.2774 | 0.3185 | 0.4731 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus granulosus | tyrosine protein kinase ABL1 | 0.0494 | 0.0386 | 0.0494 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.037 | 0.0233 | 0.0263 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Entamoeba histolytica | hypothetical protein | 0.0288 | 0.0133 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Brugia malayi | Variant SH3 domain containing protein | 0.027 | 0.0111 | 0.0052 |
Onchocerca volvulus | Putative zinc finger protein | 0.0228 | 0.0059 | 0.5 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.532 | 0.6313 | 0.9465 |
Schistosoma mansoni | development and differentiation-enhancing factor ddef | 0.0269 | 0.0109 | 0.0076 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.2774 | 0.3185 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Trypanosoma brucei | serine/threonine-protein kinase NrkA | 0.0288 | 0.0133 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Blk | 0.0329 | 0.0182 | 0.0187 |
Trichomonas vaginalis | ribosomal protein S6 kinase, 90kD, polypeptide, putative | 0.0288 | 0.0133 | 0.0074 |
Brugia malayi | SRC-1 | 0.037 | 0.0233 | 0.0175 |
Entamoeba histolytica | protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0288 | 0.0133 | 0.0111 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | tyrosine protein kinase Fgr | 0.037 | 0.0233 | 0.0263 |
Echinococcus multilocularis | proto oncogene tyrosine protein kinase LCK | 0.037 | 0.0233 | 0.0263 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Schistosoma mansoni | tyrosine kinase | 0.0452 | 0.0334 | 0.0416 |
Echinococcus multilocularis | tyrosine protein kinase Srms | 0.0329 | 0.0182 | 0.0187 |
Echinococcus granulosus | tyrosine kinase | 0.0329 | 0.0182 | 0.0187 |
Echinococcus granulosus | proto oncogene tyrosine protein kinase LCK | 0.037 | 0.0233 | 0.0263 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.037 | 0.0233 | 0.0263 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.5608 | 0.6667 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Echinococcus granulosus | protein kinase c epsilon type | 0.2774 | 0.3185 | 0.4731 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.5608 | 0.6667 | 1 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.2774 | 0.3185 | 0.4731 |
Echinococcus multilocularis | nervana 2 | 0.532 | 0.6313 | 0.9465 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.0288 | 0.0133 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.2774 | 0.3185 | 0.3145 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Trypanosoma brucei | NEK family Serine/threonine-protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Echinococcus granulosus | arf GAP with SH3 domain ANK repeat and PH | 0.0269 | 0.0109 | 0.0076 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Toxoplasma gondii | AGC kinase | 0.8094 | 0.972 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0329 | 0.0182 | 0.0187 |
Leishmania major | protein kinase, putative | 0.0288 | 0.0133 | 1 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.8094 | 0.972 | 0.972 |
Echinococcus granulosus | serine/threonine protein kinase | 0.5608 | 0.6667 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Leishmania major | protein kinase, putative | 0.0288 | 0.0133 | 1 |
Loa Loa (eye worm) | GTP-ase activating protein for Arf containing protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.2774 | 0.3185 | 0.4731 |
Echinococcus granulosus | nervana 2 | 0.532 | 0.6313 | 0.9465 |
Brugia malayi | Hr1 repeat family protein | 0.2774 | 0.3185 | 0.3145 |
Echinococcus multilocularis | tyrosine protein kinase ABL1 | 0.0494 | 0.0386 | 0.0494 |
Entamoeba histolytica | protein kinase, putative | 0.8322 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | TK/ABL protein kinase | 0.0494 | 0.0386 | 0.0386 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.538 | 0.6387 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.2774 | 0.3185 | 0.3185 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0317 | 0.0168 | 0.0165 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.2774 | 0.3185 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.2774 | 0.3185 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Echinococcus granulosus | NDR protein kinase | 0.2774 | 0.3185 | 0.4731 |
Loa Loa (eye worm) | GTP-ase activating protein for Arf containing protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | nervana 2 | 0.532 | 0.6313 | 0.9465 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.8094 | 0.972 | 0.9718 |
Entamoeba histolytica | p21-activated kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Loa Loa (eye worm) | oxysterol binding protein | 0.0228 | 0.0059 | 0.0059 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.2774 | 0.3185 | 0.3185 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.037 | 0.0233 | 0.0263 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Trypanosoma brucei | Serine/threonine-protein kinase NEK21, putative | 0.0288 | 0.0133 | 0.0074 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.2774 | 0.3185 | 0.4731 |
Entamoeba histolytica | hypothetical protein | 0.0269 | 0.0109 | 0.0051 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Loa Loa (eye worm) | RhoGEF domain-containing protein | 0.0228 | 0.0059 | 0.0059 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.2714 | 0.3112 | 0.3071 |
Loa Loa (eye worm) | TK protein kinase | 0.0287 | 0.0131 | 0.0131 |
Echinococcus multilocularis | protein kinase c iota type | 0.2774 | 0.3185 | 0.4731 |
Loa Loa (eye worm) | hypothetical protein | 0.2774 | 0.3185 | 0.3185 |
Trichomonas vaginalis | AGC family protein kinase | 0.2774 | 0.3185 | 0.3145 |
Echinococcus granulosus | tyrosine protein kinase HCK | 0.0287 | 0.0131 | 0.0109 |
Trypanosoma cruzi | Protein kinase B | 0.5608 | 0.6667 | 1 |
Schistosoma mansoni | atypical protein kinase C | 0.2774 | 0.3185 | 0.4731 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.2774 | 0.3185 | 0.4731 |
Brugia malayi | protein-tyrosine kinase | 0.0329 | 0.0182 | 0.0124 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.538 | 0.6387 | 0.9576 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.538 | 0.6387 | 0.9576 |
Trichomonas vaginalis | AGC family protein kinase | 0.3002 | 0.3466 | 0.3427 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.2774 | 0.3185 | 0.4731 |
Onchocerca volvulus | Putative neuronal RhoA GEF protein | 0.0228 | 0.0059 | 0.5 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Echinococcus multilocularis | tyrosine protein kinase lyn lyn a protein tyrosine kinase lymphocyte specific protein tyrosine kinase | 0.037 | 0.0233 | 0.0263 |
Brugia malayi | Tyrosine-protein kinase abl-1 | 0.0272 | 0.0113 | 0.0054 |
Brugia malayi | Protein kinase domain containing protein | 0.2774 | 0.3185 | 0.3145 |
Entamoeba histolytica | protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.8322 | 1 | 1 |
Loa Loa (eye worm) | PH domain-containing protein | 0.0228 | 0.0059 | 0.0059 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2774 | 0.3185 | 0.4731 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.2774 | 0.3185 | 0.3185 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.037 | 0.0233 | 0.0263 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Trypanosoma cruzi | NEK family Serine/threonine-protein kinase, putative | 0.0288 | 0.0133 | 0.0111 |
Entamoeba histolytica | protein kinase, putative | 0.0287 | 0.0131 | 0.0072 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.0288 | 0.0133 | 0.0111 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.5608 | 0.6667 | 0.6647 |
Echinococcus granulosus | 3'partial|tyrosine protein kinase Fgr | 0.037 | 0.0233 | 0.0263 |
Loa Loa (eye worm) | TK protein kinase | 0.0329 | 0.0182 | 0.0182 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.2774 | 0.3185 | 0.3185 |
Echinococcus multilocularis | tyrosine protein kinase Src64B | 0.037 | 0.0233 | 0.0263 |
Onchocerca volvulus | Abnormal cell migration protein 10 homolog | 0.0228 | 0.0059 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Abl | 0.0263 | 0.0102 | 0.0065 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.8322 | 1 | 1 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.8322 | 1 | 1 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.538 | 0.6387 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Onchocerca volvulus | Protein melted homolog | 0.0228 | 0.0059 | 0.5 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.0288 | 0.0133 | 0.0111 |
Loa Loa (eye worm) | cytohesin 3 | 0.0228 | 0.0059 | 0.0059 |
Giardia lamblia | Kinase, AGC PKA | 0.538 | 0.6387 | 0.5 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.2774 | 0.3185 | 0.4731 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0288 | 0.0133 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Schistosoma mansoni | tyrosine kinase | 0.037 | 0.0233 | 0.0263 |
Schistosoma mansoni | serine/threonine kinase | 0.2774 | 0.3185 | 0.4731 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Schistosoma mansoni | vav2 | 0.027 | 0.0111 | 0.0078 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.2774 | 0.3185 | 0.4731 |
Echinococcus granulosus | tyrosine protein kinase Blk | 0.0329 | 0.0182 | 0.0187 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.0288 | 0.0133 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.0288 | 0.0133 | 0.0074 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.5608 | 0.6667 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0228 | 0.0059 | 0.0059 |
Onchocerca volvulus | 0.0228 | 0.0059 | 0.5 | |
Toxoplasma gondii | protein kinase domain-containing protein | 0.0288 | 0.0133 | 0.0076 |
Echinococcus granulosus | nervana 2 | 0.532 | 0.6313 | 0.9465 |
Plasmodium vivax | calcium-dependent protein kinase 7, putative | 0.0288 | 0.0133 | 0.0116 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.5608 | 0.6667 | 0.6647 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Cell viability (functional) | = 20 uM | Inhibitory concentration against BCL1 cell proliferation in WST-1 assay; Range 10-20 | ChEMBL. | 16220989 |
T1/2 (ADMET) | >> 7 day | Half-life of the conjugate when treated with 10% foetal bovine serum for enzymatic stability | ChEMBL. | 16220989 |
T1/2 (ADMET) | = 18 hr | Half-life of the conjugate when treated with 25% murine serum for enzymatic stability | ChEMBL. | 16220989 |
UTC (functional) | = 34 % | Percent inhibition of CD40 expression in BCL1 cells treated with 10 uM peptide nucleic acid (PNA)conjugate; n=3 | ChEMBL. | 16220989 |
UTC (functional) | = 65 % | Percent inhibition of CD40 expression in BCL1 cells treated with 3 uM peptide nucleic acid (PNA)conjugate; n=3 | ChEMBL. | 16220989 |
UTC (functional) | = 94 % | Percent inhibition of CD40 expression in BCL1 cells treated with 1 uM peptide nucleic acid (PNA)conjugate; n=3 | ChEMBL. | 16220989 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.